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2. Induction of Therapeutic Senescence in Vemurafenib-Resistant Melanoma by Extended Inhibition of CDK4/6. Yoshida A; Lee EK; Diehl JA Cancer Res; 2016 May; 76(10):2990-3002. PubMed ID: 26988987 [TBL] [Abstract][Full Text] [Related]
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4. An In Vivo Reporter to Quantitatively and Temporally Analyze the Effects of CDK4/6 Inhibitor-Based Therapies in Melanoma. Teh JL; Purwin TJ; Greenawalt EJ; Chervoneva I; Goldberg A; Davies MA; Aplin AE Cancer Res; 2016 Sep; 76(18):5455-66. PubMed ID: 27488531 [TBL] [Abstract][Full Text] [Related]
5. Senescence-associated secretory factors induced by cisplatin in melanoma cells promote non-senescent melanoma cell growth through activation of the ERK1/2-RSK1 pathway. Sun X; Shi B; Zheng H; Min L; Yang J; Li X; Liao X; Huang W; Zhang M; Xu S; Zhu Z; Cui H; Liu X Cell Death Dis; 2018 Feb; 9(3):260. PubMed ID: 29449532 [TBL] [Abstract][Full Text] [Related]
6. Efficacy of the combination of MEK and CDK4/6 inhibitors in vitro and in vivo in KRAS mutant colorectal cancer models. Lee MS; Helms TL; Feng N; Gay J; Chang QE; Tian F; Wu JY; Toniatti C; Heffernan TP; Powis G; Kwong LN; Kopetz S Oncotarget; 2016 Jun; 7(26):39595-39608. PubMed ID: 27167191 [TBL] [Abstract][Full Text] [Related]
8. Palbociclib-induced autophagy and senescence in gastric cancer cells. Valenzuela CA; Vargas L; Martinez V; Bravo S; Brown NE Exp Cell Res; 2017 Nov; 360(2):390-396. PubMed ID: 28947133 [TBL] [Abstract][Full Text] [Related]
9. Preclinical development of G1T38: A novel, potent and selective inhibitor of cyclin dependent kinases 4/6 for use as an oral antineoplastic in patients with CDK4/6 sensitive tumors. Bisi JE; Sorrentino JA; Jordan JL; Darr DD; Roberts PJ; Tavares FX; Strum JC Oncotarget; 2017 Jun; 8(26):42343-42358. PubMed ID: 28418845 [TBL] [Abstract][Full Text] [Related]
10. Combined Inhibition of CDK4/6 and PI3K/AKT/mTOR Pathways Induces a Synergistic Anti-Tumor Effect in Malignant Pleural Mesothelioma Cells. Bonelli MA; Digiacomo G; Fumarola C; Alfieri R; Quaini F; Falco A; Madeddu D; La Monica S; Cretella D; Ravelli A; Ulivi P; Tebaldi M; Calistri D; Delmonte A; Ampollini L; Carbognani P; Tiseo M; Cavazzoni A; Petronini PG Neoplasia; 2017 Aug; 19(8):637-648. PubMed ID: 28704762 [TBL] [Abstract][Full Text] [Related]
11. Biological specificity of CDK4/6 inhibitors: dose response relationship, in vivo signaling, and composite response signature. Knudsen ES; Hutcheson J; Vail P; Witkiewicz AK Oncotarget; 2017 Jul; 8(27):43678-43691. PubMed ID: 28620137 [TBL] [Abstract][Full Text] [Related]
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13. Pharmacological CDK4/6 inhibition reveals a p53-dependent senescent state with restricted toxicity. Wang B; Varela-Eirin M; Brandenburg SM; Hernandez-Segura A; van Vliet T; Jongbloed EM; Wilting SM; Ohtani N; Jager A; Demaria M EMBO J; 2022 Mar; 41(6):e108946. PubMed ID: 34985783 [TBL] [Abstract][Full Text] [Related]
14. Regulation of PRMT5-MDM4 axis is critical in the response to CDK4/6 inhibitors in melanoma. AbuHammad S; Cullinane C; Martin C; Bacolas Z; Ward T; Chen H; Slater A; Ardley K; Kirby L; Chan KT; Brajanovski N; Smith LK; Rao AD; Lelliott EJ; Kleinschmidt M; Vergara IA; Papenfuss AT; Lau P; Ghosh P; Haupt S; Haupt Y; Sanij E; Poortinga G; Pearson RB; Falk H; Curtis DJ; Stupple P; Devlin M; Street I; Davies MA; McArthur GA; Sheppard KE Proc Natl Acad Sci U S A; 2019 Sep; 116(36):17990-18000. PubMed ID: 31439820 [TBL] [Abstract][Full Text] [Related]
15. Combined Blockade of MEK and CDK4/6 Pathways Induces Senescence to Improve Survival in Pancreatic Ductal Adenocarcinoma. Willobee BA; Gaidarski AA; Dosch AR; Castellanos JA; Dai X; Mehra S; Messaggio F; Srinivasan S; VanSaun MN; Nagathihalli NS; Merchant NB Mol Cancer Ther; 2021 Jul; 20(7):1246-1256. PubMed ID: 34001634 [TBL] [Abstract][Full Text] [Related]
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