BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

118 related articles for article (PubMed ID: 28337330)

  • 1. Antimalarial Properties of Simplified Kalihinol Analogues.
    Daub ME; Prudhomme J; Ben Mamoun C; Le Roch KG; Vanderwal CD
    ACS Med Chem Lett; 2017 Mar; 8(3):355-360. PubMed ID: 28337330
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A Potent Kalihinol Analogue Disrupts Apicoplast Function and Vesicular Trafficking in
    Chahine Z; Abel S; Hollin T; Chung JH; Barnes GL; Daub ME; Renard I; Choi JY; Pratap V; Pal A; Alba-Argomaniz M; Banks C; Kirkwood J; Saraf A; Camino I; Castaneda P; Cuevas MC; De Mercado-Arnanz J; Fernandez-Alvaro E; Garcia-Perez A; Ibarz N; Viera-Morilla S; Prudhomme J; Joyner CJ; Bei AK; Florens L; Ben Mamoun C; Vanderwal CD; Le Roch KG
    bioRxiv; 2023 Nov; ():. PubMed ID: 38045341
    [TBL] [Abstract][Full Text] [Related]  

  • 3. N-cinnamoylation of antimalarial classics: quinacrine analogues with decreased toxicity and dual-stage activity.
    Gomes A; Pérez B; Albuquerque I; Machado M; Prudêncio M; Nogueira F; Teixeira C; Gomes P
    ChemMedChem; 2014 Feb; 9(2):305-10. PubMed ID: 24474655
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Borrelidin analogues with antimalarial activity: design, synthesis and biological evaluation against Plasmodium falciparum parasites.
    Sugawara A; Tanaka T; Hirose T; Ishiyama A; Iwatsuki M; Takahashi Y; Otoguro K; Ōmura S; Sunazuka T
    Bioorg Med Chem Lett; 2013 Apr; 23(8):2302-5. PubMed ID: 23499502
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Lerisetron Analogues with Antimalarial Properties: Synthesis, Structure-Activity Relationship Studies, and Biological Assessment.
    Mueller R; Reddy V; Nchinda AT; Mebrahtu F; Taylor D; Lawrence N; Tanner L; Barnabe M; Eyermann CJ; Zou B; Kondreddi RR; Lakshminarayana SB; Rottmann M; Street LJ; Chibale K
    ACS Omega; 2020 Mar; 5(12):6967-6982. PubMed ID: 32258933
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design and synthesis of simplified speciophylline analogues and β-carbolines as active molecules against Plasmodium falciparum.
    Pierrot D; Sinou V; Bun SS; Parzy D; Taudon N; Rodriguez J; Ollivier E; Bonne D
    Drug Dev Res; 2019 Feb; 80(1):133-137. PubMed ID: 30499121
    [TBL] [Abstract][Full Text] [Related]  

  • 7. New quinoline derivatives demonstrate a promising antimalarial activity against Plasmodium falciparum in vitro and Plasmodium berghei in vivo.
    Soares RR; da Silva JM; Carlos BC; da Fonseca CC; de Souza LS; Lopes FV; de Paula Dias RM; Moreira PO; Abramo C; Viana GH; de Pila Varotti F; da Silva AD; Scopel KK
    Bioorg Med Chem Lett; 2015 Jun; 25(11):2308-13. PubMed ID: 25920564
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and antimalarial evaluation of amide and urea derivatives based on the thiaplakortone A natural product scaffold.
    Schwartz BD; Skinner-Adams TS; Andrews KT; Coster MJ; Edstein MD; MacKenzie D; Charman SA; Koltun M; Blundell S; Campbell A; Pouwer RH; Quinn RJ; Beattie KD; Healy PC; Davis RA
    Org Biomol Chem; 2015 Feb; 13(5):1558-70. PubMed ID: 25490858
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Metabolites of febrifugine and its synthetic analogue by mouse liver S9 and their antimalarial activity against Plasmodium malaria parasite.
    Hirai S; Kikuchi H; Kim HS; Begum K; Wataya Y; Tasaka H; Miyazawa Y; Yamamoto K; Oshima Y
    J Med Chem; 2003 Sep; 46(20):4351-9. PubMed ID: 13678413
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Total synthesis of antimalarial diterpenoid (+)-kalihinol A.
    Miyaoka H; Abe Y; Sekiya N; Mitome H; Kawashima E
    Chem Commun (Camb); 2012 Jan; 48(6):901-3. PubMed ID: 22138854
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of gallinamide A analogues as potent falcipain inhibitors and antimalarials.
    Conroy T; Guo JT; Elias N; Cergol KM; Gut J; Legac J; Khatoon L; Liu Y; McGowan S; Rosenthal PJ; Hunt NH; Payne RJ
    J Med Chem; 2014 Dec; 57(24):10557-63. PubMed ID: 25412465
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Potent antimalarial febrifugine analogues against the plasmodium malaria parasite.
    Kikuchi H; Tasaka H; Hirai S; Takaya Y; Iwabuchi Y; Ooi H; Hatakeyama S; Kim HS; Wataya Y; Oshima Y
    J Med Chem; 2002 Jun; 45(12):2563-70. PubMed ID: 12036365
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Norepinephrine alkaloids as antiplasmodial agents: Synthesis of syncarpamide and insight into the structure-activity relationships of its analogues as antiplasmodial agents.
    Aratikatla EK; Valkute TR; Puri SK; Srivastava K; Bhattacharya AK
    Eur J Med Chem; 2017 Sep; 138():1089-1105. PubMed ID: 28763644
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design and Synthesis of Metabolically Stable tRNA Synthetase Inhibitors Derived from Cladosporin.
    Rusch M; Thevenon A; Hoepfner D; Aust T; Studer C; Patoor M; Rollin P; Livendahl M; Ranieri B; Schmitt E; Spanka C; Gademann K; Bouchez LC
    Chembiochem; 2019 Mar; 20(5):644-649. PubMed ID: 30462880
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Caged Garcinia Xanthones, a Novel Chemical Scaffold with Potent Antimalarial Activity.
    Ke H; Morrisey JM; Qu S; Chantarasriwong O; Mather MW; Theodorakis EA; Vaidya AB
    Antimicrob Agents Chemother; 2017 Jan; 61(1):. PubMed ID: 27799215
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Antimalarial activity of synthetic analogues of distamycin.
    Lombardi P; Crisanti A
    Pharmacol Ther; 1997; 76(1-3):125-33. PubMed ID: 9535174
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of antimalarial amide analogues based on the plant serrulatane diterpenoid 3,7,8-trihydroxyserrulat-14-en-19-oic acid.
    Kumar R; Duffy S; Avery VM; Davis RA
    Bioorg Med Chem Lett; 2017 Sep; 27(17):4091-4095. PubMed ID: 28774427
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Antimalarial benzoheterocyclic 4-aminoquinolines: Structure-activity relationship, in vivo evaluation, mechanistic and bioactivation studies.
    Ongarora DS; Strydom N; Wicht K; Njoroge M; Wiesner L; Egan TJ; Wittlin S; Jurva U; Masimirembwa CM; Chibale K
    Bioorg Med Chem; 2015 Sep; 23(17):5419-32. PubMed ID: 26264839
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis of alpha-substituted fosmidomycin analogues as highly potent Plasmodium falciparum growth inhibitors.
    Haemers T; Wiesner J; Van Poecke S; Goeman J; Henschker D; Beck E; Jomaa H; Van Calenbergh S
    Bioorg Med Chem Lett; 2006 Apr; 16(7):1888-91. PubMed ID: 16439126
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis, Biological Evaluation, and Molecular Modeling Studies of Chiral Chloroquine Analogues as Antimalarial Agents.
    Kondaparla S; Debnath U; Soni A; Dola VR; Sinha M; Srivastava K; Puri SK; Katti SB
    Antimicrob Agents Chemother; 2018 Dec; 62(12):. PubMed ID: 30224532
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.