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4. Studies of H3K4me3 demethylation by KDM5B/Jarid1B/PLU1 reveals strong substrate recognition in vitro and identifies 2,4-pyridine-dicarboxylic acid as an in vitro and in cell inhibitor. Kristensen LH; Nielsen AL; Helgstrand C; Lees M; Cloos P; Kastrup JS; Helin K; Olsen L; Gajhede M FEBS J; 2012 Jun; 279(11):1905-14. PubMed ID: 22420752 [TBL] [Abstract][Full Text] [Related]
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6. Structure of the Arabidopsis JMJ14-H3K4me3 Complex Provides Insight into the Substrate Specificity of KDM5 Subfamily Histone Demethylases. Yang Z; Qiu Q; Chen W; Jia B; Chen X; Hu H; He K; Deng X; Li S; Tao WA; Cao X; Du J Plant Cell; 2018 Jan; 30(1):167-177. PubMed ID: 29233856 [TBL] [Abstract][Full Text] [Related]
7. The oncometabolite 2-hydroxyglutarate inhibits histone lysine demethylases. Chowdhury R; Yeoh KK; Tian YM; Hillringhaus L; Bagg EA; Rose NR; Leung IK; Li XS; Woon EC; Yang M; McDonough MA; King ON; Clifton IJ; Klose RJ; Claridge TD; Ratcliffe PJ; Schofield CJ; Kawamura A EMBO Rep; 2011 May; 12(5):463-9. PubMed ID: 21460794 [TBL] [Abstract][Full Text] [Related]
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10. Histone demethylase lysine demethylase 5B in development and cancer. Han M; Xu W; Cheng P; Jin H; Wang X Oncotarget; 2017 Jan; 8(5):8980-8991. PubMed ID: 27974677 [TBL] [Abstract][Full Text] [Related]
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12. Inhibition of the histone demethylase, KDM5B, directly induces re-expression of tumor suppressor protein HEXIM1 in cancer cells. Montano MM; Yeh IJ; Chen Y; Hernandez C; Kiselar JG; de la Fuente M; Lawes AM; Nieman MT; Kiser PD; Jacobberger J; Exner AA; Lawes MC Breast Cancer Res; 2019 Dec; 21(1):138. PubMed ID: 31805991 [TBL] [Abstract][Full Text] [Related]
13. Depletion of histone demethylase KDM5B inhibits cell proliferation of hepatocellular carcinoma by regulation of cell cycle checkpoint proteins p15 and p27. Wang D; Han S; Peng R; Jiao C; Wang X; Yang X; Yang R; Li X J Exp Clin Cancer Res; 2016 Feb; 35():37. PubMed ID: 26911146 [TBL] [Abstract][Full Text] [Related]
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