BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

80 related articles for article (PubMed ID: 28635318)

  • 1. What structural modifications can be used for BRD4 inhibitors for their use in leukemia therapy?
    Yao D; Liu J; Ouyang L
    Future Med Chem; 2017 Jun; 9(9):839-842. PubMed ID: 28635318
    [No Abstract]   [Full Text] [Related]  

  • 2. Design and characterization of bivalent BET inhibitors.
    Tanaka M; Roberts JM; Seo HS; Souza A; Paulk J; Scott TG; DeAngelo SL; Dhe-Paganon S; Bradner JE
    Nat Chem Biol; 2016 Dec; 12(12):1089-1096. PubMed ID: 27775715
    [TBL] [Abstract][Full Text] [Related]  

  • 3. An Overview on Small Molecule Inhibitors of BRD4.
    Huang W; Zheng X; Yang Y; Wang X; Shen Z
    Mini Rev Med Chem; 2016; 16(17):1403-1414. PubMed ID: 27290915
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Phthalimide-Conjugated Ligands Promote Selective Protein Destabilization.
    Cancer Discov; 2015 Jul; 5(7):691. PubMed ID: 26045013
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Disrupting the reader of histone language.
    Oliver SS; Denu JM
    Angew Chem Int Ed Engl; 2011 Jun; 50(26):5801-3. PubMed ID: 21618372
    [No Abstract]   [Full Text] [Related]  

  • 6. Discovery of novel BRD4 inhibitors by high-throughput screening, crystallography, and cell-based assays.
    Sun Z; Zhang H; Chen Z; Xie Y; Jiang H; Chen L; Ding H; Zhang Y; Jiang H; Zheng M; Luo C
    Bioorg Med Chem Lett; 2017 May; 27(9):2003-2009. PubMed ID: 28347667
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Cancer research: Open ambition.
    Maxmen A
    Nature; 2012 Aug; 488(7410):148-50. PubMed ID: 22874946
    [No Abstract]   [Full Text] [Related]  

  • 8. Cancer: Bet on drug resistance.
    Settleman J
    Nature; 2016 Jan; 529(7586):289-90. PubMed ID: 26735017
    [No Abstract]   [Full Text] [Related]  

  • 9. BRD4: a BET(ter) target for the treatment of AML?
    Valent P; Zuber J
    Cell Cycle; 2014; 13(5):689-90. PubMed ID: 24526121
    [No Abstract]   [Full Text] [Related]  

  • 10. Heart failure: BRD4 inhibition slows HF progression.
    Ummarino D
    Nat Rev Cardiol; 2017 Jul; 14(7):382-383. PubMed ID: 28569271
    [No Abstract]   [Full Text] [Related]  

  • 11. Bromodomain and extraterminal domain inhibitors (BETi) for cancer therapy: chemical modulation of chromatin structure.
    Qi J
    Cold Spring Harb Perspect Biol; 2014 Dec; 6(12):a018663. PubMed ID: 25452384
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Mapping the chemical chromatin reactivation landscape identifies BRD4-TAF1 cross-talk.
    Sdelci S; Lardeau CH; Tallant C; Klepsch F; Klaiber B; Bennett J; Rathert P; Schuster M; Penz T; Fedorov O; Superti-Furga G; Bock C; Zuber J; Huber KV; Knapp S; Müller S; Kubicek S
    Nat Chem Biol; 2016 Jul; 12(7):504-10. PubMed ID: 27159579
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Targeting the BET family for the treatment of leukemia.
    Lucas X; Günther S
    Epigenomics; 2014 Apr; 6(2):153-5. PubMed ID: 24811781
    [No Abstract]   [Full Text] [Related]  

  • 14. Structure-Activity Relationship Study of N(6)-Benzoyladenine-Type BRD4 Inhibitors and Their Effects on Cell Differentiation and TNF-α Production.
    Amemiya S; Yamaguchi T; Sakai T; Hashimoto Y; Noguchi-Yachide T
    Chem Pharm Bull (Tokyo); 2016; 64(9):1378-83. PubMed ID: 27581642
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Suppression of BRD4 inhibits human hepatocellular carcinoma by repressing MYC and enhancing BIM expression.
    Li GQ; Guo WZ; Zhang Y; Seng JJ; Zhang HP; Ma XX; Zhang G; Li J; Yan B; Tang HW; Li SS; Wang LD; Zhang SJ
    Oncotarget; 2016 Jan; 7(3):2462-74. PubMed ID: 26575167
    [TBL] [Abstract][Full Text] [Related]  

  • 16. BET Bromodomain Blockade Mitigates Intimal Hyperplasia in Rat Carotid Arteries.
    Wang B; Zhang M; Takayama T; Shi X; Roenneburg DA; Kent KC; Guo LW
    EBioMedicine; 2015 Nov; 2(11):1650-61. PubMed ID: 26870791
    [TBL] [Abstract][Full Text] [Related]  

  • 17. BET Bromodomain Inhibition as a Therapeutic Strategy in Ovarian Cancer by Downregulating FoxM1.
    Zhang Z; Ma P; Jing Y; Yan Y; Cai MC; Zhang M; Zhang S; Peng H; Ji ZL; Di W; Gu Z; Gao WQ; Zhuang G
    Theranostics; 2016; 6(2):219-30. PubMed ID: 26877780
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Synthesis and evaluation of novel dual BRD4/HDAC inhibitors.
    Amemiya S; Yamaguchi T; Hashimoto Y; Noguchi-Yachide T
    Bioorg Med Chem; 2017 Jul; 25(14):3677-3684. PubMed ID: 28549889
    [TBL] [Abstract][Full Text] [Related]  

  • 19. 4-Acyl Pyrrole Capped HDAC Inhibitors: A New Scaffold for Hybrid Inhibitors of BET Proteins and Histone Deacetylases as Antileukemia Drug Leads.
    Schäker-Hübner L; Warstat R; Ahlert H; Mishra P; Kraft FB; Schliehe-Diecks J; Schöler A; Borkhardt A; Breit B; Bhatia S; Hügle M; Günther S; Hansen FK
    J Med Chem; 2021 Oct; 64(19):14620-14646. PubMed ID: 34582215
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds.
    Chan KH; Zengerle M; Testa A; Ciulli A
    J Med Chem; 2018 Jan; 61(2):504-513. PubMed ID: 28595007
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 4.