BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

243 related articles for article (PubMed ID: 28372909)

  • 1. Y-shaped bis-arylethenesulfonic acid esters: Potential potent and membrane permeable protein tyrosine phosphatase 1B inhibitors.
    Yang F; Xie F; Zhang Y; Xia Y; Liu W; Jiang F; Lam C; Qiao Y; Xie D; Li J; Fu L
    Bioorg Med Chem Lett; 2017 May; 27(10):2166-2170. PubMed ID: 28372909
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis, and biological evaluation of 2-substituted ethenesulfonic acid ester derivatives as selective PTP1B inhibitors.
    Liu J; Deng X; Jin Y; Xu B; Liu W; Jiang F; Fu L
    Pharmazie; 2015 Jul; 70(7):446-51. PubMed ID: 26373204
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and biological evaluation of geniposide derivatives as potent and selective PTPlB inhibitors.
    Lei S; Zhang D; Qi Y; Chowdhury SR; Sun R; Wang J; Du Y; Fu L; Jiang F
    Eur J Med Chem; 2020 Nov; 205():112508. PubMed ID: 32738350
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Identification of lipid-like salicylic acid-based derivatives as potent and membrane-permeable PTP1B inhibitors.
    Li L; Tavallaie MS; Xie F; Xia Y; Liang Y; Jiang F; Fu L
    Bioorg Chem; 2019 Dec; 93():103296. PubMed ID: 31585268
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Investigation of stereoisomeric bisarylethenesulfonic acid esters for discovering potent and selective PTP1B inhibitors.
    Xie F; Yang F; Liang Y; Li L; Xia Y; Jiang F; Liu W; Qi Y; Chowdhury SR; Xie D; Fu L
    Eur J Med Chem; 2019 Feb; 164():408-422. PubMed ID: 30611982
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Identification of 2-substituted ethenesulfonic acid ester derivatives as novel, potent and selective inhibitors of protein tyrosine phosphatase 1B.
    Deng X; Liu J; Jin Y; Zhang Y; He W; Bao J; Liu W; Jiang F; Fu L
    Pharmazie; 2015 Dec; 70(12):777-83. PubMed ID: 26817274
    [TBL] [Abstract][Full Text] [Related]  

  • 7. [Design, synthesis and evaluation of malonic acid-based PTP1B inhibitors].
    Du X; Zhang SE; Liu JZ; Nie FL; Ye F; Tian JY; Xiao ZY
    Yao Xue Xue Bao; 2012 Mar; 47(3):367-73. PubMed ID: 22645761
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design, synthesis and in vitro activity of phidianidine B derivatives as novel PTP1B inhibitors with specific selectivity.
    Zhang L; Jiang CS; Gao LX; Gong JX; Wang ZH; Li JY; Li J; Li XW; Guo YW
    Bioorg Med Chem Lett; 2016 Feb; 26(3):778-781. PubMed ID: 26774579
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel, potent, selective and cellular active ABC type PTP1B inhibitors containing (methanesulfonyl-phenyl-amino)-acetic acid methyl ester phosphotyrosine mimetic.
    Liu P; Du Y; Song L; Shen J; Li Q
    Bioorg Med Chem; 2015 Nov; 23(21):7079-88. PubMed ID: 26481657
    [TBL] [Abstract][Full Text] [Related]  

  • 10. The development of protein tyrosine phosphatase1B inhibitors defined by binding sites in crystalline complexes.
    Zhang Y; Du Y
    Future Med Chem; 2018 Oct; 10(19):2345-2367. PubMed ID: 30273014
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Novel thiophene derivatives as PTP1B inhibitors with selectivity and cellular activity.
    Ye D; Zhang Y; Wang F; Zheng M; Zhang X; Luo X; Shen X; Jiang H; Liu H
    Bioorg Med Chem; 2010 Mar; 18(5):1773-82. PubMed ID: 20153651
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis and biological evaluation of uncharged catechol derivatives as selective inhibitors of PTP1B.
    Li XQ; Xu Q; Luo J; Wang LJ; Jiang B; Zhang RS; Shi DY
    Eur J Med Chem; 2017 Aug; 136():348-359. PubMed ID: 28511130
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Benzo[c][1,2,5]thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
    Wang WL; Chen XY; Gao Y; Gao LX; Sheng L; Zhu J; Xu L; Ding ZZ; Zhang C; Li JY; Li J; Zhou YB
    Bioorg Med Chem Lett; 2017 Dec; 27(23):5154-5157. PubMed ID: 29100798
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Discovery of novel, high potent, ABC type PTP1B inhibitors with TCPTP selectivity and cellular activity.
    Liu P; Du Y; Song L; Shen J; Li Q
    Eur J Med Chem; 2016 Aug; 118():27-33. PubMed ID: 27123900
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors.
    Wang WL; Huang C; Gao LX; Tang CL; Wang JQ; Wu MC; Sheng L; Chen HJ; Nan FJ; Li JY; Li J; Feng B
    Bioorg Med Chem Lett; 2014 Apr; 24(8):1889-94. PubMed ID: 24684845
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and biological evaluation of novel N-aryl-ω-(benzoazol-2-yl)-sulfanylalkanamides as dual inhibitors of α-glucosidase and protein tyrosine phosphatase 1B.
    Wang MY; Cheng XC; Chen XB; Li Y; Zang LL; Duan YQ; Chen MZ; Yu P; Sun H; Wang RL
    Chem Biol Drug Des; 2018 Sep; 92(3):1647-1656. PubMed ID: 29745030
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Characterization of the inhibitory activity of natural tanshinones from Salvia miltiorrhiza roots on protein tyrosine phosphatase 1B.
    Kim DH; Paudel P; Yu T; Ngo TM; Kim JA; Jung HA; Yokozawa T; Choi JS
    Chem Biol Interact; 2017 Dec; 278():65-73. PubMed ID: 29031618
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Discovery and evaluation of the hybrid of bromophenol and saccharide as potent and selective protein tyrosine phosphatase 1B inhibitors.
    Zhang R; Yu R; Xu Q; Li X; Luo J; Jiang B; Wang L; Guo S; Wu N; Shi D
    Eur J Med Chem; 2017 Jul; 134():24-33. PubMed ID: 28395151
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Discovery of 2-ethoxy-4-(methoxymethyl)benzamide derivatives as potent and selective PTP1B inhibitors.
    Xie F; Liang Y; Xia Y; Luo S; Jiang F; Fu L
    Bioorg Chem; 2019 Nov; 92():103273. PubMed ID: 31539748
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design, synthesis and docking study of 5-(substituted benzylidene)thiazolidine-2,4-dione derivatives as inhibitors of protein tyrosine phosphatase 1B.
    Wang Z; Liu Z; Lee W; Kim SN; Yoon G; Cheon SH
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3337-40. PubMed ID: 24953600
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 13.