138 related articles for article (PubMed ID: 28161251)
1. Carbonic anhydrases activation with 3-amino-1H-1,2,4-triazole-1-carboxamides: Discovery of subnanomolar isoform II activators.
Le Duc Y; Licsandru E; Vullo D; Barboiu M; Supuran CT
Bioorg Med Chem; 2017 Mar; 25(5):1681-1686. PubMed ID: 28161251
[TBL] [Abstract][Full Text] [Related]
2. α-Carbonic anhydrases are strongly activated by spinaceamine derivatives.
Akocak S; Lolak N; Bua S; Nocentini A; Karakoc G; Supuran CT
Bioorg Med Chem; 2019 Mar; 27(5):800-804. PubMed ID: 30683554
[TBL] [Abstract][Full Text] [Related]
3. Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with l- and d-histidine and crystallographic analysis of their adducts with isoform II: engineering proton-transfer processes within the active site of an enzyme.
Temperini C; Scozzafava A; Vullo D; Supuran CT
Chemistry; 2006 Sep; 12(27):7057-66. PubMed ID: 16807956
[TBL] [Abstract][Full Text] [Related]
4. A class of carbonic anhydrase I - selective activators.
Licsandru E; Tanc M; Kocsis I; Barboiu M; Supuran CT
J Enzyme Inhib Med Chem; 2017 Dec; 32(1):37-46. PubMed ID: 27798977
[TBL] [Abstract][Full Text] [Related]
5. Designing of novel carbonic anhydrase inhibitors and activators.
Supuran CT; Vullo D; Manole G; Casini A; Scozzafava A
Curr Med Chem Cardiovasc Hematol Agents; 2004 Jan; 2(1):49-68. PubMed ID: 15328829
[TBL] [Abstract][Full Text] [Related]
6. Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II, and IX with a series of 1,3,4-thiadiazole- and 1,2,4-triazole-thiols.
Almajan GL; Innocenti A; Puccetti L; Manole G; Barbuceanu S; Saramet I; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2005 May; 15(9):2347-52. PubMed ID: 15837323
[TBL] [Abstract][Full Text] [Related]
7. Carbonic anhydrase activation profile of indole-based derivatives.
Barresi E; Ravichandran R; Germelli L; Angeli A; Baglini E; Salerno S; Marini AM; Costa B; Da Pozzo E; Martini C; Da Settimo F; Supuran C; Cosconati S; Taliani S
J Enzyme Inhib Med Chem; 2021 Dec; 36(1):1783-1797. PubMed ID: 34340630
[TBL] [Abstract][Full Text] [Related]
8. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole.
Supuran CT; Scozzafava A
J Enzyme Inhib; 2000; 15(5):471-86. PubMed ID: 11030087
[TBL] [Abstract][Full Text] [Related]
9. Carbonic anhydrase activators. Activation of isoforms I, II, IV, VA, VII, and XIV with L- and D-phenylalanine and crystallographic analysis of their adducts with isozyme II: stereospecific recognition within the active site of an enzyme and its consequences for the drug design.
Temperini C; Scozzafava A; Vullo D; Supuran CT
J Med Chem; 2006 May; 49(10):3019-27. PubMed ID: 16686544
[TBL] [Abstract][Full Text] [Related]
10. 6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII.
Grandane A; Tanc M; Zalubovskis R; Supuran CT
Bioorg Med Chem Lett; 2014 Mar; 24(5):1256-60. PubMed ID: 24518190
[TBL] [Abstract][Full Text] [Related]
11. Carbonic anhydrase activators: activation of isozyme XIII with amino acids and amines.
Parkkila S; Vullo D; Puccetti L; Parkkila AK; Scozzafava A; Supuran CT
Bioorg Med Chem Lett; 2006 Aug; 16(15):3955-9. PubMed ID: 16730978
[TBL] [Abstract][Full Text] [Related]
12. (Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators.
Rami M; Winum JY; Supuran CT; Melnyk P; Yous S
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):224-229. PubMed ID: 30734616
[TBL] [Abstract][Full Text] [Related]
13. Mono- and di-halogenated histamine, histidine and carnosine derivatives are potent carbonic anhydrase I, II, VII, XII and XIV activators.
Saada MC; Vullo D; Montero JL; Scozzafava A; Supuran CT; Winum JY
Bioorg Med Chem; 2014 Sep; 22(17):4752-8. PubMed ID: 25082511
[TBL] [Abstract][Full Text] [Related]
14. Carbonic anhydrase activators: X-ray crystal structure of the adduct of human isozyme II with L-histidine as a platform for the design of stronger activators.
Temperini C; Scozzafava A; Puccetti L; Supuran CT
Bioorg Med Chem Lett; 2005 Dec; 15(23):5136-41. PubMed ID: 16214338
[TBL] [Abstract][Full Text] [Related]
15. Carbonic anhydrase activators: activation of the human isoforms VII (cytosolic) and XIV (transmembrane) with amino acids and amines.
Vullo D; Innocenti A; Nishimori I; Scozzafava A; Kaila K; Supuran CT
Bioorg Med Chem Lett; 2007 Aug; 17(15):4107-12. PubMed ID: 17540561
[TBL] [Abstract][Full Text] [Related]
16. Carbonic anhydrase activators - part 21. Novel activators of isozymes I, II and IV incorporating carboxamido and ureido histamine moieties.
Scozzafava A; Supuran CT
Eur J Med Chem; 2000 Jan; 35(1):31-9. PubMed ID: 10733601
[TBL] [Abstract][Full Text] [Related]
17. Carbonic anhydrase activators: gold nanoparticles coated with derivatized histamine, histidine, and carnosine show enhanced activatory effects on several mammalian isoforms.
Saada MC; Montero JL; Vullo D; Scozzafava A; Winum JY; Supuran CT
J Med Chem; 2011 Mar; 54(5):1170-7. PubMed ID: 21291238
[TBL] [Abstract][Full Text] [Related]
18. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(4-tosylureido-amino acyl)ethyl-1H-imidazole (histamine derivatives).
Scozzafava A; Iorga B; Supuran CT
J Enzyme Inhib; 2000; 15(2):139-61. PubMed ID: 10938540
[TBL] [Abstract][Full Text] [Related]
19. Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators.
Angeli A; Berrino E; Carradori S; Supuran CT; Cirri M; Carta F; Costantino G
Molecules; 2021 Dec; 26(23):. PubMed ID: 34885917
[TBL] [Abstract][Full Text] [Related]
20. Benzenesulfonamide bearing 1,2,4-triazole scaffolds as potent inhibitors of tumor associated carbonic anhydrase isoforms hCA IX and hCA XII.
SitaRam ; Celik G; Khloya P; Vullo D; Supuran CT; Sharma PK
Bioorg Med Chem; 2014 Mar; 22(6):1873-82. PubMed ID: 24560737
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]