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4. A close structural analog of 2-methyl-6-(phenylethynyl)-pyridine acts as a neutral allosteric site ligand on metabotropic glutamate receptor subtype 5 and blocks the effects of multiple allosteric modulators. Rodriguez AL; Nong Y; Sekaran NK; Alagille D; Tamagnan GD; Conn PJ Mol Pharmacol; 2005 Dec; 68(6):1793-802. PubMed ID: 16155210 [TBL] [Abstract][Full Text] [Related]
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