BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

148 related articles for article (PubMed ID: 28756263)

  • 1. Synthesis and pharmacological evaluation of benzamide derivatives as potent and selective sigma-1 protein ligands.
    Donnier-Maréchal M; Carato P; Larchanché PE; Ravez S; Boulahjar R; Barczyk A; Oxombre B; Vermersch P; Melnyk P
    Eur J Med Chem; 2017 Sep; 138():964-978. PubMed ID: 28756263
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Synthesis and in vitro evaluation of tetrahydroisoquinolinyl benzamides as ligands for sigma receptors.
    Xu R; Lever JR; Lever SZ
    Bioorg Med Chem Lett; 2007 May; 17(9):2594-7. PubMed ID: 17317173
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Synthesis and pharmacological evaluation of benzannulated derivatives as potent and selective sigma-1 protein ligands.
    Donnier-Maréchal M; Carato P; Le Broc D; Furman C; Melnyk P
    Eur J Med Chem; 2015 Mar; 92():575-82. PubMed ID: 25602932
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Improving selectivity preserving affinity: new piperidine-4-carboxamide derivatives as effective sigma-1-ligands.
    Zampieri D; Laurini E; Vio L; Fermeglia M; Pricl S; Wünsch B; Schepmann D; Mamolo MG
    Eur J Med Chem; 2015 Jan; 90():797-808. PubMed ID: 25528334
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Novel High Affinity Sigma-1 Receptor Ligands from Minimal Ensemble Docking-Based Virtual Screening.
    Dvorácskó S; Lázár L; Fülöp F; Palkó M; Zalán Z; Penke B; Fülöp L; Tömböly C; Bogár F
    Int J Mol Sci; 2021 Jul; 22(15):. PubMed ID: 34360878
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and pharmacological evaluation of SNC80 analogues with a bridged piperazine ring.
    Holl R; Jung B; Schepmann D; Humpf HU; Grünert R; Bednarski PJ; Englberger W; Wünsch B
    ChemMedChem; 2009 Dec; 4(12):2111-22. PubMed ID: 19827086
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and pharmacological evaluation of 6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as sigma-2 receptor ligands.
    Sun YT; Wang GF; Yang YQ; Jin F; Wang Y; Xie XY; Mach RH; Huang YS
    Eur J Med Chem; 2018 Mar; 147():227-237. PubMed ID: 29438891
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Novel heterocyclic trans olefin analogues of N-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl}arylcarboxamides as selective probes with high affinity for the dopamine D3 receptor.
    Grundt P; Carlson EE; Cao J; Bennett CJ; McElveen E; Taylor M; Luedtke RR; Newman AH
    J Med Chem; 2005 Feb; 48(3):839-48. PubMed ID: 15689168
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Gaining in pan-affinity towards sigma 1 and sigma 2 receptors. SAR studies on arylalkylamines.
    Rossi D; Rui M; Di Giacomo M; Schepmann D; Wünsch B; Monteleone S; Liedl KR; Collina S
    Bioorg Med Chem; 2017 Jan; 25(1):11-19. PubMed ID: 27838169
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Effect of structural modification in the amine portion of substituted aminobutyl-benzamides as ligands for binding σ1 and σ2 receptors.
    Fan KH; Lever JR; Lever SZ
    Bioorg Med Chem; 2011 Mar; 19(6):1852-9. PubMed ID: 21376604
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Design, synthesis and receptor affinity of novel conformationally restricted σ ligands based on the [4.3.3]propellane scaffold.
    Torres-Gómez H; Lehmkuhl K; Schepmann D; Wünsch B
    Eur J Med Chem; 2013; 70():78-87. PubMed ID: 24140950
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis, Computational Insights, and Evaluation of Novel Sigma Receptors Ligands.
    Dichiara M; Ambrosio FA; Barbaraci C; González-Cano R; Costa G; Parenti C; Marrazzo A; Pasquinucci L; Cobos EJ; Alcaro S; Amata E
    ACS Chem Neurosci; 2023 May; 14(10):1845-1858. PubMed ID: 37155827
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Synthesis and quantitative structure-activity relationships of N-(1-benzylpiperidin-4-yl)phenylacetamides and related analogues as potent and selective sigma1 receptor ligands.
    Huang Y; Hammond PS; Whirrett BR; Kuhner RJ; Wu L; Childers SR; Mach RH
    J Med Chem; 1998 Jun; 41(13):2361-70. PubMed ID: 9632369
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Discovery of 3-(2-aminoethyl)-thiazolidine-2,4-diones as a novel chemotype of sigma-1 receptor ligands.
    Elkholy N; Abdelwaly A; Mohamed K; Amata E; Lombino J; Cosentino G; Intagliata S; Helal MA
    Chem Biol Drug Des; 2022 Jul; 100(1):25-40. PubMed ID: 35353926
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis and receptor binding studies of some new arylcarboxamide derivatives as sigma-1 ligands.
    Zampieri D; Laurini E; Vio L; Golob S; Fermeglia M; Pricl S; Mamolo MG
    Bioorg Med Chem Lett; 2014 Feb; 24(4):1021-5. PubMed ID: 24486131
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands.
    Romeo G; Prezzavento O; Intagliata S; Pittalà V; Modica MN; Marrazzo A; Turnaturi R; Parenti C; Chiechio S; Arena E; Campisi A; Sposito G; Salerno L
    Eur J Med Chem; 2019 Jul; 174():226-235. PubMed ID: 31042618
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Synthesis of benzamide derivatives and their evaluation as antiprion agents.
    Fiorino F; Eiden M; Giese A; Severino B; Esposito A; Groschup MH; Perissutti E; Magli E; Incisivo GM; Ciano A; Frecentese F; Kretzschmar HA; Wagner J; Santagada V; Caliendo G
    Bioorg Med Chem; 2012 Aug; 20(16):5001-11. PubMed ID: 22795751
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Probes for narcotic receptor-mediated phenomena. 25. Synthesis and evaluation of N-alkyl-substituted (alpha-piperazinylbenzyl)benzamides as novel, highly selective delta opioid receptor agonists.
    Katsura Y; Zhang X; Homma K; Rice KC; Calderon SN; Rothman RB; Yamamura HI; Davis P; Flippen-Anderson JL; Xu H; Becketts K; Foltz EJ; Porreca F
    J Med Chem; 1997 Aug; 40(18):2936-47. PubMed ID: 9288176
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and structure-activity relationship studies of conformationally flexible tetrahydroisoquinolinyl triazole carboxamide and triazole substituted benzamide analogues as σ2 receptor ligands.
    Bai S; Li S; Xu J; Peng X; Sai K; Chu W; Tu Z; Zeng C; Mach RH
    J Med Chem; 2014 May; 57(10):4239-51. PubMed ID: 24821398
    [TBL] [Abstract][Full Text] [Related]  

  • 20. A systematic exploration of the effects of flexibility and basicity on sigma (σ) receptor binding in a series of substituted diamines.
    Conroy T; Manohar M; Gong Y; Wilkinson SM; Webster M; Lieberman BP; Banister SD; Reekie TA; Mach RH; Rendina LM; Kassiou M
    Org Biomol Chem; 2016 Oct; 14(39):9388-9405. PubMed ID: 27714195
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.