152 related articles for article (PubMed ID: 28733082)
1. Effects of novel triple-stage antimalarial ionic liquids on lipid membrane models.
Ferraz R; Pinheiro M; Gomes A; Teixeira C; Prudêncio C; Reis S; Gomes P
Bioorg Med Chem Lett; 2017 Sep; 27(17):4190-4193. PubMed ID: 28733082
[TBL] [Abstract][Full Text] [Related]
2. Building on Surface-Active Ionic Liquids for the Rescuing of the Antimalarial Drug Chloroquine.
Silva AT; Lobo L; Oliveira IS; Gomes J; Teixeira C; Nogueira F; Marques EF; Ferraz R; Gomes P
Int J Mol Sci; 2020 Jul; 21(15):. PubMed ID: 32727096
[TBL] [Abstract][Full Text] [Related]
3. Drug-Derived Surface-Active Ionic Liquids: A Cost-Effective Way To Expressively Increase the Blood-Stage Antimalarial Activity of Primaquine.
Silva AT; Oliveira IS; Gomes J; Aguiar L; Fontinha D; Duarte D; Nogueira F; Prudêncio M; Marques EF; Teixeira C; Ferraz R; Gomes P
ChemMedChem; 2022 Mar; 17(5):e202100650. PubMed ID: 34882979
[TBL] [Abstract][Full Text] [Related]
4. Machine learning prioritizes synthesis of primaquine ureidoamides with high antimalarial activity and attenuated cytotoxicity.
Levatić J; Pavić K; Perković I; Uzelac L; Ester K; Kralj M; Kaiser M; Rottmann M; Supek F; Zorc B
Eur J Med Chem; 2018 Feb; 146():651-667. PubMed ID: 29407988
[TBL] [Abstract][Full Text] [Related]
5. Probing the Azaaurone Scaffold against the Hepatic and Erythrocytic Stages of Malaria Parasites.
Carrasco MP; Machado M; Gonçalves L; Sharma M; Gut J; Lukens AK; Wirth DF; André V; Duarte MT; Guedes RC; Dos Santos DJ; Rosenthal PJ; Mazitschek R; Prudêncio M; Moreira R
ChemMedChem; 2016 Oct; 11(19):2194-2204. PubMed ID: 27538856
[TBL] [Abstract][Full Text] [Related]
6. In vitro efficiency of 9-(N-cinnamoylbutyl)aminoacridines against blood- and liver-stage malaria parasites.
Pérez B; Teixeira C; Gomes AS; Albuquerque IS; Gut J; Rosenthal PJ; Prudêncio M; Gomes P
Bioorg Med Chem Lett; 2013 Feb; 23(3):610-3. PubMed ID: 23290049
[TBL] [Abstract][Full Text] [Related]
7. 4,9-Diaminoacridines and 4-Aminoacridines as Dual-Stage Antiplasmodial Hits.
Fonte M; Tassi N; Fontinha D; Bouzón-Arnáiz I; Ferraz R; Araújo MJ; Fernàndez-Busquets X; Prudêncio M; Gomes P; Teixeira C
ChemMedChem; 2021 Mar; 16(5):788-792. PubMed ID: 33217195
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and in vitro evaluation of hydrazinyl phthalazines against malaria parasite, Plasmodium falciparum.
Subramanian G; Babu Rajeev CP; Mohan CD; Sinha A; Chu TTT; Anusha S; Ximei H; Fuchs JE; Bender A; Rangappa KS; Chandramohanadas R; Basappa
Bioorg Med Chem Lett; 2016 Jul; 26(14):3300-3306. PubMed ID: 27261180
[TBL] [Abstract][Full Text] [Related]
9. Cinnamoylated chloroquine analogues: A new structural class of antimalarial agents.
Gayam V; Ravi S
Eur J Med Chem; 2017 Jul; 135():382-391. PubMed ID: 28460312
[TBL] [Abstract][Full Text] [Related]
10. Emergence of pyrido quinoxalines as new family of antimalarial agents.
Chandra Shekhar A; Shanthan Rao P; Narsaiah B; Allanki AD; Sijwali PS
Eur J Med Chem; 2014 Apr; 77():280-7. PubMed ID: 24650715
[TBL] [Abstract][Full Text] [Related]
11. Structure activity refinement of phenylsulfonyl piperazines as antimalarials that block erythrocytic invasion.
Nguyen W; Dans MG; Ngo A; Gancheva MR; Romeo O; Duffy S; de Koning-Ward TF; Lowes KN; Sabroux HJ; Avery VM; Wilson DW; Gilson PR; Sleebs BE
Eur J Med Chem; 2021 Mar; 214():113253. PubMed ID: 33610028
[TBL] [Abstract][Full Text] [Related]
12. Micelle carriers based on dendritic macromolecules containing bis-MPA and glycine for antimalarial drug delivery.
Martí Coma-Cros E; Lancelot A; San Anselmo M; Neves Borgheti-Cardoso L; Valle-Delgado JJ; Serrano JL; Fernàndez-Busquets X; Sierra T
Biomater Sci; 2019 Mar; 7(4):1661-1674. PubMed ID: 30741274
[TBL] [Abstract][Full Text] [Related]
13. Antiplasmodial activity of new 4-aminoquinoline derivatives against chloroquine resistant strain.
Sinha M; Dola VR; Agarwal P; Srivastava K; Haq W; Puri SK; Katti SB
Bioorg Med Chem; 2014 Jul; 22(14):3573-86. PubMed ID: 24906512
[TBL] [Abstract][Full Text] [Related]
14. Optimisation of 2-(N-phenyl carboxamide) triazolopyrimidine antimalarials with moderate to slow acting erythrocytic stage activity.
Bailey BL; Nguyen W; Ngo A; Goodman CD; Gancheva MR; Favuzza P; Sanz LM; Gamo FJ; Lowes KN; McFadden GI; Wilson DW; Laleu B; Brand S; Jackson PF; Cowman AF; Sleebs BE
Bioorg Chem; 2021 Oct; 115():105244. PubMed ID: 34452759
[TBL] [Abstract][Full Text] [Related]
15. Primaquine-pyrimidine hybrids: synthesis and dual-stage antiplasmodial activity.
Kaur H; Machado M; de Kock C; Smith P; Chibale K; Prudêncio M; Singh K
Eur J Med Chem; 2015 Aug; 101():266-73. PubMed ID: 26142491
[TBL] [Abstract][Full Text] [Related]
16. Flavones as isosteres of 4(1H)-quinolones: discovery of ligand efficient and dual stage antimalarial lead compounds.
Rodrigues T; Ressurreição AS; da Cruz FP; Albuquerque IS; Gut J; Carrasco MP; Gonçalves D; Guedes RC; dos Santos DJ; Mota MM; Rosenthal PJ; Moreira R; Prudêncio M; Lopes F
Eur J Med Chem; 2013 Nov; 69():872-80. PubMed ID: 24125849
[TBL] [Abstract][Full Text] [Related]
17. In vitro efficiency of new acridyl derivatives against Plasmodium falciparum.
Guetzoyan L; Ramiandrasoa F; Dorizon H; Desprez C; Bridoux A; Rogier C; Pradines B; Perrée-Fauvet M
Bioorg Med Chem; 2007 May; 15(9):3278-89. PubMed ID: 17339112
[TBL] [Abstract][Full Text] [Related]
18. Coupling the Antimalarial Cell Penetrating Peptide TP10 to Classical Antimalarial Drugs Primaquine and Chloroquine Produces Strongly Hemolytic Conjugates.
Aguiar L; Biosca A; Lantero E; Gut J; Vale N; Rosenthal PJ; Nogueira F; Andreu D; Fernàndez-Busquets X; Gomes P
Molecules; 2019 Dec; 24(24):. PubMed ID: 31842498
[TBL] [Abstract][Full Text] [Related]
19. Selective anti-malarial minor groove binders.
Scott FJ; Khalaf AI; Duffy S; Avery VM; Suckling CJ
Bioorg Med Chem Lett; 2016 Jul; 26(14):3326-3329. PubMed ID: 27212070
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and antimalarial activity of chain substituted pivaloyloxymethyl ester analogues of Fosmidomycin and FR900098.
Kurz T; Schlüter K; Kaula U; Bergmann B; Walter RD; Geffken D
Bioorg Med Chem; 2006 Aug; 14(15):5121-35. PubMed ID: 16679022
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]