188 related articles for article (PubMed ID: 28555756)
1. Design and chemical syntheses of potent matriptase-2 inhibitors based on trypsin inhibitor SFTI-1 isolated from sunflower seeds.
Gitlin-Domagalska A; Dębowski D; Łęgowska A; Stirnberg M; Okońska J; Gütschow M; Rolka K
Biopolymers; 2017 Nov; 108(6):. PubMed ID: 28555756
[TBL] [Abstract][Full Text] [Related]
2. Design and synthesis of redox stable analogues of sunflower trypsin inhibitors (SFTI-1) on solid support, potent inhibitors of matriptase.
Jiang S; Li P; Lee SL; Lin CY; Long YQ; Johnson MD; Dickson RB; Roller PP
Org Lett; 2007 Jan; 9(1):9-12. PubMed ID: 17192072
[TBL] [Abstract][Full Text] [Related]
3. Inhibitors of Matriptase-2 Based on the Trypsin Inhibitor SFTI-1.
Gitlin A; Dębowski D; Karna N; Łęgowska A; Stirnberg M; Gütschow M; Rolka K
Chembiochem; 2015 Jul; 16(11):1601-7. PubMed ID: 25999208
[TBL] [Abstract][Full Text] [Related]
4. High-affinity cyclic peptide matriptase inhibitors.
Quimbar P; Malik U; Sommerhoff CP; Kaas Q; Chan LY; Huang YH; Grundhuber M; Dunse K; Craik DJ; Anderson MA; Daly NL
J Biol Chem; 2013 May; 288(19):13885-96. PubMed ID: 23548907
[TBL] [Abstract][Full Text] [Related]
5. Introduction of alpha-hydroxymethyamino acid residues in substrate specificity P1 position of trypsin inhibitor SFTI-1 from sunflower seeds retains its activity.
Zabłotna E; Kret A; Jaśkiewicz A; Olma A; Leplawy MT; Rolka K
Biochem Biophys Res Commun; 2006 Feb; 340(3):823-8. PubMed ID: 16380077
[TBL] [Abstract][Full Text] [Related]
6. Synthesis and evaluation of the sunflower derived trypsin inhibitor as a potent inhibitor of the type II transmembrane serine protease, matriptase.
Long YQ; Lee SL; Lin CY; Enyedy IJ; Wang S; Li P; Dickson RB; Roller PP
Bioorg Med Chem Lett; 2001 Sep; 11(18):2515-9. PubMed ID: 11549459
[TBL] [Abstract][Full Text] [Related]
7. Design and synthesis of novel and potent inhibitors of the type II transmembrane serine protease, matriptase, based upon the sunflower trypsin inhibitor-1.
Li P; Jiang S; Lee SL; Lin CY; Johnson MD; Dickson RB; Michejda CJ; Roller PP
J Med Chem; 2007 Nov; 50(24):5976-83. PubMed ID: 17985858
[TBL] [Abstract][Full Text] [Related]
8. Evaluation of bisbenzamidines as inhibitors for matriptase-2.
Beckmann AM; Gilberg E; Gattner S; Huang TL; Vanden Eynde JJ; Mayence A; Bajorath J; Stirnberg M; Gütschow M
Bioorg Med Chem Lett; 2016 Aug; 26(15):3741-5. PubMed ID: 27287367
[TBL] [Abstract][Full Text] [Related]
9. Potent inhibitors of human matriptase-1 based on the scaffold of sunflower trypsin inhibitor.
Fittler H; Avrutina O; Empting M; Kolmar H
J Pept Sci; 2014 Jun; 20(6):415-20. PubMed ID: 24723440
[TBL] [Abstract][Full Text] [Related]
10. Design of serine proteinase inhibitors by combinatorial chemistry using trypsin inhibitor SFTI-1 as a starting structure.
Zabłotna E; Jaśkiewicz A; Łegowska A; Miecznikowska H; Lesner A; Rolka K
J Pept Sci; 2007 Nov; 13(11):749-55. PubMed ID: 17828796
[TBL] [Abstract][Full Text] [Related]
11. Peptomeric analogues of trypsin inhibitor SFTI-1 isolated from sunflower seeds.
Łegowska A; Bulak E; Wysocka M; Jaśkiewicz A; Lesner A; Debowski D; Rolka K
Bioorg Med Chem; 2008 May; 16(10):5644-52. PubMed ID: 18448341
[TBL] [Abstract][Full Text] [Related]
12. Engineering potent mesotrypsin inhibitors based on the plant-derived cyclic peptide, sunflower trypsin inhibitor-1.
de Veer SJ; Li CY; Swedberg JE; Schroeder CI; Craik DJ
Eur J Med Chem; 2018 Jul; 155():695-704. PubMed ID: 29936356
[TBL] [Abstract][Full Text] [Related]
13. Phosphono Bisbenzguanidines as Irreversible Dipeptidomimetic Inhibitors and Activity-Based Probes of Matriptase-2.
Häußler D; Mangold M; Furtmann N; Braune A; Blaut M; Bajorath J; Stirnberg M; Gütschow M
Chemistry; 2016 Jun; 22(25):8525-35. PubMed ID: 27214780
[TBL] [Abstract][Full Text] [Related]
14. Sunflower trypsin inhibitor-1, proteolytic studies on a trypsin inhibitor peptide and its analogs.
Colgrave ML; Korsinczky MJ; Clark RJ; Foley F; Craik DJ
Biopolymers; 2010; 94(5):665-72. PubMed ID: 20564016
[TBL] [Abstract][Full Text] [Related]
15. Investigation of Serine-Proteinase-Catalyzed Peptide Splicing in Analogues of Sunflower Trypsin Inhibitor 1 (SFTI-1).
Karna N; Łęgowska A; Malicki S; Dębowski D; Golik P; Gitlin A; Grudnik P; Wladyka B; Brzozowski K; Dubin G; Rolka K
Chembiochem; 2015 Sep; 16(14):2036-45. PubMed ID: 26212347
[TBL] [Abstract][Full Text] [Related]
16. Structure-based approach for the discovery of bis-benzamidines as novel inhibitors of matriptase.
Enyedy IJ; Lee SL; Kuo AH; Dickson RB; Lin CY; Wang S
J Med Chem; 2001 Apr; 44(9):1349-55. PubMed ID: 11311057
[TBL] [Abstract][Full Text] [Related]
17. Design of Potent and Selective Cathepsin G Inhibitors Based on the Sunflower Trypsin Inhibitor-1 Scaffold.
Swedberg JE; Li CY; de Veer SJ; Wang CK; Craik DJ
J Med Chem; 2017 Jan; 60(2):658-667. PubMed ID: 28045523
[TBL] [Abstract][Full Text] [Related]
18. Immobilized analogues of sunflower trypsin inhibitor-1 constitute a versatile group of affinity sorbents for selective isolation of serine proteases.
Pereira HJ; Salgado MC; Oliveira EB
J Chromatogr B Analyt Technol Biomed Life Sci; 2009 Jul; 877(22):2039-44. PubMed ID: 19515617
[TBL] [Abstract][Full Text] [Related]
19. Solution structures by 1H NMR of the novel cyclic trypsin inhibitor SFTI-1 from sunflower seeds and an acyclic permutant.
Korsinczky ML; Schirra HJ; Rosengren KJ; West J; Condie BA; Otvos L; Anderson MA; Craik DJ
J Mol Biol; 2001 Aug; 311(3):579-91. PubMed ID: 11493011
[TBL] [Abstract][Full Text] [Related]
20. Mechanism-based selection of a potent kallikrein-related peptidase 7 inhibitor from a versatile library based on the sunflower trypsin inhibitor SFTI-1.
de Veer SJ; Ukolova SS; Munro CA; Swedberg JE; Buckle AM; Harris JM
Biopolymers; 2013 Sep; 100(5):510-8. PubMed ID: 24078181
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
