232 related articles for article (PubMed ID: 28152429)
1. Synthesis and biological evaluation of fluorinated N-benzoyl and N-phenylacetoyl derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as steroid sulfatase inhibitors.
Daśko M; Przybyłowska M; Rachon J; Masłyk M; Kubiński K; Misiak M; Składanowski A; Demkowicz S
Eur J Med Chem; 2017 Mar; 128():79-87. PubMed ID: 28152429
[TBL] [Abstract][Full Text] [Related]
2. Synthesis and Biological Evaluation of Fluorinated 3-Phenylcoumarin-7-O-Sulfamate Derivatives as Steroid Sulfatase Inhibitors.
Demkowicz S; Daśko M; Kozak W; Krawczyk K; Witt D; Masłyk M; Kubiński K; Rachon J
Chem Biol Drug Des; 2016 Feb; 87(2):233-8. PubMed ID: 26280898
[TBL] [Abstract][Full Text] [Related]
3. Novel steroid sulfatase inhibitors based on N-thiophosphorylated 3-(4-aminophenyl)-coumarin-7-O-sulfamates.
Daśko M; Demkowicz S; Biernacki K; Harrous A; Rachon J; Kozak W; Martyna A; Masłyk M; Kubiński K; Boguszewska-Czubara A
Drug Dev Res; 2019 Sep; 80(6):857-866. PubMed ID: 31301181
[TBL] [Abstract][Full Text] [Related]
4. Design and synthesis of 3-benzylaminocoumarin-7-O-sulfamate derivatives as steroid sulfatase inhibitors.
Hng Y; Lin MH; Lin TS; Liu IC; Lin IC; Lu YL; Chang CN; Chiu PF; Tsai KC; Chen MJ; Liang PH
Bioorg Chem; 2020 Mar; 96():103618. PubMed ID: 32059152
[TBL] [Abstract][Full Text] [Related]
5. Steroidal and nonsteroidal sulfamates as potent inhibitors of steroid sulfatase.
Woo LW; Howarth NM; Purohit A; Hejaz HA; Reed MJ; Potter BV
J Med Chem; 1998 Mar; 41(7):1068-83. PubMed ID: 9544207
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and biological evaluation of N-acylated tyramine sulfamates containing C-F bonds as steroid sulfatase inhibitors.
Daśko M; Rachon J; Masłyk M; Kubiński K; Demkowicz S
Chem Biol Drug Des; 2017 Jul; 90(1):156-161. PubMed ID: 28032462
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and biological evaluation of thiophosphate tricyclic coumarin derivatives as steroid sulfatase inhibitors.
Kozak W; Daśko M; Masłyk M; Gielniewski B; Rachon J; Demkowicz S
J Asian Nat Prod Res; 2015; 17(11):1091-6. PubMed ID: 26269086
[TBL] [Abstract][Full Text] [Related]
8. Estrogen O-sulfamates and their analogues: Clinical steroid sulfatase inhibitors with broad potential.
Thomas MP; Potter BV
J Steroid Biochem Mol Biol; 2015 Sep; 153():160-9. PubMed ID: 25843211
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitors.
Demkowicz S; Kozak W; Daśko M; Masłyk M; Gielniewski B; Rachon J
Eur J Med Chem; 2015 Aug; 101():358-66. PubMed ID: 26163883
[TBL] [Abstract][Full Text] [Related]
10. A novel steroidal selective steroid sulfatase inhibitor KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells in vitro and in animal models.
Ishida H; Nakata T; Suzuki M; Shiotsu Y; Tanaka H; Sato N; Terasaki Y; Takebayashi M; Anazawa H; Murakata C; Li PK; Kuwabara T; Akinaga S
Breast Cancer Res Treat; 2007 Dec; 106(2):215-27. PubMed ID: 17268815
[TBL] [Abstract][Full Text] [Related]
11. 2-phenylindole sulfamates: inhibitors of steroid sulfatase with antiproliferative activity in MCF-7 breast cancer cells.
Walter G; Liebl R; von Angerer E
J Steroid Biochem Mol Biol; 2004 Apr; 88(4-5):409-20. PubMed ID: 15145451
[TBL] [Abstract][Full Text] [Related]
12. Development of novel steroid sulfatase inhibitors. I. Synthesis and biological evaluation of biphenyl-4-O-sulfamates.
Okada M; Nakagawa T; Iwashita S; Takegawa S; Fujii T; Koizumi N
J Steroid Biochem Mol Biol; 2003 Nov; 87(2-3):141-8. PubMed ID: 14672734
[TBL] [Abstract][Full Text] [Related]
13. Design, structure-activity relationships, and enzyme kinetic studies of tricyclic and tetracyclic coumarin-based sulfamates as steroid sulfatase inhibitors.
Chiu PF; Lin IC; Lu YL; Chang CN; Chan HY; Lin TS; Tsai KC; Hsieh YSY; Chen MJ; Lin MH; Liang PH
Bioorg Chem; 2023 Sep; 138():106581. PubMed ID: 37172437
[TBL] [Abstract][Full Text] [Related]
14. Phosphate and thiophosphate biphenyl analogs as steroid sulfatase inhibitors.
Demkowicz S; Kozak W; Daśko M; Masłyk M; Kubiński K; Rachon J
Drug Dev Res; 2015 Mar; 76(2):94-104. PubMed ID: 25845343
[TBL] [Abstract][Full Text] [Related]
15. Steroid Sulfatase Inhibitors Based on Phosphate and Thiophosphate Flavone Analogs.
Kozak W; Daśko M; Masłyk M; Kubiński K; Rachon J; Demkowicz S
Drug Dev Res; 2015 Dec; 76(8):450-62. PubMed ID: 26415657
[TBL] [Abstract][Full Text] [Related]
16. Inhibition of steroid sulfatase activity and cell proliferation in ZR-75-1 and BT-474 human breast cancer cells by KW-2581 in vitro and in vivo.
Ishida H; Nakata T; Sato N; Li PK; Kuwabara T; Akinaga S
Breast Cancer Res Treat; 2007 Aug; 104(2):211-9. PubMed ID: 17061037
[TBL] [Abstract][Full Text] [Related]
17. New potent STS inhibitors based on fluorinated 4-(1-phenyl-1
Daśko M; Demkowicz S; Rachon J; Biernacki K; Aszyk J; Kozak W; Masłyk M; Kubiński K
J Asian Nat Prod Res; 2020 Nov; 22(11):1037-1044. PubMed ID: 31773975
[TBL] [Abstract][Full Text] [Related]
18. Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors.
El-Gamal MI; Semreen MH; Foster PA; Potter BV
Bioorg Med Chem; 2016 Jun; 24(12):2762-7. PubMed ID: 27143133
[TBL] [Abstract][Full Text] [Related]
19. A novel dual-target steroid sulfatase inhibitor and antiestrogen: SR 16157, a promising agent for the therapy of breast cancer.
Rasmussen LM; Zaveri NT; Stenvang J; Peters RH; Lykkesfeldt AE
Breast Cancer Res Treat; 2007 Dec; 106(2):191-203. PubMed ID: 17268816
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and evaluation of analogues of estrone-3-O-sulfamate as potent steroid sulfatase inhibitors.
Lawrence Woo LW; Leblond B; Purohit A; Potter BV
Bioorg Med Chem; 2012 Apr; 20(8):2506-19. PubMed ID: 22455789
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
