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2. New structure-activity relationships of the quinolone antibacterials using the target enzyme. The development and application of a DNA gyrase assay. Domagala JM; Hanna LD; Heifetz CL; Hutt MP; Mich TF; Sanchez JP; Solomon M J Med Chem; 1986 Mar; 29(3):394-404. PubMed ID: 3005575 [TBL] [Abstract][Full Text] [Related]
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5. [Mechanism of action of quinolones]. Smith JT Infection; 1986; 14 Suppl 1():S3-15. PubMed ID: 2420724 [TBL] [Abstract][Full Text] [Related]
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10. Comparative antibacterial activity of new quinolone-carboxylic acid derivatives. Mitsuhashi S Rev Infect Dis; 1988; 10 Suppl 1():S27-31. PubMed ID: 3347811 [TBL] [Abstract][Full Text] [Related]
11. Synthesis and anti-staphylococcal activity of novel bacterial topoisomerase inhibitors with a 5-amino-1,3-dioxane linker moiety. Li L; Okumu A; Dellos-Nolan S; Li Z; Karmahapatra S; English A; Yalowich JC; Wozniak DJ; Mitton-Fry MJ Bioorg Med Chem Lett; 2018 Aug; 28(14):2477-2480. PubMed ID: 29871847 [TBL] [Abstract][Full Text] [Related]
12. Discrepancy between the antibacterial activities and the inhibitory effects on Micrococcus luteus DNA gyrase of 13 quinolones. Fu KP; Grace ME; McCloud SJ; Gregory FJ; Hung PP Chemotherapy; 1986; 32(6):494-8. PubMed ID: 3026740 [TBL] [Abstract][Full Text] [Related]
13. Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV. Mitton-Fry MJ; Brickner SJ; Hamel JC; Brennan L; Casavant JM; Chen M; Chen T; Ding X; Driscoll J; Hardink J; Hoang T; Hua E; Huband MD; Maloney M; Marfat A; McCurdy SP; McLeod D; Plotkin M; Reilly U; Robinson S; Schafer J; Shepard RM; Smith JF; Stone GG; Subramanyam C; Yoon K; Yuan W; Zaniewski RP; Zook C Bioorg Med Chem Lett; 2013 May; 23(10):2955-61. PubMed ID: 23566517 [TBL] [Abstract][Full Text] [Related]
14. The fluoroquinolones: structures, mechanisms of action and resistance, and spectra of activity in vitro. Wolfson JS; Hooper DC Antimicrob Agents Chemother; 1985 Oct; 28(4):581-6. PubMed ID: 3000292 [No Abstract] [Full Text] [Related]
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19. International experiences with ofloxacin, a new quinolone. Mitsuhashi S Infection; 1986; 14 Suppl 4():S223-5. PubMed ID: 3028965 [TBL] [Abstract][Full Text] [Related]
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