BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

34 related articles for article (PubMed ID: 28076825)

  • 1. Spirocyclic Motifs in Natural Products.
    Chupakhin E; Babich O; Prosekov A; Asyakina L; Krasavin M
    Molecules; 2019 Nov; 24(22):. PubMed ID: 31744211
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Structure-Activity Relationship Studies and Optimization of 4-Hydroxypyridones as GPR84 Agonists.
    Ieremias L; Kaspersen MH; Manandhar A; Schultz-Knudsen K; Vrettou CI; Pokhrel R; Heidtmann CV; Jenkins L; Kanellou C; Marsango S; Li Y; Bräuner-Osborne H; Rexen Ulven E; Milligan G; Ulven T
    J Med Chem; 2024 Mar; 67(5):3542-3570. PubMed ID: 38381650
    [TBL] [Abstract][Full Text] [Related]  

  • 3. The development of diphenyleneiodonium analogs as GPR3 agonists.
    Gay EA; Harris DL; Wilson JW; Blough BE
    Bioorg Med Chem Lett; 2023 Oct; 94():129427. PubMed ID: 37541631
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Structure-Activity Relationship Studies of Tetrahydroquinolone Free Fatty Acid Receptor 3 Modulators.
    Ulven ER; Quon T; Sergeev E; Barki N; Brvar M; Hudson BD; Dutta P; Hansen AH; Bielefeldt LØ; Tobin AB; McKenzie CJ; Milligan G; Ulven T
    J Med Chem; 2020 Apr; 63(7):3577-3595. PubMed ID: 32141297
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Exploration of Spirocyclic Derivatives of Ciprofloxacin as Antibacterial Agents.
    Lukin A; Chudinov M; Vedekhina T; Rogacheva E; Kraeva L; Bakulina O; Krasavin M
    Molecules; 2022 Jul; 27(15):. PubMed ID: 35956812
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Recent developments in the discovery of FFA1 receptor agonists as novel oral treatment for type 2 diabetes mellitus.
    Defossa E; Wagner M
    Bioorg Med Chem Lett; 2014 Jul; 24(14):2991-3000. PubMed ID: 24881568
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Free fatty acid receptor 1 (GPR40) agonists containing spirocyclic periphery inspired by LY2881835.
    Krasavin M; Lukin A; Bagnyukova D; Zhurilo N; Zahanich I; Zozulya S; Ihalainen J; Forsberg MM; Lehtonen M; Rautio J; Moore D; Tikhonova IG
    Bioorg Med Chem; 2016 Nov; 24(21):5481-5494. PubMed ID: 27647366
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Novel FFA1 (GPR40) agonists containing spirocyclic periphery: polar azine periphery as a driver of potency.
    Krasavin M; Lukin A; Bagnyukova D; Zhurilo N; Zahanich I; Zozulya S
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):29-36. PubMed ID: 27781494
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design, synthesis and structure-activity relationship studies of GPR40 agonists containing amide linker.
    Chen T; Ning M; Ye Y; Wang K; Leng Y; Shen J
    Eur J Med Chem; 2018 May; 152():175-194. PubMed ID: 29705709
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis and Structure-activity relationship studies of new thiazole-based free fatty acid receptor 1 agonists for the treatment of type 2 diabetes.
    Li Z; Qiu Q; Xu X; Wang X; Jiao L; Su X; Pan M; Huang W; Qian H
    Eur J Med Chem; 2016 May; 113():246-57. PubMed ID: 26945112
    [TBL] [Abstract][Full Text] [Related]  

  • 11. The Discovery, Preclinical, and Early Clinical Development of Potent and Selective GPR40 Agonists for the Treatment of Type 2 Diabetes Mellitus (LY2881835, LY2922083, and LY2922470).
    Hamdouchi C; Kahl SD; Patel Lewis A; Cardona GR; Zink RW; Chen K; Eessalu TE; Ficorilli JV; Marcelo MC; Otto KA; Wilbur KL; Lineswala JP; Piper JL; Coffey DS; Sweetana SA; Haas JV; Brooks DA; Pratt EJ; Belin RM; Deeg MA; Ma X; Cannady EA; Johnson JT; Yumibe NP; Chen Q; Maiti P; Montrose-Rafizadeh C; Chen Y; Reifel Miller A
    J Med Chem; 2016 Dec; 59(24):10891-10916. PubMed ID: 27749056
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Polar aromatic periphery increases agonist potency of spirocyclic free fatty acid receptor (GPR40) agonists inspired by LY2881835.
    Krasavin M; Lukin A; Bagnyukova D; Zhurilo N; Golovanov A; Zozulya S; Zahanich I; Moore D; Tikhonova IG
    Eur J Med Chem; 2017 Feb; 127():357-368. PubMed ID: 28076825
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Progress in the discovery and development of small-molecule modulators of G-protein-coupled receptor 40 (GPR40/FFA1/FFAR1): an emerging target for type 2 diabetes.
    Bharate SB; Nemmani KV; Vishwakarma RA
    Expert Opin Ther Pat; 2009 Feb; 19(2):237-64. PubMed ID: 19441920
    [TBL] [Abstract][Full Text] [Related]  

  • 14.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 15.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 16.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 17.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 18.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 19.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 20.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 2.