BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

105 related articles for article (PubMed ID: 28400239)

  • 1. Efficient synthesis of a multi-substituted diphenylmethane skeleton as a steroid mimetic.
    Misawa T; Tanaka K; Demizu Y; Kurihara M
    Bioorg Med Chem Lett; 2017 Jun; 27(11):2590-2593. PubMed ID: 28400239
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Structure-activity relationships of bisphenol A analogs at estrogen receptors (ERs): discovery of an ERα-selective antagonist.
    Maruyama K; Nakamura M; Tomoshige S; Sugita K; Makishima M; Hashimoto Y; Ishikawa M
    Bioorg Med Chem Lett; 2013 Jul; 23(14):4031-6. PubMed ID: 23768907
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Structure-activity relationship study of estrogen receptor down-regulators with a diphenylmethane skeleton.
    Nanjyo S; Ohgane K; Yoshioka H; Makishima M; Hashimoto Y; Noguchi-Yachide T
    Bioorg Med Chem; 2019 May; 27(10):1952-1961. PubMed ID: 30940565
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Development of Photoswitchable Estrogen Receptor Ligands.
    Tsuchiya K; Umeno T; Tsuji G; Yokoo H; Tanaka M; Fukuhara K; Demizu Y; Misawa T
    Chem Pharm Bull (Tokyo); 2020; 68(4):398-402. PubMed ID: 32238658
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Diphenylmethane skeleton as a multi-template for nuclear receptor ligands: preparation of FXR and PPAR ligands.
    Kainuma M; Kasuga J; Hosoda S; Wakabayashi K; Tanatani A; Nagasawa K; Miyachi H; Makishima M; Hashimoto Y
    Bioorg Med Chem Lett; 2006 Jun; 16(12):3213-8. PubMed ID: 16617018
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Symmetric 4,4'-(piperidin-4-ylidenemethylene)bisphenol derivatives as novel tunable estrogen receptor (ER) modulators.
    Sato M; Ohta K; Kaise A; Aoto S; Endo Y
    Bioorg Med Chem; 2016 Mar; 24(5):1089-94. PubMed ID: 26822566
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design and synthesis of silicon-containing steroid sulfatase inhibitors possessing pro-estrogen antagonistic character.
    Kajita D; Nakamura M; Matsumoto Y; Makishima M; Hashimoto Y
    Bioorg Med Chem; 2014 Apr; 22(7):2244-52. PubMed ID: 24630694
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Structure-based approach for the discovery of novel selective estrogen receptor modulators.
    Rosano C; Stec-Martyna E; Lappano R; Maggiolini M
    Curr Med Chem; 2011; 18(8):1188-94. PubMed ID: 21291367
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and binding affinities of fluoroalkylated raloxifenes.
    Lee KC; Moon BS; Lee JH; Chung KH; Katzenellenbogen JA; Chi DY
    Bioorg Med Chem; 2003 Aug; 11(17):3649-58. PubMed ID: 12901910
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Tetrahydroquinoline-based selective estrogen receptor modulators (SERMs).
    Wallace OB; Lauwers KS; Jones SA; Dodge JA
    Bioorg Med Chem Lett; 2003 Jun; 13(11):1907-10. PubMed ID: 12749895
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Estrogenic activity of bis(4-hydroxyphenyl)methanes with cyclic hydrophobic structure.
    Kojima T; Ogawa T; Kitao S; Sato M; Oda A; Ohta K; Endo Y
    Bioorg Med Chem; 2015 Nov; 23(21):6900-11. PubMed ID: 26462053
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Estrogen receptor ligands. Part 3: The SAR of dihydrobenzoxathiin SERMs.
    Chen HY; Kim S; Wu JY; Birzin ET; Chan W; Yang YT; Dahllund J; DiNinno F; Rohrer SP; Schaeffer JM; Hammond ML
    Bioorg Med Chem Lett; 2004 May; 14(10):2551-4. PubMed ID: 15109649
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Rapid synthesis of 4-benzylidene and 4-[bis-(4-methoxyphenyl)-methylene-2-substituted phenyl-benzopyrans as potential selective estrogen receptor modulators (SERMs) using McMurry coupling reaction.
    Gupta A; Dwivedy A; Keshri G; Sharma R; Balapure AK; Singh MM; Ray S
    Bioorg Med Chem Lett; 2006 Dec; 16(23):6006-12. PubMed ID: 16979337
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Discovery and structure-activity analysis of selective estrogen receptor modulators via similarity-based virtual screening.
    Shen J; Jiang J; Kuang G; Tan C; Liu G; Huang J; Tang Y
    Eur J Med Chem; 2012 Aug; 54():188-96. PubMed ID: 22647217
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Discovery of diphenylmethane analogs as anti-bovine diarrhea viral agents.
    Hosoda S; Aoyama H; Goto Y; Salim MT; Okamoto M; Hashimoto M; Baba M; Hashimoto Y
    Bioorg Med Chem Lett; 2009 Jun; 19(12):3157-61. PubMed ID: 19447037
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis of 4,4'-Diaminotriphenylmethanes with Potential Selective Estrogen Receptor Modulator (SERM)-like Activity.
    Guedes G; Amesty Á; Jiménez-Monzón R; Marrero-Alonso J; Díaz M; Fernández-Pérez L; Estévez-Braun A
    ChemMedChem; 2015 Aug; 10(8):1403-12. PubMed ID: 26076185
    [TBL] [Abstract][Full Text] [Related]  

  • 17. New scaffolds for the design of selective estrogen receptor modulators.
    Martín-Santamaría S; Rodríguez JJ; de Pascual-Teresa S; Gordon S; Bengtsson M; Garrido-Laguna I; Rubio-Viqueira B; López-Casas PP; Hidalgo M; de Pascual-Teresa B; Ramos A
    Org Biomol Chem; 2008 Oct; 6(19):3486-96. PubMed ID: 19082149
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Estrogen receptor ligands. Part 6: Synthesis and binding affinity of dihydrobenzodithiins.
    Tan Q; Birzin ET; Chan W; Yang YT; Pai LY; Hayes EC; DaSilva CA; DiNinno F; Rohrer SP; Schaeffer JM; Hammond ML
    Bioorg Med Chem Lett; 2004 Jul; 14(14):3753-5. PubMed ID: 15203156
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Estrogen to antiestrogen with a single methylene group resulting in an unusual steroidal selective estrogen receptor modulator.
    Zhang JX; Labaree DC; Mor G; Hochberg RB
    J Clin Endocrinol Metab; 2004 Jul; 89(7):3527-35. PubMed ID: 15240642
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Antagonists selective for estrogen receptor alpha.
    Sun J; Huang YR; Harrington WR; Sheng S; Katzenellenbogen JA; Katzenellenbogen BS
    Endocrinology; 2002 Mar; 143(3):941-7. PubMed ID: 11861516
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.