These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
4. Effects of high-affinity inhibitors on partial reactions, charge movements, and conformational States of the Ca2+ transport ATPase (sarco-endoplasmic reticulum Ca2+ ATPase). Tadini-Buoninsegni F; Bartolommei G; Moncelli MR; Tal DM; Lewis D; Inesi G Mol Pharmacol; 2008 Apr; 73(4):1134-40. PubMed ID: 18212248 [TBL] [Abstract][Full Text] [Related]
5. Functional comparison between secretory pathway Ca2+/Mn2+-ATPase (SPCA) 1 and sarcoplasmic reticulum Ca2+-ATPase (SERCA) 1 isoforms by steady-state and transient kinetic analyses. Dode L; Andersen JP; Raeymaekers L; Missiaen L; Vilsen B; Wuytack F J Biol Chem; 2005 Nov; 280(47):39124-34. PubMed ID: 16192278 [TBL] [Abstract][Full Text] [Related]
6. Identification of novel inhibitors of human SPCA2. Yamamoto S; Takehara M; Kabashima Y; Fukutomi T; Ushimaru M Biochem Biophys Res Commun; 2016 Aug; 477(2):266-70. PubMed ID: 27297103 [TBL] [Abstract][Full Text] [Related]
7. Critical roles of hydrophobicity and orientation of side chains for inactivation of sarcoplasmic reticulum Ca2+-ATPase with thapsigargin and thapsigargin analogs. Winther AM; Liu H; Sonntag Y; Olesen C; le Maire M; Soehoel H; Olsen CE; Christensen SB; Nissen P; Møller JV J Biol Chem; 2010 Sep; 285(37):28883-92. PubMed ID: 20551329 [TBL] [Abstract][Full Text] [Related]
8. Applying linear interaction energy method for rational design of noncompetitive allosteric inhibitors of the sarco- and endoplasmic reticulum calcium-ATPase. Singh P; Mhaka AM; Christensen SB; Gray JJ; Denmeade SR; Isaacs JT J Med Chem; 2005 Apr; 48(8):3005-14. PubMed ID: 15828839 [TBL] [Abstract][Full Text] [Related]
9. Specific structural requirements for the inhibitory effect of thapsigargin on the Ca2+ ATPase SERCA. Xu C; Ma H; Inesi G; Al-Shawi MK; Toyoshima C J Biol Chem; 2004 Apr; 279(17):17973-9. PubMed ID: 14970206 [TBL] [Abstract][Full Text] [Related]
10. Elucidation of the topography of the thapsigargin binding site in the sarco-endoplasmic calcium ATPase. Skytte DM; Møller JV; Liu H; Nielsen HØ; Svenningsen LE; Jensen CM; Olsen CE; Christensen SB Bioorg Med Chem; 2010 Aug; 18(15):5634-46. PubMed ID: 20615710 [TBL] [Abstract][Full Text] [Related]
12. Molecular determinants of thapsigargin binding by SERCA Ca2+-ATPase: a computational docking study. Paula S; Ball WJ Proteins; 2004 Aug; 56(3):595-606. PubMed ID: 15229891 [TBL] [Abstract][Full Text] [Related]
13. Ca2+ uptake and release properties of a thapsigargin-insensitive nonmitochondrial Ca2+ store in A7r5 and 16HBE14o- cells. Missiaen L; Vanoevelen J; Parys JB; Raeymaekers L; De Smedt H; Callewaert G; Erneux C; Wuytack F J Biol Chem; 2002 Mar; 277(9):6898-902. PubMed ID: 11861657 [TBL] [Abstract][Full Text] [Related]
14. Identifying the sarco(endo)plasmic reticulum Ca2+ ATPase (SERCA) as a potential target for hypericin--a theoretical study. Eriksson ES; Eriksson LA Phys Chem Chem Phys; 2012 Sep; 14(36):12637-46. PubMed ID: 22892582 [TBL] [Abstract][Full Text] [Related]
15. Cryo-EM structures of human SPCA1a reveal the mechanism of Ca Chen Z; Watanabe S; Hashida H; Inoue M; Daigaku Y; Kikkawa M; Inaba K Sci Adv; 2023 Mar; 9(9):eadd9742. PubMed ID: 36867705 [TBL] [Abstract][Full Text] [Related]
16. A Darier disease mutation relieves kinetic constraints imposed by the tail of sarco(endo)plasmic reticulum Ca Mikkelsen SA; Vangheluwe P; Andersen JP J Biol Chem; 2018 Mar; 293(11):3880-3889. PubMed ID: 29363575 [TBL] [Abstract][Full Text] [Related]
17. Design, synthesis, and pharmacological evaluation of thapsigargin analogues for targeting apoptosis to prostatic cancer cells. Jakobsen CM; Denmeade SR; Isaacs JT; Gady A; Olsen CE; Christensen SB J Med Chem; 2001 Dec; 44(26):4696-703. PubMed ID: 11741487 [TBL] [Abstract][Full Text] [Related]
18. Comparison of current docking tools for the simulation of inhibitor binding by the transmembrane domain of the sarco/endoplasmic reticulum calcium ATPase. Lape M; Elam C; Paula S Biophys Chem; 2010 Aug; 150(1-3):88-97. PubMed ID: 20167416 [TBL] [Abstract][Full Text] [Related]
19. Overlapping effects of S3 stalk segment mutations on the affinity of Ca2+-ATPase (SERCA) for thapsigargin and cyclopiazonic acid. Ma H; Zhong L; Inesi G; Fortea I; Soler F; Fernandez-Belda F Biochemistry; 1999 Nov; 38(47):15522-7. PubMed ID: 10569935 [TBL] [Abstract][Full Text] [Related]
20. Functional characterization of the Ca Maréchal X; De Mendonça R; Miras R; Revilloud J; Catty P Biochem J; 2018 Jan; 475(1):289-303. PubMed ID: 29229760 [No Abstract] [Full Text] [Related] [Next] [New Search]