163 related articles for article (PubMed ID: 28192916)
1. Combating Enhanced Intracellular Survival (Eis)-Mediated Kanamycin Resistance of Mycobacterium tuberculosis by Novel Pyrrolo[1,5-a]pyrazine-Based Eis Inhibitors.
Garzan A; Willby MJ; Ngo HX; Gajadeera CS; Green KD; Holbrook SY; Hou C; Posey JE; Tsodikov OV; Garneau-Tsodikova S
ACS Infect Dis; 2017 Apr; 3(4):302-309. PubMed ID: 28192916
[TBL] [Abstract][Full Text] [Related]
2. Potent Inhibitors of Acetyltransferase Eis Overcome Kanamycin Resistance in Mycobacterium tuberculosis.
Willby MJ; Green KD; Gajadeera CS; Hou C; Tsodikov OV; Posey JE; Garneau-Tsodikova S
ACS Chem Biol; 2016 Jun; 11(6):1639-46. PubMed ID: 27010218
[TBL] [Abstract][Full Text] [Related]
3. Potent 1,2,4-Triazino[5,6 b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis.
Ngo HX; Green KD; Gajadeera CS; Willby MJ; Holbrook SYL; Hou C; Garzan A; Mayhoub AS; Posey JE; Tsodikov OV; Garneau-Tsodikova S
ACS Infect Dis; 2018 Jun; 4(6):1030-1040. PubMed ID: 29601176
[TBL] [Abstract][Full Text] [Related]
4. Structure-Guided Optimization of Inhibitors of Acetyltransferase Eis from
Punetha A; Ngo HX; Holbrook SYL; Green KD; Willby MJ; Bonnett SA; Krieger K; Dennis EK; Posey JE; Parish T; Tsodikov OV; Garneau-Tsodikova S
ACS Chem Biol; 2020 Jun; 15(6):1581-1594. PubMed ID: 32421305
[TBL] [Abstract][Full Text] [Related]
5. Sulfonamide-Based Inhibitors of Aminoglycoside Acetyltransferase Eis Abolish Resistance to Kanamycin in Mycobacterium tuberculosis.
Garzan A; Willby MJ; Green KD; Gajadeera CS; Hou C; Tsodikov OV; Posey JE; Garneau-Tsodikova S
J Med Chem; 2016 Dec; 59(23):10619-10628. PubMed ID: 27933949
[TBL] [Abstract][Full Text] [Related]
6. Probing the Robustness of Inhibitors of Tuberculosis Aminoglycoside Resistance Enzyme Eis by Mutagenesis.
Green KD; Punetha A; Hou C; Garneau-Tsodikova S; Tsodikov OV
ACS Infect Dis; 2019 Oct; 5(10):1772-1778. PubMed ID: 31433614
[TBL] [Abstract][Full Text] [Related]
7. Discovery of substituted benzyloxy-benzylamine inhibitors of acetyltransferase Eis and their anti-mycobacterial activity.
Pang AH; Green KD; Chandrika NT; Garzan A; Punetha A; Holbrook SYL; Willby MJ; Posey JE; Tsodikov OV; Garneau-Tsodikova S
Eur J Med Chem; 2022 Nov; 242():114698. PubMed ID: 36037791
[TBL] [Abstract][Full Text] [Related]
8. Discovery and Mechanistic Analysis of Structurally Diverse Inhibitors of Acetyltransferase Eis among FDA-Approved Drugs.
Pang AH; Green KD; Punetha A; Thamban Chandrika N; Howard KC; Garneau-Tsodikova S; Tsodikov OV
Biochemistry; 2023 Feb; 62(3):710-721. PubMed ID: 36657084
[TBL] [Abstract][Full Text] [Related]
9. A consensus reverse docking approach for identification of a competitive inhibitor of acetyltransferase enhanced intracellular survival protein from Mycobacterium tuberculosis.
Santos-Júnior PFDS; Batista VM; Nascimento IJDS; Nunes IC; Silva LR; Costa CACB; Freitas JD; Quintans-Júnior LJ; Araújo-Júnior JX; Freitas MEG; Zhan P; Green KD; Garneau-Tsodikova S; Mendonça-Júnior FJB; Rodrigues-Junior VS; Silva-Júnior EFD
Bioorg Med Chem; 2024 Jun; 108():117774. PubMed ID: 38833750
[TBL] [Abstract][Full Text] [Related]
10. Identification and characterization of inhibitors of the aminoglycoside resistance acetyltransferase Eis from Mycobacterium tuberculosis.
Green KD; Chen W; Garneau-Tsodikova S
ChemMedChem; 2012 Jan; 7(1):73-7. PubMed ID: 21898832
[No Abstract] [Full Text] [Related]
11. Redesign of substrate specificity and identification of the aminoglycoside binding residues of Eis from Mycobacterium tuberculosis.
Jennings BC; Labby KJ; Green KD; Garneau-Tsodikova S
Biochemistry; 2013 Jul; 52(30):5125-32. PubMed ID: 23837529
[TBL] [Abstract][Full Text] [Related]
12. Biochemical and structural analysis of aminoglycoside acetyltransferase Eis from Anabaena variabilis.
Pricer RE; Houghton JL; Green KD; Mayhoub AS; Garneau-Tsodikova S
Mol Biosyst; 2012 Oct; 8(12):3305-13. PubMed ID: 23090428
[TBL] [Abstract][Full Text] [Related]
13. Development of ssDNA aptamers as potent inhibitors of Mycobacterium tuberculosis acetohydroxyacid synthase.
Baig IA; Moon JY; Lee SC; Ryoo SW; Yoon MY
Biochim Biophys Acta; 2015 Oct; 1854(10 Pt A):1338-50. PubMed ID: 25988243
[TBL] [Abstract][Full Text] [Related]
14. Andrographolide: A potent antituberculosis compound that targets Aminoglycoside 2'-N-acetyltransferase in Mycobacterium tuberculosis.
Prabu A; Hassan S; Prabuseenivasan ; Shainaba AS; Hanna LE; Kumar V
J Mol Graph Model; 2015 Sep; 61():133-40. PubMed ID: 26245695
[TBL] [Abstract][Full Text] [Related]
15. Targeting Aminoglycoside Acetyltransferase Activity of Mycobacterium tuberculosis (H37Rv) Derived Eis (Enhanced Intracellular Survival) Protein with Quercetin.
Radhakrishnan L; Dani R; Navabshan I; Jamal S; Ahmed N
Protein J; 2024 Feb; 43(1):12-23. PubMed ID: 37932619
[TBL] [Abstract][Full Text] [Related]
16. eis Promoter C14G and C15G Mutations Do Not Confer Kanamycin Resistance in Mycobacterium tuberculosis.
Pholwat S; Stroup S; Heysell S; Ogarkov O; Zhdanova S; Ramakrishnan G; Houpt E
Antimicrob Agents Chemother; 2016 Dec; 60(12):7522-7523. PubMed ID: 27736762
[TBL] [Abstract][Full Text] [Related]
17. Discovery of novel lysine ɛ-aminotransferase inhibitors: An intriguing potential target for latent tuberculosis.
Devi PB; Sridevi JP; Kakan SS; Saxena S; Jeankumar VU; Soni V; Anantaraju HS; Yogeeswari P; Sriram D
Tuberculosis (Edinb); 2015 Dec; 95(6):786-794. PubMed ID: 26299907
[TBL] [Abstract][Full Text] [Related]
18. Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from
Punetha A; Green KD; Garzan A; Thamban Chandrika N; Willby MJ; Pang AH; Hou C; Holbrook SYL; Krieger K; Posey JE; Parish T; Tsodikov OV; Garneau-Tsodikova S
RSC Med Chem; 2021 Nov; 12(11):1894-1909. PubMed ID: 34825186
[TBL] [Abstract][Full Text] [Related]
19. Discovery and development of inhibitors of acetyltransferase Eis to combat Mycobacterium tuberculosis.
Pang AH; Green KD; Tsodikov OV; Garneau-Tsodikova S
Methods Enzymol; 2023; 690():369-396. PubMed ID: 37858535
[TBL] [Abstract][Full Text] [Related]
20. Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB.
Chen W; Biswas T; Porter VR; Tsodikov OV; Garneau-Tsodikova S
Proc Natl Acad Sci U S A; 2011 Jun; 108(24):9804-8. PubMed ID: 21628583
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]