BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

142 related articles for article (PubMed ID: 28811071)

  • 1. Biological evaluation of 2-pyrazolinyl-1-carbothioamide derivatives against HCT116 human colorectal cancer cell lines and elucidation on QSAR and molecular binding modes.
    Kim BS; Shin SY; Ahn S; Koh D; Lee YH; Lim Y
    Bioorg Med Chem; 2017 Oct; 25(20):5423-5432. PubMed ID: 28811071
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Anticancer and structure-activity relationship evaluation of 3-(naphthalen-2-yl)-N,5-diphenyl-pyrazoline-1-carbothioamide analogs of chalcone.
    Lee Y; Kim BS; Ahn S; Koh D; Lee YH; Shin SY; Lim Y
    Bioorg Chem; 2016 Oct; 68():166-76. PubMed ID: 27543822
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Colorectal anticancer activities of polymethoxylated 3-naphthyl-5-phenylpyrazoline-carbothioamides.
    Shin SY; Ahn S; Yoon H; Jung H; Jung Y; Koh D; Lee YH; Lim Y
    Bioorg Med Chem Lett; 2016 Sep; 26(17):4301-9. PubMed ID: 27476140
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design, synthesis, and biological evaluation of polyphenols with 4,6-diphenylpyrimidin-2-amine derivatives for inhibition of Aurora kinase A.
    Lee YH; Park J; Ahn S; Lee Y; Lee J; Shin SY; Koh D; Lim Y
    Daru; 2019 Jun; 27(1):265-281. PubMed ID: 31154600
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Benzochalcones bearing pyrazoline moieties show anti-colorectal cancer activities and selective inhibitory effects on aurora kinases.
    Shin SY; Yoon H; Hwang D; Ahn S; Kim DW; Koh D; Lee YH; Lim Y
    Bioorg Med Chem; 2013 Nov; 21(22):7018-24. PubMed ID: 24095020
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and cytotoxic activity of some novel steroidal C-17 pyrazolinyl derivatives.
    Fan NJ; Tang JJ; Li H; Li XJ; Luo B; Gao JM
    Eur J Med Chem; 2013 Nov; 69():182-90. PubMed ID: 24021891
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Design, synthesis, biological evaluation and molecular docking studies of novel benzofuran-pyrazole derivatives as anticancer agents.
    Abd El-Karim SS; Anwar MM; Mohamed NA; Nasr T; Elseginy SA
    Bioorg Chem; 2015 Dec; 63():1-12. PubMed ID: 26368040
    [TBL] [Abstract][Full Text] [Related]  

  • 8. New indenopyrazole linked oxadiazole conjugates as anti-pancreatic cancer agents: Design, synthesis, in silico studies including 3D-QSAR analysis.
    Khan I; Ganapathi T; Rehman MM; Shareef MA; Kumar CG; Kamal A
    Bioorg Med Chem Lett; 2021 Jul; 44():128094. PubMed ID: 33964437
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Design and biological evaluation of novel triaryl pyrazoline derivatives with dioxane moiety for selective BRAF
    Li HL; Su MM; Xu YJ; Xu C; Yang YS; Zhu HL
    Eur J Med Chem; 2018 Jul; 155():725-735. PubMed ID: 29940463
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis, biological evaluation, and molecular docking studies of N,1,3-triphenyl-1H-pyrazole-4-carboxamide derivatives as anticancer agents.
    Li X; Lu X; Xing M; Yang XH; Zhao TT; Gong HB; Zhu HL
    Bioorg Med Chem Lett; 2012 Jun; 22(11):3589-93. PubMed ID: 22572580
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Sulfonamide derivatives containing dihydropyrazole moieties selectively and potently inhibit MMP-2/MMP-9: Design, synthesis, inhibitory activity and 3D-QSAR analysis.
    Yan XQ; Wang ZC; Li Z; Wang PF; Qiu HY; Chen LW; Lu XY; Lv PC; Zhu HL
    Bioorg Med Chem Lett; 2015 Oct; 25(20):4664-71. PubMed ID: 26346367
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis and biological evaluation of novel 5-phenyl-1H-pyrazole derivatives as potential BRAF(V600E) inhibitors.
    Wang SF; Zhu YL; Zhu PT; Makawana JA; Zhang YL; Zhao MY; Lv PC; Zhu HL
    Bioorg Med Chem; 2014 Nov; 22(21):6201-8. PubMed ID: 25267006
    [TBL] [Abstract][Full Text] [Related]  

  • 13. In vitro targeting of colon cancer cells using spiropyrazoline oxindoles.
    Nunes RC; Ribeiro CJA; Monteiro Â; Rodrigues CMP; Amaral JD; Santos MMM
    Eur J Med Chem; 2017 Oct; 139():168-179. PubMed ID: 28800455
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis, biological evaluation, and molecular docking studies of N-((1,3-diphenyl-1H-pyrazol-4-yl)methyl)aniline derivatives as novel anticancer agents.
    Huang XF; Lu X; Zhang Y; Song GQ; He QL; Li QS; Yang XH; Wei Y; Zhu HL
    Bioorg Med Chem; 2012 Aug; 20(16):4895-900. PubMed ID: 22819191
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Synthesis, biological evaluation and molecular docking studies of 3-(1,3-diphenyl-1H-pyrazol-4-yl)-N-phenylacrylamide derivatives as inhibitors of HDAC activity.
    Li X; Liu JL; Yang XH; Lu X; Zhao TT; Gong HB; Zhu HL
    Bioorg Med Chem; 2012 Jul; 20(14):4430-6. PubMed ID: 22705022
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Green Synthesis and Molecular Docking of Thiazolyl-thiazole Derivatives as Potential Cytotoxic Agents.
    Gomha SM; Abdelaziz MR; Abdel-Aziz HM; Hassan SA
    Mini Rev Med Chem; 2017; 17(9):805-815. PubMed ID: 28019641
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Design, synthesis and anticancer activity of 1-acyl-3-amino-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole derivatives.
    Bai XG; Yu DK; Wang JX; Zhang H; He HW; Shao RG; Li XM; Wang YC
    Bioorg Med Chem Lett; 2012 Nov; 22(22):6947-51. PubMed ID: 23036956
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Hybrid Pharmacophoric Approach in the Design and Synthesis of Coumarin Linked Pyrazolinyl as Urease Inhibitors, Kinetic Mechanism and Molecular Docking.
    Saeed A; Mahesar PA; Channar PA; Larik FA; Abbas Q; Hassan M; Raza H; Seo SY
    Chem Biodivers; 2017 Aug; 14(8):. PubMed ID: 28574649
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Synthesis and biological evaluation of (3/4-(pyrimidin-2-ylamino)benzoyl)-based hydrazine-1-carboxamide/carbothioamide derivatives as novel RXRα antagonists.
    Qin J; Liu J; Wu C; Xu J; Tang B; Guo K; Chen X; Liu W; Wu T; Zhou H; Fang M; Wu Z
    J Enzyme Inhib Med Chem; 2020 Dec; 35(1):880-896. PubMed ID: 32223461
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Synthesis, EGFR Inhibition and Anti-cancer Activity of New 3,6-dimethyl-1-phenyl-4-(substituted-methoxy)pyrazolo[3,4-d] pyrimidine Derivatives.
    Bakr RB; Mehany ABM; Abdellatif KRA
    Anticancer Agents Med Chem; 2017; 17(10):1389-1400. PubMed ID: 28270084
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.