These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

346 related articles for article (PubMed ID: 28784300)

  • 1. Synthesis and biological evaluation of Aspergillomarasmine A derivatives as novel NDM-1 inhibitor to overcome antibiotics resistance.
    Zhang J; Wang S; Wei Q; Guo Q; Bai Y; Yang S; Song F; Zhang L; Lei X
    Bioorg Med Chem; 2017 Oct; 25(19):5133-5141. PubMed ID: 28784300
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Aspergillomarasmine A overcomes metallo-β-lactamase antibiotic resistance.
    King AM; Reid-Yu SA; Wang W; King DT; De Pascale G; Strynadka NC; Walsh TR; Coombes BK; Wright GD
    Nature; 2014 Jun; 510(7506):503-6. PubMed ID: 24965651
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Total Synthesis and Activity of the Metallo-β-lactamase Inhibitor Aspergillomarasmine A.
    Koteva K; King AM; Capretta A; Wright GD
    Angew Chem Int Ed Engl; 2016 Feb; 55(6):2210-2. PubMed ID: 26709849
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Suppression of β-Lactam Resistance by Aspergillomarasmine A Is Influenced by both the Metallo-β-Lactamase Target and the Antibiotic Partner.
    Rotondo CM; Sychantha D; Koteva K; Wright GD
    Antimicrob Agents Chemother; 2020 Mar; 64(4):. PubMed ID: 31932375
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Efficacy of aspergillomarasmine A/meropenem combinations with and without avibactam against bacterial strains producing multiple β-lactamases.
    Rotondo CM; Wright GD
    Antimicrob Agents Chemother; 2024 Sep; 68(9):e0027224. PubMed ID: 39133022
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Probing the Interaction of Aspergillomarasmine A with Metallo-β-lactamases NDM-1, VIM-2, and IMP-7.
    Bergstrom A; Katko A; Adkins Z; Hill J; Cheng Z; Burnett M; Yang H; Aitha M; Mehaffey MR; Brodbelt JS; Tehrani KHME; Martin NI; Bonomo RA; Page RC; Tierney DL; Fast W; Wright GD; Crowder MW
    ACS Infect Dis; 2018 Feb; 4(2):135-145. PubMed ID: 29091730
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Total Synthesis and Structural Reassignment of Aspergillomarasmine A.
    Liao D; Yang S; Wang J; Zhang J; Hong B; Wu F; Lei X
    Angew Chem Int Ed Engl; 2016 Mar; 55(13):4291-5. PubMed ID: 26592805
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Synthesis and Preclinical Evaluation of TPA-Based Zinc Chelators as Metallo-β-lactamase Inhibitors.
    Schnaars C; Kildahl-Andersen G; Prandina A; Popal R; Radix S; Le Borgne M; Gjøen T; Andresen AMS; Heikal A; Økstad OA; Fröhlich C; Samuelsen Ø; Lauksund S; Jordheim LP; Rongved P; Åstrand OAH
    ACS Infect Dis; 2018 Sep; 4(9):1407-1422. PubMed ID: 30022668
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Aspergillomarasmine A, an inhibitor of bacterial metallo-β-lactamases conferring blaNDM and blaVIM resistance.
    von Nussbaum F; Schiffer G
    Angew Chem Int Ed Engl; 2014 Oct; 53(44):11696-8. PubMed ID: 25256630
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Structural studies of triazole inhibitors with promising inhibitor effects against antibiotic resistance metallo-β-lactamases.
    Muhammad Z; Skagseth S; Boomgaren M; Akhter S; Fröhlich C; Ismael A; Christopeit T; Bayer A; Leiros HS
    Bioorg Med Chem; 2020 Aug; 28(15):115598. PubMed ID: 32631568
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Aspergillomarasmine A inhibits metallo-β-lactamases by selectively sequestering Zn
    Sychantha D; Rotondo CM; Tehrani KHME; Martin NI; Wright GD
    J Biol Chem; 2021 Aug; 297(2):100918. PubMed ID: 34181945
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Dipicolinic Acid Derivatives as Inhibitors of New Delhi Metallo-β-lactamase-1.
    Chen AY; Thomas PW; Stewart AC; Bergstrom A; Cheng Z; Miller C; Bethel CR; Marshall SH; Credille CV; Riley CL; Page RC; Bonomo RA; Crowder MW; Tierney DL; Fast W; Cohen SM
    J Med Chem; 2017 Sep; 60(17):7267-7283. PubMed ID: 28809565
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Approved Drugs Containing Thiols as Inhibitors of Metallo-β-lactamases: Strategy To Combat Multidrug-Resistant Bacteria.
    Klingler FM; Wichelhaus TA; Frank D; Cuesta-Bernal J; El-Delik J; Müller HF; Sjuts H; Göttig S; Koenigs A; Pos KM; Pogoryelov D; Proschak E
    J Med Chem; 2015 Apr; 58(8):3626-30. PubMed ID: 25815530
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Aminocarboxylic acids related to aspergillomarasmine A (AMA) and ethylenediamine-N,N'-disuccinic acid (EDDS) are strong zinc-binders and inhibitors of the metallo-beta-lactamase NDM-1.
    Tehrani KHME; Fu H; Brüchle NC; Mashayekhi V; Prats Luján A; van Haren MJ; Poelarends GJ; Martin NI
    Chem Commun (Camb); 2020 Mar; 56(20):3047-3049. PubMed ID: 32048688
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Drug Repurposing of the Unithiol: Inhibition of Metallo-β-Lactamases for the Treatment of Carbapenem-Resistant Gram-Negative Bacterial Infections.
    Grigorenko VG; Khrenova MG; Andreeva IP; Rubtsova MY; Lev AI; Novikova TS; Detusheva EV; Fursova NK; Dyatlov IA; Egorov AM
    Int J Mol Sci; 2022 Feb; 23(3):. PubMed ID: 35163756
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Design, synthesis, and in vitro and biological evaluation of potent amino acid-derived thiol inhibitors of the metallo-β-lactamase IMP-1.
    Arjomandi OK; Hussein WM; Vella P; Yusof Y; Sidjabat HE; Schenk G; McGeary RP
    Eur J Med Chem; 2016 May; 114():318-27. PubMed ID: 27017264
    [TBL] [Abstract][Full Text] [Related]  

  • 17. NOTA analogue: A first dithiocarbamate inhibitor of metallo-β-lactamases.
    Zhang E; Wang MM; Huang SC; Xu SM; Cui DY; Bo YL; Bai PY; Hua YG; Xiao CL; Qin S
    Bioorg Med Chem Lett; 2018 Jan; 28(2):214-221. PubMed ID: 29248295
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Vancomycin Analogue Restores Meropenem Activity against NDM-1 Gram-Negative Pathogens.
    Yarlagadda V; Sarkar P; Samaddar S; Manjunath GB; Mitra SD; Paramanandham K; Shome BR; Haldar J
    ACS Infect Dis; 2018 Jul; 4(7):1093-1101. PubMed ID: 29726673
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Fragment-based discovery of inhibitor scaffolds targeting the metallo-β-lactamases NDM-1 and VIM-2.
    Christopeit T; Leiros HK
    Bioorg Med Chem Lett; 2016 Apr; 26(8):1973-7. PubMed ID: 26976213
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Iminodiacetic Acid as a Novel Metal-Binding Pharmacophore for New Delhi Metallo-β-lactamase Inhibitor Development.
    Chen AY; Thomas CA; Thomas PW; Yang K; Cheng Z; Fast W; Crowder MW; Cohen SM
    ChemMedChem; 2020 Jul; 15(14):1272-1282. PubMed ID: 32315115
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 18.