BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

199 related articles for article (PubMed ID: 28407766)

  • 1. Novel lead structures with both Plasmodium falciparum gametocytocidal and asexual blood stage activity identified from high throughput compound screening.
    Sun W; Huang X; Li H; Tawa G; Fisher E; Tanaka TQ; Shinn P; Huang W; Williamson KC; Zheng W
    Malar J; 2017 Apr; 16(1):147. PubMed ID: 28407766
    [TBL] [Abstract][Full Text] [Related]  

  • 2. A quantitative high throughput assay for identifying gametocytocidal compounds.
    Tanaka TQ; Dehdashti SJ; Nguyen DT; McKew JC; Zheng W; Williamson KC
    Mol Biochem Parasitol; 2013 Mar; 188(1):20-5. PubMed ID: 23454872
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials.
    van der Watt ME; Reader J; Churchyard A; Nondaba SH; Lauterbach SB; Niemand J; Abayomi S; van Biljon RA; Connacher JI; van Wyk RDJ; Le Manach C; Paquet T; González Cabrera D; Brunschwig C; Theron A; Lozano-Arias S; Rodrigues JFI; Herreros E; Leroy D; Duffy J; Street LJ; Chibale K; Mancama D; Coetzer TL; Birkholtz LM
    J Antimicrob Chemother; 2018 May; 73(5):1279-1290. PubMed ID: 29420756
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Potent Plasmodium falciparum gametocytocidal activity of diaminonaphthoquinones, lead antimalarial chemotypes identified in an antimalarial compound screen.
    Tanaka TQ; Guiguemde WA; Barnett DS; Maron MI; Min J; Connelly MC; Suryadevara PK; Guy RK; Williamson KC
    Antimicrob Agents Chemother; 2015 Mar; 59(3):1389-97. PubMed ID: 25512421
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Identification of inhibitors of Plasmodium falciparum gametocyte development.
    Duffy S; Avery VM
    Malar J; 2013 Nov; 12():408. PubMed ID: 24206914
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Identification of MMV malaria box inhibitors of plasmodium falciparum early-stage gametocytes using a luciferase-based high-throughput assay.
    Lucantoni L; Duffy S; Adjalley SH; Fidock DA; Avery VM
    Antimicrob Agents Chemother; 2013 Dec; 57(12):6050-62. PubMed ID: 24060871
    [TBL] [Abstract][Full Text] [Related]  

  • 7. A randomized feasibility trial comparing four antimalarial drug regimens to induce
    Reuling IJ; van de Schans LA; Coffeng LE; Lanke K; Meerstein-Kessel L; Graumans W; van Gemert GJ; Teelen K; Siebelink-Stoter R; van de Vegte-Bolmer M; de Mast Q; van der Ven AJ; Ivinson K; Hermsen CC; de Vlas S; Bradley J; Collins KA; Ockenhouse CF; McCarthy J; Sauerwein RW; Bousema T
    Elife; 2018 Feb; 7():. PubMed ID: 29482720
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Chemoprotective antimalarials identified through quantitative high-throughput screening of Plasmodium blood and liver stage parasites.
    Dorjsuren D; Eastman RT; Wicht KJ; Jansen D; Talley DC; Sigmon BA; Zakharov AV; Roncal N; Girvin AT; Antonova-Koch Y; Will PM; Shah P; Sun H; Klumpp-Thomas C; Mok S; Yeo T; Meister S; Marugan JJ; Ross LS; Xu X; Maloney DJ; Jadhav A; Mott BT; Sciotti RJ; Winzeler EA; Waters NC; Campbell RF; Huang W; Simeonov A; Fidock DA
    Sci Rep; 2021 Jan; 11(1):2121. PubMed ID: 33483532
    [TBL] [Abstract][Full Text] [Related]  

  • 9. In vitro evaluation of imidazo[4,5-c]quinolin-2-ones as gametocytocidal antimalarial agents.
    Patel PR; Sun W; Kim M; Huang X; Sanderson PE; Tanaka TQ; McKew JC; Simeonov A; Williamson KC; Zheng W; Huang W
    Bioorg Med Chem Lett; 2016 Jun; 26(12):2907-2911. PubMed ID: 27156776
    [TBL] [Abstract][Full Text] [Related]  

  • 10. A New Set of Chemical Starting Points with Plasmodium falciparum Transmission-Blocking Potential for Antimalarial Drug Discovery.
    Almela MJ; Lozano S; Lelièvre J; Colmenarejo G; Coterón JM; Rodrigues J; Gonzalez C; Herreros E
    PLoS One; 2015; 10(8):e0135139. PubMed ID: 26317851
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials.
    Abraham M; Gagaring K; Martino ML; Vanaerschot M; Plouffe DM; Calla J; Godinez-Macias KP; Du AY; Wree M; Antonova-Koch Y; Eribez K; Luth MR; Ottilie S; Fidock DA; McNamara CW; Winzeler EA
    ACS Infect Dis; 2020 Apr; 6(4):613-628. PubMed ID: 32078764
    [TBL] [Abstract][Full Text] [Related]  

  • 12. A Plasmodium falciparum screening assay for anti-gametocyte drugs based on parasite lactate dehydrogenase detection.
    D'Alessandro S; Silvestrini F; Dechering K; Corbett Y; Parapini S; Timmerman M; Galastri L; Basilico N; Sauerwein R; Alano P; Taramelli D
    J Antimicrob Chemother; 2013 Sep; 68(9):2048-58. PubMed ID: 23645588
    [TBL] [Abstract][Full Text] [Related]  

  • 13. A novel validated assay to support the discovery of new anti-malarial gametocytocidal agents.
    Bahamontes-Rosa N; Gomez-Lorenzo MG; Lelièvre J; Rodriguez Alejandre A; Almela MJ; Lozano S; Herreros E; Gamo FJ
    Malar J; 2016 Jul; 15(1):385. PubMed ID: 27448565
    [TBL] [Abstract][Full Text] [Related]  

  • 14. A novel approach for the discovery of chemically diverse anti-malarial compounds targeting the Plasmodium falciparum Coenzyme A synthesis pathway.
    Fletcher S; Avery VM
    Malar J; 2014 Aug; 13():343. PubMed ID: 25174342
    [TBL] [Abstract][Full Text] [Related]  

  • 15. High-Throughput Assay and Discovery of Small Molecules that Interrupt Malaria Transmission.
    Plouffe DM; Wree M; Du AY; Meister S; Li F; Patra K; Lubar A; Okitsu SL; Flannery EL; Kato N; Tanaseichuk O; Comer E; Zhou B; Kuhen K; Zhou Y; Leroy D; Schreiber SL; Scherer CA; Vinetz J; Winzeler EA
    Cell Host Microbe; 2016 Jan; 19(1):114-26. PubMed ID: 26749441
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Maduramicin Rapidly Eliminates Malaria Parasites and Potentiates the Gametocytocidal Activity of the Pyrazoleamide PA21A050.
    Maron MI; Magle CT; Czesny B; Turturice BA; Huang R; Zheng W; Vaidya AB; Williamson KC
    Antimicrob Agents Chemother; 2015 Dec; 60(3):1492-9. PubMed ID: 26711768
    [TBL] [Abstract][Full Text] [Related]  

  • 17. In vitro inhibition of Plasmodium falciparum early and late stage gametocyte viability by extracts from eight traditionally used South African plant species.
    Moyo P; Botha ME; Nondaba S; Niemand J; Maharaj VJ; Eloff JN; Louw AI; Birkholtz L
    J Ethnopharmacol; 2016 Jun; 185():235-42. PubMed ID: 26994818
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Luciferase-Based, High-Throughput Assay for Screening and Profiling Transmission-Blocking Compounds against Plasmodium falciparum Gametocytes.
    Lucantoni L; Fidock DA; Avery VM
    Antimicrob Agents Chemother; 2016 Apr; 60(4):2097-107. PubMed ID: 26787698
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria elimination.
    Reader J; Botha M; Theron A; Lauterbach SB; Rossouw C; Engelbrecht D; Wepener M; Smit A; Leroy D; Mancama D; Coetzer TL; Birkholtz LM
    Malar J; 2015 May; 14():213. PubMed ID: 25994518
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Gametocyte-specific and all-blood-stage transmission-blocking chemotypes discovered from high throughput screening on Plasmodium falciparum gametocytes.
    Paonessa G; Siciliano G; Graziani R; Lalli C; Cecchetti O; Alli C; La Valle R; Petrocchi A; Sferrazza A; Bisbocci M; Falchi M; Toniatti C; Bresciani A; Alano P
    Commun Biol; 2022 Jun; 5(1):547. PubMed ID: 35668202
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.