BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

213 related articles for article (PubMed ID: 28498611)

  • 1. Design, Synthesis, and Biological Evaluation of Peptidomimetic N-Substituted Cbz-4-Hyp-Hpa-Amides as Novel Inhibitors of Plasmodium falciparum.
    Bacherikov VA; Chittiboyina AG; Avery MA
    Chem Biodivers; 2017 Aug; 14(8):. PubMed ID: 28498611
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis, biological evaluation, hydration site thermodynamics, and chemical reactivity analysis of α-keto substituted peptidomimetics for the inhibition of Plasmodium falciparum.
    Weldon DJ; Shah F; Chittiboyina AG; Sheri A; Chada RR; Gut J; Rosenthal PJ; Shivakumar D; Sherman W; Desai P; Jung JC; Avery MA
    Bioorg Med Chem Lett; 2014 Mar; 24(5):1274-9. PubMed ID: 24507921
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Antimalarial and antitrypanosomal activity of a series of amide and sulfonamide derivatives of a 2,5-diaminobenzophenone.
    Altenkämper M; Bechem B; Perruchon J; Heinrich S; Mädel A; Ortmann R; Dahse HM; Freunscht E; Wang Y; Rath J; Stich A; Hitzler M; Chiba P; Lanzer M; Schlitzer M
    Bioorg Med Chem; 2009 Nov; 17(22):7690-7. PubMed ID: 19819706
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Machine learning prioritizes synthesis of primaquine ureidoamides with high antimalarial activity and attenuated cytotoxicity.
    Levatić J; Pavić K; Perković I; Uzelac L; Ester K; Kralj M; Kaiser M; Rottmann M; Supek F; Zorc B
    Eur J Med Chem; 2018 Feb; 146():651-667. PubMed ID: 29407988
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Synthesis and molecular modeling studies of derivatives of a highly potent peptidomimetic vinyl ester as falcipain-2 inhibitors.
    Ettari R; Micale N; Grazioso G; Bova F; Schirmeister T; Grasso S; Zappalà M
    ChemMedChem; 2012 Sep; 7(9):1594-600. PubMed ID: 22753258
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological characterisation of ester and amide derivatives of fusidic acid as antiplasmodial agents.
    Espinoza-Moraga M; Singh K; Njoroge M; Kaur G; Okombo J; De Kock C; Smith PJ; Wittlin S; Chibale K
    Bioorg Med Chem Lett; 2017 Feb; 27(3):658-661. PubMed ID: 28012840
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and evaluation of phosphoramidate and phosphorothioamidate analogues of amiprophos methyl as potential antimalarial agents.
    Mara C; Dempsey E; Bell A; Barlow JW
    Bioorg Med Chem Lett; 2011 Oct; 21(20):6180-3. PubMed ID: 21889338
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Design, Synthesis, and Biological Evaluation of Novel 1,2,4-Trioxanes as Potential Antimalarial Agents.
    Gupta AK; Varshney K; Kumar V; Srivastava K; Pant AB; Puri SK; Saxena AK
    Arch Pharm (Weinheim); 2017 Apr; 350(3-4):. PubMed ID: 28207169
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and antimalarial activity of N-benzylated (N-arylcarbamoyl)alkylphosphonic acid derivatives.
    Adeyemi CM; Faridoon ; Isaacs M; Mnkandhla D; Hoppe HC; Krause RW; Kaye PT
    Bioorg Med Chem; 2016 Dec; 24(23):6131-6138. PubMed ID: 27773366
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Design, synthesis, and evaluation of new chemosensitizers in multi-drug-resistant Plasmodium falciparum.
    Guan J; Kyle DE; Gerena L; Zhang Q; Milhous WK; Lin AJ
    J Med Chem; 2002 Jun; 45(13):2741-8. PubMed ID: 12061877
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline.
    Delarue-Cochin S; Grellier P; Maes L; Mouray E; Sergheraert C; Melnyk P
    Eur J Med Chem; 2008 Oct; 43(10):2045-55. PubMed ID: 18226428
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Tetraoxane-pyrimidine nitrile hybrids as dual stage antimalarials.
    Oliveira R; Guedes RC; Meireles P; Albuquerque IS; Gonçalves LM; Pires E; Bronze MR; Gut J; Rosenthal PJ; Prudêncio M; Moreira R; O'Neill PM; Lopes F
    J Med Chem; 2014 Jun; 57(11):4916-23. PubMed ID: 24824551
    [TBL] [Abstract][Full Text] [Related]  

  • 13. KBE009: An antimalarial bestatin-like inhibitor of the Plasmodium falciparum M1 aminopeptidase discovered in an Ugi multicomponent reaction-derived peptidomimetic library.
    González-Bacerio J; Maluf SEC; Méndez Y; Pascual I; Florent I; Melo PMS; Budu A; Ferreira JC; Moreno E; Carmona AK; Rivera DG; Alonso Del Rivero M; Gazarini ML
    Bioorg Med Chem; 2017 Sep; 25(17):4628-4636. PubMed ID: 28728898
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis of pyrazole acrylic acid based oxadiazole and amide derivatives as antimalarial and anticancer agents.
    Verma G; Chashoo G; Ali A; Khan MF; Akhtar W; Ali I; Akhtar M; Alam MM; Shaquiquzzaman M
    Bioorg Chem; 2018 Apr; 77():106-124. PubMed ID: 29353728
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis of oxalamide and triazine derivatives as a novel class of hybrid 4-aminoquinoline with potent antiplasmodial activity.
    Sunduru N; Sharma M; Srivastava K; Rajakumar S; Puri SK; Saxena JK; Chauhan PM
    Bioorg Med Chem; 2009 Sep; 17(17):6451-62. PubMed ID: 19665899
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and anti-parasitic activity of achiral N-benzylated phosphoramidic acid derivatives.
    Adeyemi CM; Conibear AC; Mutorwa MK; Nokalipa IC; Isaacs M; Mnkandhla D; Hoppe HC; Lobb KA; Klein R; Kaye PT
    Bioorg Chem; 2020 Aug; 101():103947. PubMed ID: 32559578
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Aryl piperazine and pyrrolidine as antimalarial agents. Synthesis and investigation of structure-activity relationships.
    Mendoza A; Pérez-Silanes S; Quiliano M; Pabón A; Galiano S; González G; Garavito G; Zimic M; Vaisberg A; Aldana I; Monge A; Deharo E
    Exp Parasitol; 2011 Jun; 128(2):97-103. PubMed ID: 21354139
    [TBL] [Abstract][Full Text] [Related]  

  • 18. 4-Arylthieno[2,3-
    Schweda SI; Alder A; Gilberger T; Kunick C
    Molecules; 2020 Jul; 25(14):. PubMed ID: 32668631
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and antiplasmodial evaluation of novel mefloquine-based fumardiamides.
    Beus M; Fontinha D; Held J; Rajić Z; Prudêncio M; Zorc B
    Acta Pharm; 2019 Jun; 69(2):233-248. PubMed ID: 31259728
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Peptidomimetic inhibitors of protein farnesyltransferase show potent antimalarial activity.
    Ohkanda J; Lockman JW; Yokoyama K; Gelb MH; Croft SL; Kendrick H; Harrell MI; Feagin JE; Blaskovich MA; Sebti SM; Hamilton AD
    Bioorg Med Chem Lett; 2001 Mar; 11(6):761-4. PubMed ID: 11277514
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.