BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

169 related articles for article (PubMed ID: 28456031)

  • 1. Identification of thiazolo[5,4-d]pyrimidine derivatives as potent antiproliferative agents through the drug repurposing strategy.
    Li ZH; Zhang J; Liu XQ; Geng PF; Ma JL; Wang B; Zhao TQ; Zhao B; Wei HM; Wang C; Fu DJ; Yu B; Liu HM
    Eur J Med Chem; 2017 Jul; 135():204-212. PubMed ID: 28456031
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design, synthesis and antiproliferative activity of thiazolo[5,4-d]pyrimidine derivatives through the atom replacement strategy.
    Li ZH; Liu XQ; Geng PF; Zhang J; Ma JL; Wang B; Zhao TQ; Zhao B; Zhang XH; Yu B; Liu HM
    Eur J Med Chem; 2017 Sep; 138():1034-1041. PubMed ID: 28759876
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis, antiproliferative and apoptosis-inducing activity of thiazolo[5,4-d]pyrimidines.
    Singh B; Guru SK; Kour S; Jain SK; Sharma R; Sharma PR; Singh SK; Bhushan S; Bharate SB; Vishwakarma RA
    Eur J Med Chem; 2013; 70():864-74. PubMed ID: 24262379
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design, synthesis and biological evaluation of [1,2,3]triazolo[4,5-d]pyrimidine derivatives possessing a hydrazone moiety as antiproliferative agents.
    Li ZH; Yang DX; Geng PF; Zhang J; Wei HM; Hu B; Guo Q; Zhang XH; Guo WG; Zhao B; Yu B; Ma LY; Liu HM
    Eur J Med Chem; 2016 Nov; 124():967-980. PubMed ID: 27771599
    [TBL] [Abstract][Full Text] [Related]  

  • 5. A Facile and Microwave-assisted Rapid Synthesis of 2-Arylamino-4-(3'-indolyl)- thiazoles as Apoptosis Inducing Cytotoxic Agents.
    Tantak MP; Mukherjee DD; Kumar A; Chakrabarti G; Kumar D
    Anticancer Agents Med Chem; 2017; 17(3):442-455. PubMed ID: 27338299
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Design, synthesis and in vitro biological evaluation of novel [1,2,3]triazolo[4,5-d]pyrimidine derivatives containing a thiosemicarbazide moiety.
    Geng PF; Liu XQ; Zhao TQ; Wang CC; Li ZH; Zhang J; Wei HM; Hu B; Ma LY; Liu HM
    Eur J Med Chem; 2018 Feb; 146():147-156. PubMed ID: 29407946
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Phenyl and Diaryl Ureas with Thiazolo[5,4-d]pyrimidine Scaffold as Angiogenesis Inhibitors: Design, Synthesis and Biological Evaluation.
    Xue WJ; Deng YH; Yan ZH; Liu JP; Liu Y; Sun LP
    Chem Biodivers; 2019 Apr; 16(4):e1800493. PubMed ID: 30688404
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Substituted thiazoles V. synthesis and antitumor activity of novel thiazolo[2,3-b]quinazoline and pyrido[4,3-d]thiazolo[3,2-a]pyrimidine analogues.
    Al-Omary FA; Hassan GS; El-Messery SM; El-Subbagh HI
    Eur J Med Chem; 2012 Jan; 47(1):65-72. PubMed ID: 22056277
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and biological evaluation of 4-amino-5-cinnamoylthiazoles as chalcone-like anticancer agents.
    Ayati A; Esmaeili R; Moghimi S; Oghabi Bakhshaiesh T; Eslami-S Z; Majidzadeh-A K; Safavi M; Emami S; Foroumadi A
    Eur J Med Chem; 2018 Feb; 145():404-412. PubMed ID: 29335206
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design and synthesis of novel DFG-out RAF/vascular endothelial growth factor receptor 2 (VEGFR2) inhibitors: 3. Evaluation of 5-amino-linked thiazolo[5,4-d]pyrimidine and thiazolo[5,4-b]pyridine derivatives.
    Hirose M; Okaniwa M; Miyazaki T; Imada T; Ohashi T; Tanaka Y; Arita T; Yabuki M; Kawamoto T; Tsutsumi S; Sumita A; Takagi T; Sang BC; Yano J; Aertgeerts K; Yoshida S; Ishikawa T
    Bioorg Med Chem; 2012 Sep; 20(18):5600-15. PubMed ID: 22883026
    [TBL] [Abstract][Full Text] [Related]  

  • 11. An investigative study of antitumor properties of a novel thiazolo[4,5-d]pyrimidine small molecule revealing superior antitumor activity with CDK1 selectivity and potent pro-apoptotic properties.
    Mohamed SH; Elgiushy HR; Taha H; Hammad SF; Abou-Taleb NA; A M Abouzid K; Al-Sawaf H; Hassan Z
    Bioorg Med Chem; 2020 Sep; 28(17):115633. PubMed ID: 32773088
    [TBL] [Abstract][Full Text] [Related]  

  • 12. One-pot synthesis of new (1,3-thiazolo[5,4-b]pyridin-2-yl)benzenediols and their antiproliferative activities against human cancer cell lines.
    Matysiak J; Karpińska MM; Niewiadomy A; Wietrzyk J; Kłopotowska D
    Chem Biodivers; 2012 Jan; 9(1):48-57. PubMed ID: 22253102
    [TBL] [Abstract][Full Text] [Related]  

  • 13. One-pot synthesis of thiazolo[3,2-a]pyrimidine derivatives, their cytotoxic evaluation and molecular docking studies.
    Sekhar T; Thriveni P; Venkateswarlu A; Daveedu T; Peddanna K; Sainath SB
    Spectrochim Acta A Mol Biomol Spectrosc; 2020 Apr; 231():118056. PubMed ID: 32006911
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Design, synthesis, and in vitro antiproliferative activity of novel Dasatinib derivatives.
    Cai J; Zhang S; Zheng M; Wu X; Chen J; Ji M
    Bioorg Med Chem Lett; 2012 Jan; 22(2):806-10. PubMed ID: 22217877
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Novel 3-(2,6,9-trisubstituted-9H-purine)-8-chalcone derivatives as potent anti-gastric cancer agents: Design, synthesis and structural optimization.
    Zhao TQ; Zhao YD; Liu XY; Li ZH; Wang B; Zhang XH; Cao YQ; Ma LY; Liu HM
    Eur J Med Chem; 2019 Jan; 161():493-505. PubMed ID: 30388465
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Drug repurposing: Discovery of troxipide analogs as potent antitumor agents.
    Lu N; Huo JL; Wang S; Yuan XH; Liu HM
    Eur J Med Chem; 2020 Sep; 202():112471. PubMed ID: 32619887
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis, anticancer activity and effects on cell cycle profile and apoptosis of novel thieno[2,3-d]pyrimidine and thieno[3,2-e] triazolo[4,3-c]pyrimidine derivatives.
    Kandeel MM; Refaat HM; Kassab AE; Shahin IG; Abdelghany TM
    Eur J Med Chem; 2015 Jan; 90():620-32. PubMed ID: 25499930
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Thienopyrimidine derivatives exert their anticancer efficacy via apoptosis induction, oxidative stress and mitotic catastrophe.
    Amawi H; Karthikeyan C; Pathak R; Hussein N; Christman R; Robey R; Ashby CR; Trivedi P; Malhotra A; Tiwari AK
    Eur J Med Chem; 2017 Sep; 138():1053-1065. PubMed ID: 28759878
    [TBL] [Abstract][Full Text] [Related]  

  • 19. One-Pot Synthesis of Novel Thiazoles as Potential Anti-Cancer Agents.
    Sayed AR; Gomha SM; Taher EA; Muhammad ZA; El-Seedi HR; Gaber HM; Ahmed MM
    Drug Des Devel Ther; 2020; 14():1363-1375. PubMed ID: 32308369
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Indolylmethylene benzo[h]thiazolo[2,3-b]quinazolinones: synthesis, characterization and evaluation of anticancer and antimicrobial activities.
    Gali R; Banothu J; Porika M; Velpula R; Hnamte S; Bavantula R; Abbagani S; Busi S
    Bioorg Med Chem Lett; 2014 Sep; 24(17):4239-42. PubMed ID: 25096298
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 9.