99 related articles for article (PubMed ID: 28128956)
1. Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents.
Pieroni M; Azzali E; Basilico N; Parapini S; Zolkiewski M; Beato C; Annunziato G; Bruno A; Vacondio F; Costantino G
J Med Chem; 2017 Mar; 60(5):1959-1970. PubMed ID: 28128956
[TBL] [Abstract][Full Text] [Related]
2. Exploration of a new type of antimalarial compounds based on febrifugine.
Kikuchi H; Yamamoto K; Horoiwa S; Hirai S; Kasahara R; Hariguchi N; Matsumoto M; Oshima Y
J Med Chem; 2006 Jul; 49(15):4698-706. PubMed ID: 16854076
[TBL] [Abstract][Full Text] [Related]
3. 2,4-Diaminothienopyrimidines as orally active antimalarial agents.
González Cabrera D; Le Manach C; Douelle F; Younis Y; Feng TS; Paquet T; Nchinda AT; Street LJ; Taylor D; de Kock C; Wiesner L; Duffy S; White KL; Zabiulla KM; Sambandan Y; Bashyam S; Waterson D; Witty MJ; Charman SA; Avery VM; Wittlin S; Chibale K
J Med Chem; 2014 Feb; 57(3):1014-22. PubMed ID: 24446664
[TBL] [Abstract][Full Text] [Related]
4. An overview of benzo[b]thiophene-based medicinal chemistry.
Keri RS; Chand K; Budagumpi S; Balappa Somappa S; Patil SA; Nagaraja BM
Eur J Med Chem; 2017 Sep; 138():1002-1033. PubMed ID: 28759875
[TBL] [Abstract][Full Text] [Related]
5. Indolyl-3-ethanone-α-thioethers: A promising new class of non-toxic antimalarial agents.
Svogie AL; Isaacs M; Hoppe HC; Khanye SD; Veale CG
Eur J Med Chem; 2016 May; 114():79-88. PubMed ID: 26974377
[TBL] [Abstract][Full Text] [Related]
6. In Vivo and In Vitro Optimization of Screening Antimalarial Hits toward Lead Molecules for Preclinical Development.
Fröhlich T; Tsogoeva SB
J Med Chem; 2016 Nov; 59(21):9668-9671. PubMed ID: 27775354
[TBL] [Abstract][Full Text] [Related]
7. Benzothiophene carboxamide derivatives as novel antimalarials.
Banerjee T; Kapoor N; Surolia N; Surolia A
IUBMB Life; 2011 Dec; 63(12):1111-5. PubMed ID: 22038932
[TBL] [Abstract][Full Text] [Related]
8. Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond.
Van Voorhis WC; Adams JH; Adelfio R; Ahyong V; Akabas MH; Alano P; Alday A; Alemán Resto Y; Alsibaee A; Alzualde A; Andrews KT; Avery SV; Avery VM; Ayong L; Baker M; Baker S; Ben Mamoun C; Bhatia S; Bickle Q; Bounaadja L; Bowling T; Bosch J; Boucher LE; Boyom FF; Brea J; Brennan M; Burton A; Caffrey CR; Camarda G; Carrasquilla M; Carter D; Belen Cassera M; Chih-Chien Cheng K; Chindaudomsate W; Chubb A; Colon BL; Colón-López DD; Corbett Y; Crowther GJ; Cowan N; D'Alessandro S; Le Dang N; Delves M; DeRisi JL; Du AY; Duffy S; Abd El-Salam El-Sayed S; Ferdig MT; Fernández Robledo JA; Fidock DA; Florent I; Fokou PV; Galstian A; Gamo FJ; Gokool S; Gold B; Golub T; Goldgof GM; Guha R; Guiguemde WA; Gural N; Guy RK; Hansen MA; Hanson KK; Hemphill A; Hooft van Huijsduijnen R; Horii T; Horrocks P; Hughes TB; Huston C; Igarashi I; Ingram-Sieber K; Itoe MA; Jadhav A; Naranuntarat Jensen A; Jensen LT; Jiang RH; Kaiser A; Keiser J; Ketas T; Kicka S; Kim S; Kirk K; Kumar VP; Kyle DE; Lafuente MJ; Landfear S; Lee N; Lee S; Lehane AM; Li F; Little D; Liu L; Llinás M; Loza MI; Lubar A; Lucantoni L; Lucet I; Maes L; Mancama D; Mansour NR; March S; McGowan S; Medina Vera I; Meister S; Mercer L; Mestres J; Mfopa AN; Misra RN; Moon S; Moore JP; Morais Rodrigues da Costa F; Müller J; Muriana A; Nakazawa Hewitt S; Nare B; Nathan C; Narraidoo N; Nawaratna S; Ojo KK; Ortiz D; Panic G; Papadatos G; Parapini S; Patra K; Pham N; Prats S; Plouffe DM; Poulsen SA; Pradhan A; Quevedo C; Quinn RJ; Rice CA; Abdo Rizk M; Ruecker A; St Onge R; Salgado Ferreira R; Samra J; Robinett NG; Schlecht U; Schmitt M; Silva Villela F; Silvestrini F; Sinden R; Smith DA; Soldati T; Spitzmüller A; Stamm SM; Sullivan DJ; Sullivan W; Suresh S; Suzuki BM; Suzuki Y; Swamidass SJ; Taramelli D; Tchokouaha LR; Theron A; Thomas D; Tonissen KF; Townson S; Tripathi AK; Trofimov V; Udenze KO; Ullah I; Vallieres C; Vigil E; Vinetz JM; Voong Vinh P; Vu H; Watanabe NA; Weatherby K; White PM; Wilks AF; Winzeler EA; Wojcik E; Wree M; Wu W; Yokoyama N; Zollo PH; Abla N; Blasco B; Burrows J; Laleu B; Leroy D; Spangenberg T; Wells T; Willis PA
PLoS Pathog; 2016 Jul; 12(7):e1005763. PubMed ID: 27467575
[TBL] [Abstract][Full Text] [Related]
9. Investigation into novel thiophene- and furan-based 4-amino-7-chloroquinolines afforded antimalarials that cure mice.
Opsenica IM; Verbić TŽ; Tot M; Sciotti RJ; Pybus BS; Djurković-Djaković O; Slavić K; Šolaja BA
Bioorg Med Chem; 2015 May; 23(9):2176-86. PubMed ID: 25801154
[TBL] [Abstract][Full Text] [Related]
10. Benzothiophene carboxamide derivatives as inhibitors of Plasmodium falciparum enoyl-ACP reductase.
Banerjee T; Sharma SK; Kapoor N; Dwivedi V; Surolia N; Surolia A
IUBMB Life; 2011 Dec; 63(12):1101-10. PubMed ID: 22006792
[TBL] [Abstract][Full Text] [Related]
11. Discovery and Characterization of ACT-451840: an Antimalarial Drug with a Novel Mechanism of Action.
Boss C; Aissaoui H; Amaral N; Bauer A; Bazire S; Binkert C; Brun R; Bürki C; Ciana CL; Corminboeuf O; Delahaye S; Dollinger C; Fischli C; Fischli W; Flock A; Frantz MC; Girault M; Grisostomi C; Friedli A; Heidmann B; Hinder C; Jacob G; Le Bihan A; Malrieu S; Mamzed S; Merot A; Meyer S; Peixoto S; Petit N; Siegrist R; Trollux J; Weller T; Wittlin S
ChemMedChem; 2016 Sep; 11(18):1995-2014. PubMed ID: 27471138
[TBL] [Abstract][Full Text] [Related]
12. Machine learning prioritizes synthesis of primaquine ureidoamides with high antimalarial activity and attenuated cytotoxicity.
Levatić J; Pavić K; Perković I; Uzelac L; Ester K; Kralj M; Kaiser M; Rottmann M; Supek F; Zorc B
Eur J Med Chem; 2018 Feb; 146():651-667. PubMed ID: 29407988
[TBL] [Abstract][Full Text] [Related]
13. [Thieno[3,4-c]quinoline-4-yl-amines--synthesis and investigation of activity against malaria].
Görlitzer K; Gabriel B; Jomaa H; Wiesner J
Pharmazie; 2006 Nov; 61(11):901-7. PubMed ID: 17152980
[TBL] [Abstract][Full Text] [Related]
14. Discovery of carbohybrid-based 2-aminopyrimidine analogues as a new class of rapid-acting antimalarial agents using image-based cytological profiling assay.
Lee S; Lim D; Lee E; Lee N; Lee HG; Cechetto J; Liuzzi M; Freitas-Junior LH; Song JS; Bae MA; Oh S; Ayong L; Park SB
J Med Chem; 2014 Sep; 57(17):7425-34. PubMed ID: 25137549
[TBL] [Abstract][Full Text] [Related]
15. Ligand-based virtual screening and in silico design of new antimalarial compounds using nonstochastic and stochastic total and atom-type quadratic maps.
Marrero-Ponce Y; Iyarreta-Veitía M; Montero-Torres A; Romero-Zaldivar C; Brandt CA; Avila PE; Kirchgatter K; Machado Y
J Chem Inf Model; 2005; 45(4):1082-100. PubMed ID: 16045304
[TBL] [Abstract][Full Text] [Related]
16. A Developability-Focused Optimization Approach Allows Identification of in Vivo Fast-Acting Antimalarials: N-[3-[(Benzimidazol-2-yl)amino]propyl]amides.
Keurulainen L; Vahermo M; Puente-Felipe M; Sandoval-Izquierdo E; Crespo-Fernández B; Guijarro-López L; Huertas-Valentín L; de las Heras-Dueña L; Leino TO; Siiskonen A; Ballell-Pages L; Sanz LM; Castañeda-Casado P; Jiménez-Díaz MB; Martínez-Martínez MS; Viera S; Kiuru P; Calderón F; Yli-Kauhaluoma J
J Med Chem; 2015 Jun; 58(11):4573-80. PubMed ID: 25906200
[TBL] [Abstract][Full Text] [Related]
17. Potent Plasmodium falciparum gametocytocidal activity of diaminonaphthoquinones, lead antimalarial chemotypes identified in an antimalarial compound screen.
Tanaka TQ; Guiguemde WA; Barnett DS; Maron MI; Min J; Connelly MC; Suryadevara PK; Guy RK; Williamson KC
Antimicrob Agents Chemother; 2015 Mar; 59(3):1389-97. PubMed ID: 25512421
[TBL] [Abstract][Full Text] [Related]
18. From crystal to compound: structure-based antimalarial drug discovery.
Drinkwater N; McGowan S
Biochem J; 2014 Aug; 461(3):349-69. PubMed ID: 25008945
[TBL] [Abstract][Full Text] [Related]
19. Synthesis, characterization, molecular docking and in vitro antimalarial properties of new carboxamides bearing sulphonamide.
Ugwu DI; Okoro UC; Ukoha PO; Okafor S; Ibezim A; Kumar NM
Eur J Med Chem; 2017 Jul; 135():349-369. PubMed ID: 28460310
[TBL] [Abstract][Full Text] [Related]
20. 2-Aminothiophene-3-carboxylates and carboxamides as adenosine A1 receptor allosteric enhancers.
Nikolakopoulos G; Figler H; Linden J; Scammells PJ
Bioorg Med Chem; 2006 Apr; 14(7):2358-65. PubMed ID: 16314104
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
