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6. A Genome-Wide CRISPR Screen Identifies Genes Critical for Resistance to FLT3 Inhibitor AC220. Hou P; Wu C; Wang Y; Qi R; Bhavanasi D; Zuo Z; Dos Santos C; Chen S; Chen Y; Zheng H; Wang H; Perl A; Guo D; Huang J Cancer Res; 2017 Aug; 77(16):4402-4413. PubMed ID: 28625976 [TBL] [Abstract][Full Text] [Related]
7. Antileukemic Activity of 2-Deoxy-d-Glucose through Inhibition of N-Linked Glycosylation in Acute Myeloid Leukemia with FLT3-ITD or c-KIT Mutations. Larrue C; Saland E; Vergez F; Serhan N; Delabesse E; Mansat-De Mas V; Hospital MA; Tamburini J; Manenti S; Sarry JE; Récher C Mol Cancer Ther; 2015 Oct; 14(10):2364-73. PubMed ID: 26206337 [TBL] [Abstract][Full Text] [Related]
8. Internal tandem duplication of FLT3 deregulates proliferation and differentiation and confers resistance to the FLT3 inhibitor AC220 by Up-regulating RUNX1 expression in hematopoietic cells. Hirade T; Abe M; Onishi C; Taketani T; Yamaguchi S; Fukuda S Int J Hematol; 2016 Jan; 103(1):95-106. PubMed ID: 26590920 [TBL] [Abstract][Full Text] [Related]
9. Upregulation of Flt3 is a passive event in Hoxa9/Meis1-induced acute myeloid leukemia in mice. Staffas A; Arabanian LS; Wei SY; Jansson A; Ståhlman S; Johansson P; Fogelstrand L; Cammenga J; Kuchenbauer F; Palmqvist L Oncogene; 2017 Mar; 36(11):1516-1524. PubMed ID: 27617578 [TBL] [Abstract][Full Text] [Related]
10. Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor for treating acute myeloid leukemia. Keegan K; Li C; Li Z; Ma J; Ragains M; Coberly S; Hollenback D; Eksterowicz J; Liang L; Weidner M; Huard J; Wang X; Alba G; Orf J; Lo MC; Zhao S; Ngo R; Chen A; Liu L; Carlson T; Quéva C; McGee LR; Medina J; Kamb A; Wickramasinghe D; Dai K Mol Cancer Ther; 2014 Apr; 13(4):880-9. PubMed ID: 24526162 [TBL] [Abstract][Full Text] [Related]
11. MZH29 is a novel potent inhibitor that overcomes drug resistance FLT3 mutations in acute myeloid leukemia. Xu B; Zhao Y; Wang X; Gong P; Ge W Leukemia; 2017 Apr; 31(4):913-921. PubMed ID: 27773927 [TBL] [Abstract][Full Text] [Related]
12. Quizartinib (AC220): a promising option for acute myeloid leukemia. Zhou F; Ge Z; Chen B Drug Des Devel Ther; 2019; 13():1117-1125. PubMed ID: 31114157 [TBL] [Abstract][Full Text] [Related]
13. AC220 and AraC cause differential inhibitory dynamics in patient-derived M5-AML with FLT3-ITD and, thus, ultimately distinct therapeutic outcomes. An X; Liu J; Wang N; Wang D; Huang L; Zhang L; Cai J; Wery JP; Zhou D; Zhou J; Li QX Exp Hematol; 2017 Jan; 45():36-44.e2. PubMed ID: 27670587 [TBL] [Abstract][Full Text] [Related]
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15. AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML). Zarrinkar PP; Gunawardane RN; Cramer MD; Gardner MF; Brigham D; Belli B; Karaman MW; Pratz KW; Pallares G; Chao Q; Sprankle KG; Patel HK; Levis M; Armstrong RC; James J; Bhagwat SS Blood; 2009 Oct; 114(14):2984-92. PubMed ID: 19654408 [TBL] [Abstract][Full Text] [Related]
16. Glucocorticoids enhance the antileukemic activity of FLT3 inhibitors in FLT3-mutant acute myeloid leukemia. Gebru MT; Atkinson JM; Young MM; Zhang L; Tang Z; Liu Z; Lu P; Dower CM; Chen L; Annageldiyev C; Sharma A; Imamura Kawasawa Y; Zhao Z; Miller BA; Claxton DF; Wang HG Blood; 2020 Aug; 136(9):1067-1079. PubMed ID: 32396937 [TBL] [Abstract][Full Text] [Related]
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18. Targeting Glutamine Metabolism and Redox State for Leukemia Therapy. Gregory MA; Nemkov T; Park HJ; Zaberezhnyy V; Gehrke S; Adane B; Jordan CT; Hansen KC; D'Alessandro A; DeGregori J Clin Cancer Res; 2019 Jul; 25(13):4079-4090. PubMed ID: 30940653 [TBL] [Abstract][Full Text] [Related]
19. The N676D and G697R mutations in the kinase domain of FLT3 confer resistance to the inhibitor AC220. Pauwels D; Sweron B; Cools J Haematologica; 2012 Nov; 97(11):1773-4. PubMed ID: 22875611 [No Abstract] [Full Text] [Related]
20. Disruption of Wnt/β-Catenin Exerts Antileukemia Activity and Synergizes with FLT3 Inhibition in Jiang X; Mak PY; Mu H; Tao W; Mak DH; Kornblau S; Zhang Q; Ruvolo P; Burks JK; Zhang W; McQueen T; Pan R; Zhou H; Konopleva M; Cortes J; Liu Q; Andreeff M; Carter BZ Clin Cancer Res; 2018 May; 24(10):2417-2429. PubMed ID: 29463558 [No Abstract] [Full Text] [Related] [Next] [New Search]