BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

238 related articles for article (PubMed ID: 28043795)

  • 1. Evaluation of substituted ebselen derivatives as potential trypanocidal agents.
    Gordhan HM; Patrick SL; Swasy MI; Hackler AL; Anayee M; Golden JE; Morris JC; Whitehead DC
    Bioorg Med Chem Lett; 2017 Feb; 27(3):537-541. PubMed ID: 28043795
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis of 5-enamine-4-thiazolidinone derivatives with trypanocidal and anticancer activity.
    Holota S; Kryshchyshyn A; Derkach H; Trufin Y; Demchuk I; Gzella A; Grellier P; Lesyk R
    Bioorg Chem; 2019 May; 86():126-136. PubMed ID: 30690336
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis of oxysterols and nitrogenous sterols with antileishmanial and trypanocidal activities.
    Bazin MA; Loiseau PM; Bories C; Letourneux Y; Rault S; El Kihel L
    Eur J Med Chem; 2006 Oct; 41(10):1109-16. PubMed ID: 16949702
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Inhibition of trypanosome alternative oxidase without its N-terminal mitochondrial targeting signal (ΔMTS-TAO) by cationic and non-cationic 4-hydroxybenzoate and 4-alkoxybenzaldehyde derivatives active against T. brucei and T. congolense.
    Ebiloma GU; Ayuga TD; Balogun EO; Gil LA; Donachie A; Kaiser M; Herraiz T; Inaoka DK; Shiba T; Harada S; Kita K; de Koning HP; Dardonville C
    Eur J Med Chem; 2018 Apr; 150():385-402. PubMed ID: 29544150
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and in vitro antikinetoplastid activity of polyamine-hydroxybenzotriazole conjugates.
    Jagu E; Pomel S; Diez-Martinez A; Ramiandrasoa F; Krauth-Siegel RL; Pethe S; Blonski C; Labruère R; Loiseau PM
    Bioorg Med Chem; 2017 Jan; 25(1):84-90. PubMed ID: 27793448
    [TBL] [Abstract][Full Text] [Related]  

  • 6. In vitro activity of salinomycin and monensin derivatives against Trypanosoma brucei.
    Steverding D; Antoszczak M; Huczyński A
    Parasit Vectors; 2016 Jul; 9(1):409. PubMed ID: 27457761
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and in vitro antitrypanosomal evaluation of novel 6-heteroarylidene-substituted quinolone derivatives.
    Angula KT; Legoabe LJ; Swart T; Hoppe HC; Beteck RM
    Eur J Med Chem; 2022 Jan; 227():113913. PubMed ID: 34656043
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and in vitro evaluation of tropane halogenated-derivatives against malaria, sleeping sickness, Chagas disease and leishmaniasis.
    Cretton S; Bartholomeusz TA; Mehl F; Allenbach Y; Matheeussen A; Cos P; Maes L; Christen P
    Med Chem; 2014; 10(8):753-8. PubMed ID: 24813684
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Antitrypanosomal structure-activity-relationship study of synthetic cynaropicrin derivatives.
    Usuki T; Sato M; Hara S; Yoshimoto Y; Kondo R; Zimmermann S; Kaiser M; Brun R; Hamburger M; Adams M
    Bioorg Med Chem Lett; 2014 Feb; 24(3):794-8. PubMed ID: 24433861
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Promising lead compounds for novel antiprotozoals.
    Otoguro K; Iwatsuki M; Ishiyama A; Namatame M; Nishihara-Tukashima A; Shibahara S; Kondo S; Yamada H; Omura S
    J Antibiot (Tokyo); 2010 Jul; 63(7):381-4. PubMed ID: 20661239
    [No Abstract]   [Full Text] [Related]  

  • 11. 9- and 11-Substituted 4-azapaullones are potent and selective inhibitors of African trypanosoma.
    Maiwald F; Benítez D; Charquero D; Dar MA; Erdmann H; Preu L; Koch O; Hölscher C; Loaëc N; Meijer L; Comini MA; Kunick C
    Eur J Med Chem; 2014 Aug; 83():274-83. PubMed ID: 24973661
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Mallotojaponins B and C: Total Synthesis, Antiparasitic Evaluation, and Preliminary SAR Studies.
    Grayfer TD; Grellier P; Mouray E; Dodd RH; Dubois J; Cariou K
    Org Lett; 2016 Feb; 18(4):708-11. PubMed ID: 26828239
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and tripanocidal activity of ferrocenyl and benzyl diamines against Trypanosoma brucei and Trypanosoma cruzi.
    Velásquez AM; Francisco AI; Kohatsu AA; Silva FA; Rodrigues DF; Teixeira RG; Chiari BG; de Almeida MG; Isaac VL; Vargas MD; Cicarelli RM
    Bioorg Med Chem Lett; 2014 Apr; 24(7):1707-10. PubMed ID: 24630563
    [TBL] [Abstract][Full Text] [Related]  

  • 14. C6-O-alkylated 7-deazainosine nucleoside analogues: Discovery of potent and selective anti-sleeping sickness agents.
    Hulpia F; Bouton J; Campagnaro GD; Alfayez IA; Mabille D; Maes L; de Koning HP; Caljon G; Van Calenbergh S
    Eur J Med Chem; 2020 Feb; 188():112018. PubMed ID: 31931339
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of novel guttiferone A derivatives: in-vitro evaluation toward Plasmodium falciparum, Trypanosoma brucei and Leishmania donovani.
    Fromentin Y; Gaboriaud-Kolar N; Lenta BN; Wansi JD; Buisson D; Mouray E; Grellier P; Loiseau PM; Lallemand MC; Michel S
    Eur J Med Chem; 2013 Jul; 65():284-94. PubMed ID: 23727538
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Anti-trypanosomal activity of doubly modified salinomycin derivatives.
    Antoszczak M; Steverding D; Sulik M; Janczak J; Huczyński A
    Eur J Med Chem; 2019 Jul; 173():90-98. PubMed ID: 30986574
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Discovery of halo-nitrobenzamides with potential application against human African trypanosomiasis.
    Hwang JY; Smithson D; Connelly M; Maier J; Zhu F; Guy KR
    Bioorg Med Chem Lett; 2010 Jan; 20(1):149-52. PubMed ID: 19963377
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals.
    Veerman J; van den Bergh T; Orrling KM; Jansen C; Cos P; Maes L; Chatelain E; Ioset JR; Edink EE; Tenor H; Seebeck T; de Esch I; Leurs R; Sterk GJ
    Bioorg Med Chem; 2016 Apr; 24(7):1573-81. PubMed ID: 26935942
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and in vitro antiprotozoal activities of water-soluble, inexpensive 3,7-bis(dialkylamino)phenoxazin-5-ium derivatives.
    Ge JF; Arai C; Kaiser M; Wittlin S; Brun R; Ihara M
    J Med Chem; 2008 Jun; 51(12):3654-8. PubMed ID: 18476684
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Novel pyrrolobenzoxaboroles: design, synthesis, and biological evaluation against Trypanosoma brucei.
    Wu P; Zhang J; Meng Q; Nare B; Jacobs RT; Zhou H
    Eur J Med Chem; 2014 Jun; 81():59-75. PubMed ID: 24826816
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 12.