BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

307 related articles for article (PubMed ID: 28480832)

  • 1. Synthesis of New Arylidene 2,5-Diketopiperazines and Evaluation of their Anti-Acetylcholinesterase, Anti-xanthine Oxidase, Anti-diabetic and Cytotoxic Activities.
    Belkacem MA; Jannet HB; Ferhout H; Mzali L; Bouajila J
    Med Chem; 2017; 13(8):744-752. PubMed ID: 28480832
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and activity evaluation of the cyclic dipeptides arylidene N-alkoxydiketopiperazines.
    Tian X; Feng J; Fan SM; Zhen XL; Han JR; Liu SX
    Bioorg Med Chem; 2016 Nov; 24(21):5197-5205. PubMed ID: 27594550
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Design, synthesis of novel pyranotriazolopyrimidines and evaluation of their anti-soybean lipoxygenase, anti-xanthine oxidase, and cytotoxic activities.
    Saïd AB; Romdhane A; Elie N; Touboul D; Jannet HB; Bouajila J
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):1277-85. PubMed ID: 26681513
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Trisubstituted barbiturates and thiobarbiturates: Synthesis and biological evaluation as xanthine oxidase inhibitors, antioxidants, antibacterial and anti-proliferative agents.
    Figueiredo J; Serrano JL; Cavalheiro E; Keurulainen L; Yli-Kauhaluoma J; Moreira VM; Ferreira S; Domingues FC; Silvestre S; Almeida P
    Eur J Med Chem; 2018 Jan; 143():829-842. PubMed ID: 29223098
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design, synthesis and cytotoxic activities of novel 2,5-diketopiperazine derivatives.
    Liao SR; Qin XC; Wang Z; Li D; Xu L; Li JS; Tu ZC; Liu Y
    Eur J Med Chem; 2016 Oct; 121():500-509. PubMed ID: 27318124
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis, cytotoxic, anti-lipoxygenase and anti-acetylcholinesterase capacities of novel derivatives from harmine.
    Filali I; Belkacem MA; Ben Nejma A; Souchard JP; Ben Jannet H; Bouajila J
    J Enzyme Inhib Med Chem; 2016; 31(sup1):23-33. PubMed ID: 27028352
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Discovery of diethyl 2,5-diaminothiophene-3,4-dicarboxylate derivatives as potent anticancer and antimicrobial agents and screening of anti-diabetic activity: synthesis and in vitro biological evaluation. Part 1.
    Bozorov K; Ma HR; Zhao JY; Zhao HQ; Chen H; Bobakulov K; Xin XL; Elmuradov B; Shakhidoyatov K; Aisa HA
    Eur J Med Chem; 2014 Sep; 84():739-45. PubMed ID: 25064350
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and Evaluation of a New Series of Arylidene Indanones as Potential Anticancer Agents.
    Özdemir A; Gökbulut S; Sever B; Çiftçi GA; Altıntop MD
    Anticancer Agents Med Chem; 2018; 18(10):1394-1404. PubMed ID: 29210665
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis, biological evaluation and molecular docking studies of bis-chalcone derivatives as xanthine oxidase inhibitors and anticancer agents.
    Burmaoglu S; Ozcan S; Balcioglu S; Gencel M; Noma SAA; Essiz S; Ates B; Algul O
    Bioorg Chem; 2019 Oct; 91():103149. PubMed ID: 31382060
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Development of novel phenoxy-diketopiperazine-type plinabulin derivatives as potent antimicrotubule agents based on the co-crystal structure.
    Ding Z; Ma M; Zhong C; Wang S; Fu Z; Hou Y; Liu Y; Zhong L; Chu Y; Li F; Song C; Wang Y; Yang J; Li W
    Bioorg Med Chem; 2020 Jan; 28(1):115186. PubMed ID: 31759826
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis of new isoxazoline derivatives from harmine and evaluation of their anti-Alzheimer, anti-cancer and anti-inflammatory activities.
    Filali I; Bouajila J; Znati M; Bousejra-El Garah F; Ben Jannet H
    J Enzyme Inhib Med Chem; 2015 Jun; 30(3):371-6. PubMed ID: 25068731
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of novel diazaphosphinanes coumarin derivatives with promoted cytotoxic and anti-tyrosinase activities.
    Gardelly M; Trimech B; Belkacem MA; Harbach M; Abdelwahed S; Mosbah A; Bouajila J; Ben Jannet H
    Bioorg Med Chem Lett; 2016 May; 26(10):2450-2454. PubMed ID: 27080182
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and bioactivity of diketopiperazine PJ147 and its derivatives from Gliocladium sp. YUP08.
    Li XZ; Chen G; Wang HF; Hua HM; Pei YH
    J Asian Nat Prod Res; 2014; 16(7):764-9. PubMed ID: 24827395
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Saroclazines A-C, thio-diketopiperazines from mangrove-derived fungi Sarocladium kiliense HDN11-84.
    Li F; Guo W; Wu L; Zhu T; Gu Q; Li D; Che Q
    Arch Pharm Res; 2018 Jan; 41(1):30-34. PubMed ID: 29103141
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Pharmacological Evaluation of Aldehydic-Pyrrolidinedione Against HCT-116, MDA-MB231, NIH/3T3, MCF-7 Cancer Cell Lines, Antioxidant and Enzyme Inhibition Studies.
    Ahmad A; Ullah F; Sadiq A; Ayaz M; Rahim H; Rashid U; Ahmad S; Jan MS; Ullah R; Shahat AA; Mahmood HM
    Drug Des Devel Ther; 2019; 13():4185-4194. PubMed ID: 31849450
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Discovery of 1,3-Disubstituted 2,5-Diketopiperazine Derivatives as Potent Class I HDACs Inhibitors.
    Gong G; Qi J; Lv Y; Dong S; Cao C; Li D; Zhao R; Li Z; Chen X
    Chem Pharm Bull (Tokyo); 2020; 68(5):466-472. PubMed ID: 32378544
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Structure-based design and synthesis of novel furan-diketopiperazine-type derivatives as potent microtubule inhibitors for treating cancer.
    Ding Z; Li F; Zhong C; Li F; Liu Y; Wang S; Zhao J; Li W
    Bioorg Med Chem; 2020 May; 28(10):115435. PubMed ID: 32278711
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design and synthesis of novel soluble 2,5-diketopiperazine derivatives as potential anticancer agents.
    Liao S; Qin X; Li D; Tu Z; Li J; Zhou X; Wang J; Yang B; Lin X; Liu J; Yang X; Liu Y
    Eur J Med Chem; 2014 Aug; 83():236-44. PubMed ID: 24960627
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Spiro[(dihydropyrazin-2,5-dione)-6,3'-(2',3'-dihydrothieno[2,3-b]naphtho-4',9'-dione)]-based cytotoxic agents: structure-activity relationship studies on the substituent at N4-position of the diketopiperazine domain.
    Gomez-Monterrey I; Campiglia P; Carotenuto A; Stiuso P; Bertamino A; Sala M; Aquino C; Grieco P; Morello S; Pinto A; Ianelli P; Novellino E
    J Med Chem; 2008 May; 51(10):2924-32. PubMed ID: 18429610
    [TBL] [Abstract][Full Text] [Related]  

  • 20. α-Aroylketene Dithioacetal Mediated Synthesis of (E)-3-(benzo[d]thiazol-2-ylamino)-2-(1-methyl-1H-indole-3-carbonyl)-3-(methylthio)acrylonitrile Derivatives and their Biological Evaluation.
    Bhale PS; Chavan HV; Dongare SB; Sankpal ST; Bandgar BP
    Anticancer Agents Med Chem; 2018; 18(5):757-764. PubMed ID: 28901263
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 16.