305 related articles for article (PubMed ID: 28969573)
1. Efficient One-Pot Access to Trisubstituted 2-Benzazepin-3-ones as Constrained Pseudopeptide Analogues and Privileged Scaffolds.
der Poorten OV; Jida M; Tourwe D; Ballet S
Med Chem; 2018; 14(4):400-408. PubMed ID: 28969573
[TBL] [Abstract][Full Text] [Related]
2. Synthesis, biological evaluation, and automated docking of constrained analogues of the opioid peptide H-Dmt-D-Ala-Phe-Gly-NH₂ using the 4- or 5-methyl substituted 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one scaffold.
De Wachter R; de Graaf C; Keresztes A; Vandormael B; Ballet S; Tóth G; Rognan D; Tourwé D
J Med Chem; 2011 Oct; 54(19):6538-47. PubMed ID: 21870874
[TBL] [Abstract][Full Text] [Related]
3. Synthesis of 2,3-Dihydro-1H-2-benzazepin-1-ones and 3H-2-Benzoxepin-1-ones by Isocyanide-Based Multicomponent Reaction/Wittig Sequence Starting from Phosphonium Salt Precursors.
Wang L; Ren ZL; Ding MW
J Org Chem; 2015 Jan; 80(1):641-6. PubMed ID: 25469708
[TBL] [Abstract][Full Text] [Related]
4. T3P-Promoted, Mild, One-Pot Syntheses of Constrained Polycyclic Lactam Dipeptide Analogues via Stereoselective Pictet-Spengler and Meyers Lactamization Reactions.
Jida M; Van der Poorten O; Guillemyn K; Urbanczyk-Lipkowska Z; Tourwé D; Ballet S
Org Lett; 2015 Sep; 17(18):4482-5. PubMed ID: 26322913
[TBL] [Abstract][Full Text] [Related]
5. Ugi 4-CR/Pictet-Spengler reaction as a short route to tryptophan-derived peptidomimetics.
Lesma G; Cecchi R; Crippa S; Giovanelli P; Meneghetti F; Musolino M; Sacchetti A; Silvani A
Org Biomol Chem; 2012 Dec; 10(45):9004-12. PubMed ID: 23073566
[TBL] [Abstract][Full Text] [Related]
6. Enantio- and diastereoselective synthesis of highly substituted benzazepines by a multicomponent strategy coupled with organocatalytic and enzymatic procedures.
Moni L; Banfi L; Basso A; Galatini A; Spallarossa M; Riva R
J Org Chem; 2014 Jan; 79(1):339-51. PubMed ID: 24328226
[TBL] [Abstract][Full Text] [Related]
7. Highly diastereoselective synthesis of 1-carbamoyl-4-aminoindoloazepinone derivatives via the Ugi reaction.
Jida M; Betti C; Urbanczyk-Lipkowska Z; Tourwé D; Ballet S
Org Lett; 2013 Nov; 15(22):5866-9. PubMed ID: 24160404
[TBL] [Abstract][Full Text] [Related]
8. Solid-phase preparation of a pilot library derived from the 2,3,4,5-tetrahydro-1H-benzo[b]azepin-5-amine scaffold.
Boeglin D; Bonnet D; Hibert M
J Comb Chem; 2007; 9(3):487-500. PubMed ID: 17358083
[TBL] [Abstract][Full Text] [Related]
9. Synthesis of Polyheterocyclic Pyrrolo[3,4-b]pyridin-5-ones via a One-Pot (Ugi-3CR/aza Diels-Alder/N-acylation/aromatization/S
Zamudio-Medina A; García-González AN; Herrera-Carrillo GK; Zárate-Zárate D; Benavides-Macías A; Tamariz J; Ibarra IA; Islas-Jácome A; González-Zamora E
Molecules; 2018 Mar; 23(4):. PubMed ID: 29584639
[TBL] [Abstract][Full Text] [Related]
10. One-Pot Synthesis of Indoles by a Sequential Ugi-3CR/Wittig Reaction Starting from Odorless Isocyanide-Substituted Phosphonium Salts.
Yan YM; Rao Y; Ding MW
J Org Chem; 2017 Mar; 82(5):2772-2776. PubMed ID: 28161949
[TBL] [Abstract][Full Text] [Related]
11. Synthesis of 5-hydroxy-2,3,4,5-tetrahydro-[1H]-2-benzazepin-4-ones: selective antagonists of muscarinic (M3) receptors.
Bradshaw B; Evans P; Fletcher J; Lee AT; Mwashimba PG; Oehlrich D; Thomas EJ; Davies RH; Allen BC; Broadley KJ; Hamrouni A; Escargueil C
Org Biomol Chem; 2008 Jun; 6(12):2138-57. PubMed ID: 18528576
[TBL] [Abstract][Full Text] [Related]
12. Bradykinin analogs containing the 4-amino-2-benzazepin-3-one scaffold at the C-terminus.
Ballet S; De Wachter R; Van Rompaey K; Tömböly C; Feytens D; Töth G; Quartara L; Cucchi P; Meini S; Tourwé D
J Pept Sci; 2007 Mar; 13(3):164-70. PubMed ID: 17266049
[TBL] [Abstract][Full Text] [Related]
13. Asymmetric synthesis of enantiomerically pure 2-substituted tetrahydro-3-benzazepines and their affinity to sigma1 receptors.
Husain SM; Fröhlich R; Schepmann D; Wünsch B
J Org Chem; 2009 Apr; 74(7):2788-93. PubMed ID: 19267485
[TBL] [Abstract][Full Text] [Related]
14. Gold(I)-catalyzed benz[c]azepin-4-ol synthesis by intermolecular [5 + 2] cycloaddition.
Iqbal N; Fiksdahl A
J Org Chem; 2013 Aug; 78(16):7885-95. PubMed ID: 23808661
[TBL] [Abstract][Full Text] [Related]
15. Desulfonylative radical ring closure onto aromatics. A modular route to benzazepin-2-ones and 5-arylpiperidin-2-ones.
Charrier N; Liu Z; Zard SZ
Org Lett; 2012 Apr; 14(8):2018-21. PubMed ID: 22463494
[TBL] [Abstract][Full Text] [Related]
16. Investigation of the one-pot synthesis of quinolin-2-(1H)-ones and the discovery of a variation of the three-component Ugi reaction.
Gordon CP; Young KA; Hizartzidis L; Deane FM; McCluskey A
Org Biomol Chem; 2011 Mar; 9(5):1419-28. PubMed ID: 21427800
[TBL] [Abstract][Full Text] [Related]
17. Novel selective human melanocortin-3 receptor ligands: use of the 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one (Aba) scaffold.
Ballet S; Mayorov AV; Cai M; Tymecka D; Chandler KB; Palmer ES; Rompaey KV; Misicka A; Tourwé D; Hruby VJ
Bioorg Med Chem Lett; 2007 May; 17(9):2492-8. PubMed ID: 17314042
[TBL] [Abstract][Full Text] [Related]
18. Synthesis and biological evaluation of constrained analogues of the opioid peptide H-Tyr-D-Ala-Phe-Gly-NH2 using the 4-amino-2-benzazepin-3-one scaffold.
Ballet S; Frycia A; Piron J; Chung NN; Schiller PW; Kosson P; Lipkowski AW; Tourwé D
J Pept Res; 2005 Nov; 66(5):222-30. PubMed ID: 16218989
[TBL] [Abstract][Full Text] [Related]
19. Efficient synthesis of (S)-4-phthalimido-1,3,4,5-tetrahydro-8-(2,6-dichlorobenzyloxy)- 3-oxo-2H-2-benzazepin-2-acetic acid (PHt-Hba(2,6-Cl2-Bn)-Gly-OH).
Casimir JR; Tourwé D; Iterbeke K; Guichard G; Briand JP
J Org Chem; 2000 Oct; 65(20):6487-92. PubMed ID: 11052092
[TBL] [Abstract][Full Text] [Related]
20. Synthesis of Highly Substituted Imidazole Uracil Containing Molecules via Ugi-4CR and Passerini-3CR.
Madhavachary R; Zarganes-Tzitzikas T; Patil P; Kurpiewska K; Kalinowska-Tłuścik J; Dömling A
ACS Comb Sci; 2018 Apr; 20(4):192-196. PubMed ID: 29457887
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
