These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

171 related articles for article (PubMed ID: 28067769)

  • 1. Identification of a Potent Allosteric Inhibitor of Human Protein Kinase CK2 by Bacterial Surface Display Library Screening.
    Nienberg C; Garmann C; Gratz A; Bollacke A; Götz C; Jose J
    Pharmaceuticals (Basel); 2017 Jan; 10(1):. PubMed ID: 28067769
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Toward selective CK2alpha and CK2alpha' inhibitors: Development of a novel whole-cell kinase assay by Autodisplay of catalytic CK2alpha'.
    Bollacke A; Nienberg C; Borgne ML; Jose J
    J Pharm Biomed Anal; 2016 Mar; 121():253-260. PubMed ID: 26786382
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Functional display of heterotetrameric human protein kinase CK2 on Escherichia coli: a novel tool for drug discovery.
    Gratz A; Bollacke A; Stephan S; Nienberg C; Le Borgne M; Götz C; Jose J
    Microb Cell Fact; 2015 Jun; 14():74. PubMed ID: 26036951
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Site-Specific Labeling of Protein Kinase CK2: Combining Surface Display and Click Chemistry for Drug Discovery Applications.
    Nienberg C; Retterath A; Becher KS; Saenger T; Mootz HD; Jose J
    Pharmaceuticals (Basel); 2016 Jun; 9(3):. PubMed ID: 27355959
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Unexpected CK2β-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2.
    Pietsch M; Viht K; Schnitzler A; Ekambaram R; Steinkrüger M; Enkvist E; Nienberg C; Nickelsen A; Lauwers M; Jose J; Uri A; Niefind K
    Bioorg Chem; 2020 Mar; 96():103608. PubMed ID: 32058103
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Identification and Biological Evaluation of CK2 Allosteric Fragments through Structure-Based Virtual Screening.
    Li C; Zhang X; Zhang N; Zhou Y; Sun G; Zhao L; Zhong R
    Molecules; 2020 Jan; 25(1):. PubMed ID: 31935979
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Development of a high-throughput screening-compatible assay to identify inhibitors of the CK2α/CK2β interaction.
    Hochscherf J; Lindenblatt D; Steinkrüger M; Yoo E; Ulucan Ö; Herzig S; Issinger OG; Helms V; Götz C; Neundorf I; Niefind K; Pietsch M
    Anal Biochem; 2015 Jan; 468():4-14. PubMed ID: 25233003
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Crystal structure of a C-terminal deletion mutant of human protein kinase CK2 catalytic subunit.
    Ermakova I; Boldyreff B; Issinger OG; Niefind K
    J Mol Biol; 2003 Jul; 330(5):925-34. PubMed ID: 12860116
    [TBL] [Abstract][Full Text] [Related]  

  • 9. First structure of protein kinase CK2 catalytic subunit with an effective CK2β-competitive ligand.
    Raaf J; Guerra B; Neundorf I; Bopp B; Issinger OG; Jose J; Pietsch M; Niefind K
    ACS Chem Biol; 2013 May; 8(5):901-7. PubMed ID: 23474121
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Discovery of a CK2α'-Biased ATP-Competitive Inhibitor from a High-Throughput Screen of an Allosteric-Inhibitor-Like Compound Library.
    Mudaliar D; Mansky RH; White A; Baudhuin G; Hawkinson J; Wong H; Walters MA; Gomez-Pastor R
    ACS Chem Neurosci; 2024 Aug; 15(15):2703-2718. PubMed ID: 38908003
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α'.
    Hochscherf J; Lindenblatt D; Witulski B; Birus R; Aichele D; Marminon C; Bouaziz Z; Le Borgne M; Jose J; Niefind K
    Pharmaceuticals (Basel); 2017 Dec; 10(4):. PubMed ID: 29236079
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Structure-based Discovery of Novel CK2α-Binding Cyclic Peptides with Anti-cancer Activity.
    Tang S; Zhang N; Zhou Y; Cortopassi WA; Jacobson MP; Zhao LJ; Zhong RG
    Mol Inform; 2019 Mar; 38(3):e1800089. PubMed ID: 30307134
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Identification of CK2α' selective inhibitors by the screening of an allosteric-kinase-inhibitor-like compound library.
    Mudaliar D; Mansky RH; White A; Baudhuin G; Hawkinson J; Wong H; Walters MA; Gomez-Pastor R
    bioRxiv; 2024 Jan; ():. PubMed ID: 38328231
    [TBL] [Abstract][Full Text] [Related]  

  • 14. First inactive conformation of CK2 alpha, the catalytic subunit of protein kinase CK2.
    Raaf J; Issinger OG; Niefind K
    J Mol Biol; 2009 Mar; 386(5):1212-21. PubMed ID: 19361447
    [TBL] [Abstract][Full Text] [Related]  

  • 15. The interaction of CK2alpha and CK2beta, the subunits of protein kinase CK2, requires CK2beta in a preformed conformation and is enthalpically driven.
    Raaf J; Brunstein E; Issinger OG; Niefind K
    Protein Sci; 2008 Dec; 17(12):2180-6. PubMed ID: 18824508
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Eukaryotic translation-initiation factor eIF2beta binds to protein kinase CK2: effects on CK2alpha activity.
    Llorens F; Roher N; Miró FA; Sarno S; Ruiz FX; Meggio F; Plana M; Pinna LA; Itarte E
    Biochem J; 2003 Nov; 375(Pt 3):623-31. PubMed ID: 12901717
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis and SAR of Tetracyclic Inhibitors of Protein Kinase CK2 Derived from Furocarbazole W16.
    Kröger L; Daniliuc CG; Ensan D; Borgert S; Nienberg C; Lauwers M; Steinkrüger M; Jose J; Pietsch M; Wünsch B
    ChemMedChem; 2020 May; 15(10):871-881. PubMed ID: 32168422
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Primary and secondary interactions between CK2alpha and CK2beta lead to ring-like structures in the crystals of the CK2 holoenzyme.
    Niefind K; Issinger OG
    Mol Cell Biochem; 2005 Jun; 274(1-2):3-14. PubMed ID: 16335523
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Structure-based design of small peptide inhibitors of protein kinase CK2 subunit interaction.
    Laudet B; Barette C; Dulery V; Renaudet O; Dumy P; Metz A; Prudent R; Deshiere A; Dideberg O; Filhol O; Cochet C
    Biochem J; 2007 Dec; 408(3):363-73. PubMed ID: 17714077
    [TBL] [Abstract][Full Text] [Related]  

  • 20. The activity of CK2 in the extracts of COS-7 cells transfected with wild type and mutant subunits of protein kinase CK2.
    Korn I; Jacob G; Allende CC; Allende JE
    Mol Cell Biochem; 2001 Nov; 227(1-2):37-44. PubMed ID: 11827173
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.