These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
2. 11 beta-amidoalkyl estradiols, a new series of pure antiestrogens. Claussner A; Nédélec L; Nique F; Philibert D; Teutsch G; Van de Velde P J Steroid Biochem Mol Biol; 1992 Mar; 41(3-8):609-14. PubMed ID: 1562531 [TBL] [Abstract][Full Text] [Related]
3. 1H and 13C nuclear magnetic resonance assignments and stereochemistry of N-n-butyl-N-methyl-11-(16'alpha-chloro-3',17'beta- and 17'alpha-dihydroxyestra-1',3',5'(10')-trien-7'alpha-yl) undecanamide. Dionne P; Singh SM; Labrie F Steroids; 1994 Aug; 59(8):493-7. PubMed ID: 7985212 [TBL] [Abstract][Full Text] [Related]
4. Synthesis and biological activity of 17 alpha-alkynylamide derivatives of estradiol. Poirier D; Labrie C; Mérand Y; Labrie F J Steroid Biochem Mol Biol; 1991 Jun; 38(6):759-74. PubMed ID: 2064992 [TBL] [Abstract][Full Text] [Related]
5. Synthesis and biological activity of new halo-steroidal antiestrogens. Levesque C; Merand Y; Dufour JM; Labrie C; Labrie F J Med Chem; 1991 May; 34(5):1624-30. PubMed ID: 2033587 [TBL] [Abstract][Full Text] [Related]
6. Influence of alkyl chain ramification on estradiol receptor binding affinity and intrinsic activity of 1,2-dialkylated 1,2-bis(4- or 3-hydroxyphenyl)ethane estrogens and antiestrogens. Hartmann RW J Med Chem; 1986 Sep; 29(9):1668-74. PubMed ID: 3018243 [TBL] [Abstract][Full Text] [Related]
8. Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl] [4-[2-(1-piperidinyl)ethoxy]-phenyl]methanone hydrochloride (LY156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity. Jones CD; Jevnikar MG; Pike AJ; Peters MK; Black LJ; Thompson AR; Falcone JF; Clemens JA J Med Chem; 1984 Aug; 27(8):1057-66. PubMed ID: 6431104 [TBL] [Abstract][Full Text] [Related]
9. Biology and mode of action of pure antioestrogens. Wakeling AE; Bowler J J Steroid Biochem; 1988; 30(1-6):141-7. PubMed ID: 3386242 [TBL] [Abstract][Full Text] [Related]
10. Synthesis and biologic activities of 11 beta-substituted estradiol as potential antiestrogens. Qian XD; Abul-Hajj YJ Steroids; 1990 May; 55(5):238-41. PubMed ID: 2360220 [TBL] [Abstract][Full Text] [Related]
12. Synthesis and biological evaluation of a series of 1,1-dichloro-2,2,3-triarylcyclopropanes as pure antiestrogens. Day BW; Magarian RA; Jain PT; Pento JT; Mousissian GK; Meyer KL J Med Chem; 1991 Feb; 34(2):842-51. PubMed ID: 1995907 [TBL] [Abstract][Full Text] [Related]
13. Structure-activity relationship of antiestrogens. Effect of the side chain and its position on the activity of 2,3-diaryl-2H-1-benzopyrans. Sharma AP; Saeed A; Durani S; Kapil RS J Med Chem; 1990 Dec; 33(12):3216-22. PubMed ID: 2258907 [TBL] [Abstract][Full Text] [Related]
14. Estrogen to antiestrogen with a single methylene group resulting in an unusual steroidal selective estrogen receptor modulator. Zhang JX; Labaree DC; Mor G; Hochberg RB J Clin Endocrinol Metab; 2004 Jul; 89(7):3527-35. PubMed ID: 15240642 [TBL] [Abstract][Full Text] [Related]
15. Differential interactions of estrogens and antiestrogens at the 17 beta-hydroxy or counterpart function with the estrogen receptor. Borgna JL; Scali J Eur J Biochem; 1991 Aug; 199(3):575-85. PubMed ID: 1868844 [TBL] [Abstract][Full Text] [Related]
16. Additive inhibitory effects of an androgen and the antiestrogen EM-170 on estradiol-stimulated growth of human ZR-75-1 breast tumors in athymic mice. Dauvois S; Geng CS; Lévesque C; Mérand Y; Labrie F Cancer Res; 1991 Jun; 51(12):3131-5. PubMed ID: 2039992 [TBL] [Abstract][Full Text] [Related]
17. Interaction of estrogen-nitrosourea conjugates with the estrogen receptor in rat uterus. Lam HY; Goldenberg GJ; Wong CM Biochem Pharmacol; 1988 Jul; 37(13):2625-31. PubMed ID: 3390222 [TBL] [Abstract][Full Text] [Related]
18. Ring-substituted 1,1,2,2-tetraalkylated 1,2-bis(hydroxyphenyl)ethanes. 4. Synthesis, estrogen receptor binding affinity, and evaluation of antiestrogenic and mammary tumor inhibiting activity of symmetrically disubstituted 1,1,2,2-tetramethyl-1,2-bis(hydroxyphenyl)ethanes. Hartmann RW; Schwarz W; Heindl A; Schönenberger H J Med Chem; 1985 Sep; 28(9):1295-301. PubMed ID: 2993619 [TBL] [Abstract][Full Text] [Related]