These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
2. Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin α Raposo Moreira Dias A; Pina A; Dal Corso A; Arosio D; Belvisi L; Pignataro L; Caruso M; Gennari C Chemistry; 2017 Oct; 23(58):14410-14415. PubMed ID: 28816404 [TBL] [Abstract][Full Text] [Related]
3. Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers. Dal Corso A; Caruso M; Belvisi L; Arosio D; Piarulli U; Albanese C; Gasparri F; Marsiglio A; Sola F; Troiani S; Valsasina B; Pignataro L; Donati D; Gennari C Chemistry; 2015 Apr; 21(18):6921-9. PubMed ID: 25784522 [TBL] [Abstract][Full Text] [Related]
4. Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α Raposo Moreira Dias A; Bodero L; Martins A; Arosio D; Gazzola S; Belvisi L; Pignataro L; Steinkühler C; Dal Corso A; Gennari C; Piarulli U ChemMedChem; 2019 May; 14(9):938-942. PubMed ID: 30840356 [TBL] [Abstract][Full Text] [Related]
5. Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate. Raposo Moreira Dias A; Pina A; Dean A; Lerchen HG; Caruso M; Gasparri F; Fraietta I; Troiani S; Arosio D; Belvisi L; Pignataro L; Dal Corso A; Gennari C Chemistry; 2019 Feb; 25(7):1696-1700. PubMed ID: 30452790 [TBL] [Abstract][Full Text] [Related]
6. RGD Peptidomimetic MMAE-Conjugate Addressing Integrin αVβ3-Expressing Cells with High Targeting Index. Paulus J; Nachtigall B; Meyer P; Sewald N Chemistry; 2023 Feb; 29(12):e202203476. PubMed ID: 36454662 [TBL] [Abstract][Full Text] [Related]
7. Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists. Panzeri S; Zanella S; Arosio D; Vahdati L; Dal Corso A; Pignataro L; Paolillo M; Schinelli S; Belvisi L; Gennari C; Piarulli U Chemistry; 2015 Apr; 21(16):6265-71. PubMed ID: 25761230 [TBL] [Abstract][Full Text] [Related]
8. Cyclic RGD and Panzeri S; Arosio D; Gazzola S; Belvisi L; Civera M; Potenza D; Vasile F; Kemker I; Ertl T; Sewald N; Reiser O; Piarulli U Molecules; 2020 Dec; 25(24):. PubMed ID: 33339382 [TBL] [Abstract][Full Text] [Related]
9. Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting. Bodero L; López Rivas P; Korsak B; Hechler T; Pahl A; Müller C; Arosio D; Pignataro L; Gennari C; Piarulli U Beilstein J Org Chem; 2018; 14():407-415. PubMed ID: 29520305 [TBL] [Abstract][Full Text] [Related]
10. Multimeric Presentation of RGD Peptidomimetics Enhances Integrin Binding and Tumor Cell Uptake. Pina A; Kadri M; Arosio D; Dal Corso A; Coll JL; Gennari C; Boturyn D Chemistry; 2020 Jun; 26(33):7492-7496. PubMed ID: 32227540 [TBL] [Abstract][Full Text] [Related]
11. Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine-glycine-aspartate (RGD) peptidomimetic-paclitaxel conjugates targeting integrin αVβ3. Colombo R; Mingozzi M; Belvisi L; Arosio D; Piarulli U; Carenini N; Perego P; Zaffaroni N; De Cesare M; Castiglioni V; Scanziani E; Gennari C J Med Chem; 2012 Dec; 55(23):10460-74. PubMed ID: 23140358 [TBL] [Abstract][Full Text] [Related]
12. High-Affinity "Click" RGD Peptidomimetics as Radiolabeled Probes for Imaging α Piras M; Testa A; Fleming IN; Dall'Angelo S; Andriu A; Menta S; Mori M; Brown GD; Forster D; Williams KJ; Zanda M ChemMedChem; 2017 Jul; 12(14):1142-1151. PubMed ID: 28608961 [TBL] [Abstract][Full Text] [Related]
13. Integrin-targeted nano-sized polymeric systems for paclitaxel conjugation: a comparative study. Eldar-Boock A; Blau R; Ryppa C; Baabur-Cohen H; Many A; Vicent MJ; Kratz F; Sanchis J; Satchi-Fainaro R J Drug Target; 2017; 25(9-10):829-844. PubMed ID: 28737432 [TBL] [Abstract][Full Text] [Related]
14. Conjugates of Cryptophycin and RGD or Borbély A; Figueras E; Martins A; Bodero L; Raposo Moreira Dias A; López Rivas P; Pina A; Arosio D; Gallinari P; Frese M; Steinkühler C; Gennari C; Piarulli U; Sewald N ChemistryOpen; 2019 Jun; 8(6):737-742. PubMed ID: 31275795 [TBL] [Abstract][Full Text] [Related]
15. Liposomes actively recognizing the glucose transporter GLUT Fu Q; Zhao Y; Yang Z; Yue Q; Xiao W; Chen Y; Yang Y; Guo L; Wu Y Arch Pharm (Weinheim); 2019 Feb; 352(2):e1800219. PubMed ID: 30609116 [TBL] [Abstract][Full Text] [Related]
16. Synthesis and biological evaluation of dimeric RGD peptide-paclitaxel conjugate as a model for integrin-targeted drug delivery. Chen X; Plasencia C; Hou Y; Neamati N J Med Chem; 2005 Feb; 48(4):1098-106. PubMed ID: 15715477 [TBL] [Abstract][Full Text] [Related]
17. Integrin-assisted drug delivery of nano-scaled polymer therapeutics bearing paclitaxel. Eldar-Boock A; Miller K; Sanchis J; Lupu R; Vicent MJ; Satchi-Fainaro R Biomaterials; 2011 May; 32(15):3862-74. PubMed ID: 21376390 [TBL] [Abstract][Full Text] [Related]