These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
165 related articles for article (PubMed ID: 28661196)
1. Design, synthesis and evaluation of 2-aryl benzoxazoles as promising hit for the A Duroux R; Renault N; Cuelho JE; Agouridas L; Blum D; Lopes LV; Melnyk P; Yous S J Enzyme Inhib Med Chem; 2017 Dec; 32(1):850-864. PubMed ID: 28661196 [TBL] [Abstract][Full Text] [Related]
2. Antagonists of the adenosine A Duroux R; Agouridas L; Renault N; El Bakali J; Furman C; Melnyk P; Yous S Eur J Med Chem; 2018 Jan; 144():151-163. PubMed ID: 29268131 [TBL] [Abstract][Full Text] [Related]
3. Design, synthesis and biological evaluation of novel scaffold benzo[4,5]imidazo [1,2-a]pyrazin-1-amine: Towards adenosine A Reddy GL; Sarma R; Liu S; Huang W; Lei J; Fu J; Hu W Eur J Med Chem; 2021 Jan; 210():113040. PubMed ID: 33316692 [TBL] [Abstract][Full Text] [Related]
4. Novel Quinazoline Derivatives as Highly Effective A2A Adenosine Receptor Antagonists. Laversin A; Dufossez R; Bolteau R; Duroux R; Ravez S; Hernandez-Tapia S; Fossart M; Coevoet M; Liberelle M; Yous S; Lebègue N; Melnyk P Molecules; 2024 Aug; 29(16):. PubMed ID: 39202926 [TBL] [Abstract][Full Text] [Related]
5. Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A Renk DR; Skraban M; Bier D; Schulze A; Wabbals E; Wedekind F; Neumaier F; Neumaier B; Holschbach M Eur J Med Chem; 2021 Mar; 214():113214. PubMed ID: 33548636 [TBL] [Abstract][Full Text] [Related]
6. Synthesis and SAR studies of analogues of 4-(3,3-dimethyl-butyrylamino)-3,5-difluoro-N-thiazol-2-yl-benzamide (Lu AA41063) as adenosine A2A receptor ligands with improved aqueous solubility. Mikkelsen GK; Langgård M; Schrøder TJ; Kreilgaard M; Jørgensen EB; Brandt G; Griffon Y; Boffey R; Bang-Andersen B Bioorg Med Chem Lett; 2015 Mar; 25(6):1212-6. PubMed ID: 25701253 [TBL] [Abstract][Full Text] [Related]
7. Replacement of amide with bioisosteres led to a new series of potent adenosine A2A receptor antagonists. Yang Z; Li X; Ma H; Zheng J; Zhen X; Zhang X Bioorg Med Chem Lett; 2014 Jan; 24(1):152-5. PubMed ID: 24332624 [TBL] [Abstract][Full Text] [Related]
8. Synthesis and evaluation of methoxy substituted 2-benzoyl-1-benzofuran derivatives as lead compounds for the development adenosine A Janse van Rensburg HD; Legoabe LJ; Terre'Blanche G; Aucamp J Bioorg Chem; 2020 Jan; 94():103459. PubMed ID: 31818481 [TBL] [Abstract][Full Text] [Related]
9. 8-Substituted 1,3-dimethyltetrahydropyrazino[2,1-f]purinediones: Water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors. Brunschweiger A; Koch P; Schlenk M; Rafehi M; Radjainia H; Küppers P; Hinz S; Pineda F; Wiese M; Hockemeyer J; Heer J; Denonne F; Müller CE Bioorg Med Chem; 2016 Nov; 24(21):5462-5480. PubMed ID: 27658798 [TBL] [Abstract][Full Text] [Related]
10. C2-substituted quinazolinone derivatives exhibit A Pieterse L; van der Walt MM; Terre'Blanche G Bioorg Med Chem Lett; 2020 Aug; 30(16):127274. PubMed ID: 32631506 [TBL] [Abstract][Full Text] [Related]
11. 5-Substituted 2-benzylidene-1-tetralone analogues as A Janse van Rensburg HD; Terre'Blanche G; van der Walt MM; Legoabe LJ Bioorg Chem; 2017 Oct; 74():251-259. PubMed ID: 28881253 [TBL] [Abstract][Full Text] [Related]
12. Discovery of 1,3-diethyl-7-methyl-8-(phenoxymethyl)-xanthine derivatives as novel adenosine A Harmse R; van der Walt MM; Petzer JP; Terre'Blanche G Bioorg Med Chem Lett; 2016 Dec; 26(24):5951-5955. PubMed ID: 27836398 [TBL] [Abstract][Full Text] [Related]
13. 2-Aminopyrimidines as dual adenosine A1/A2A antagonists. Robinson SJ; Petzer JP; Terre'Blanche G; Petzer A; van der Walt MM; Bergh JJ; Lourens AC Eur J Med Chem; 2015 Nov; 104():177-88. PubMed ID: 26462195 [TBL] [Abstract][Full Text] [Related]
14. The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3-d]pyrimidine core in affecting adenosine A Squarcialupi L; Betti M; Catarzi D; Varano F; Falsini M; Ravani A; Pasquini S; Vincenzi F; Salmaso V; Sturlese M; Varani K; Moro S; Colotta V J Enzyme Inhib Med Chem; 2017 Dec; 32(1):248-263. PubMed ID: 28114825 [TBL] [Abstract][Full Text] [Related]
15. Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A Basu S; Barawkar DA; Thorat S; Shejul YD; Patel M; Naykodi M; Jain V; Salve Y; Prasad V; Chaudhary S; Ghosh I; Bhat G; Quraishi A; Patil H; Ansari S; Menon S; Unadkat V; Thakare R; Seervi MS; Meru AV; De S; Bhamidipati RK; Rouduri SR; Palle VP; Chug A; Mookhtiar KA J Med Chem; 2017 Jan; 60(2):681-694. PubMed ID: 28055204 [TBL] [Abstract][Full Text] [Related]
16. The adenosine A(2A) antagonistic properties of selected C8-substituted xanthines. Van der Walt MM; Terre'Blanche G; Petzer A; Lourens AC; Petzer JP Bioorg Chem; 2013 Aug; 49():49-58. PubMed ID: 23892098 [TBL] [Abstract][Full Text] [Related]
17. Design and synthesis of (4E)-4-(4-substitutedbenzylideneamino)-3-substituted-2,3-dihydro-2-thioxothiazole-5-carbonitrile as novel A2A receptor antagonists. Mishra CB; Sharma D; Prakash A; Kumari N; Kumar N; Luthra PM Bioorg Med Chem; 2013 Oct; 21(19):6077-83. PubMed ID: 23953686 [TBL] [Abstract][Full Text] [Related]
18. Discovery of Novel and Selective Adenosine A Tian S; Wang X; Li L; Zhang X; Li Y; Zhu F; Hou T; Zhen X J Chem Inf Model; 2017 Jun; 57(6):1474-1487. PubMed ID: 28463561 [TBL] [Abstract][Full Text] [Related]
19. Synthesis, biological evaluation and molecular modelling studies of 1,3,7,8-tetrasubstituted xanthines as potent and selective A Rohilla S; Bansal R; Kachler S; Klotz KN Bioorg Chem; 2019 Jun; 87():601-612. PubMed ID: 30933785 [TBL] [Abstract][Full Text] [Related]
20. 2-Benzylidene-1-Indanone Analogues as Dual Adenosine A1/A2a Receptor Antagonists for the Potential Treatment of Neurological Conditions. van Rensburg HJ; Legoabe L; Terre'Blanche G; Van der Walt M Drug Res (Stuttg); 2019 Jul; 69(7):382-391. PubMed ID: 30616250 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]