182 related articles for article (PubMed ID: 29024590)
1. Efficient Synthesis of 1,9-Substituted Benzo[h][1,6]naphthyridin-2(1H)-ones and Evaluation of their Plasmodium falciparum Gametocytocidal Activities.
Li H; Sun W; Huang X; Lu X; Patel PR; Kim M; Orr MJ; Fisher RM; Tanaka TQ; McKew JC; Simeonov A; Sanderson PE; Zheng W; Williamson KC; Huang W
ACS Comb Sci; 2017 Dec; 19(12):748-754. PubMed ID: 29024590
[TBL] [Abstract][Full Text] [Related]
2. In vitro evaluation of imidazo[4,5-c]quinolin-2-ones as gametocytocidal antimalarial agents.
Patel PR; Sun W; Kim M; Huang X; Sanderson PE; Tanaka TQ; McKew JC; Simeonov A; Williamson KC; Zheng W; Huang W
Bioorg Med Chem Lett; 2016 Jun; 26(12):2907-2911. PubMed ID: 27156776
[TBL] [Abstract][Full Text] [Related]
3. Antimalarial and cytotoxic activities of chiral triamines.
Dellai A; Appel J; Bouraoui A; Croft S; Nefzi A
Bioorg Med Chem Lett; 2013 Aug; 23(16):4579-82. PubMed ID: 23835293
[TBL] [Abstract][Full Text] [Related]
4. Potent Plasmodium falciparum gametocytocidal activity of diaminonaphthoquinones, lead antimalarial chemotypes identified in an antimalarial compound screen.
Tanaka TQ; Guiguemde WA; Barnett DS; Maron MI; Min J; Connelly MC; Suryadevara PK; Guy RK; Williamson KC
Antimicrob Agents Chemother; 2015 Mar; 59(3):1389-97. PubMed ID: 25512421
[TBL] [Abstract][Full Text] [Related]
5. Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials.
van der Watt ME; Reader J; Churchyard A; Nondaba SH; Lauterbach SB; Niemand J; Abayomi S; van Biljon RA; Connacher JI; van Wyk RDJ; Le Manach C; Paquet T; González Cabrera D; Brunschwig C; Theron A; Lozano-Arias S; Rodrigues JFI; Herreros E; Leroy D; Duffy J; Street LJ; Chibale K; Mancama D; Coetzer TL; Birkholtz LM
J Antimicrob Chemother; 2018 May; 73(5):1279-1290. PubMed ID: 29420756
[TBL] [Abstract][Full Text] [Related]
6. Novel lead structures with both Plasmodium falciparum gametocytocidal and asexual blood stage activity identified from high throughput compound screening.
Sun W; Huang X; Li H; Tawa G; Fisher E; Tanaka TQ; Shinn P; Huang W; Williamson KC; Zheng W
Malar J; 2017 Apr; 16(1):147. PubMed ID: 28407766
[TBL] [Abstract][Full Text] [Related]
7. Structure-activity relationships amongst 4-position quinoline methanol antimalarials that inhibit the growth of drug sensitive and resistant strains of Plasmodium falciparum.
Milner E; McCalmont W; Bhonsle J; Caridha D; Carroll D; Gardner S; Gerena L; Gettayacamin M; Lanteri C; Luong T; Melendez V; Moon J; Roncal N; Sousa J; Tungtaeng A; Wipf P; Dow G
Bioorg Med Chem Lett; 2010 Feb; 20(4):1347-51. PubMed ID: 20097070
[TBL] [Abstract][Full Text] [Related]
8. Chemical signatures and new drug targets for gametocytocidal drug development.
Sun W; Tanaka TQ; Magle CT; Huang W; Southall N; Huang R; Dehdashti SJ; McKew JC; Williamson KC; Zheng W
Sci Rep; 2014 Jan; 4():3743. PubMed ID: 24434750
[TBL] [Abstract][Full Text] [Related]
9. Luciferase-Based, High-Throughput Assay for Screening and Profiling Transmission-Blocking Compounds against Plasmodium falciparum Gametocytes.
Lucantoni L; Fidock DA; Avery VM
Antimicrob Agents Chemother; 2016 Apr; 60(4):2097-107. PubMed ID: 26787698
[TBL] [Abstract][Full Text] [Related]
10. [Benzo[c][2,7]naphthyridine-2-yl-, 5-yl- and 2,5-diyl novaldiamines--synthesis and investigation of anti-malarial activity].
Görlitzer K; Enge CH; Jones PG; Jomaa H; Wiesner J
Pharmazie; 2006 Dec; 61(12):975-80. PubMed ID: 17283651
[TBL] [Abstract][Full Text] [Related]
11. Design, synthesis and biological evaluation of small molecules as potent glucosidase inhibitors.
Hati S; Madurkar SM; Bathula C; Thulluri C; Agarwal R; Siddiqui FA; Dangi P; Adepally U; Singh A; Singh S; Sen S
Eur J Med Chem; 2015 Jul; 100():188-96. PubMed ID: 26087029
[TBL] [Abstract][Full Text] [Related]
12. Synthesis and structure-activity relationships of 7-substituted 3-(2, 6-dichlorophenyl)-1,6-naphthyridin-2(1H)-ones as selective inhibitors of pp60(c-src).
Thompson AM; Rewcastle GW; Boushelle SL; Hartl BG; Kraker AJ; Lu GH; Batley BL; Panek RL; Showalter HD; Denny WA
J Med Chem; 2000 Aug; 43(16):3134-47. PubMed ID: 10956222
[TBL] [Abstract][Full Text] [Related]
13. Whole-cell in vitro screening for gametocytocidal compounds.
Lucantoni L; Avery V
Future Med Chem; 2012 Dec; 4(18):2337-60. PubMed ID: 23234555
[TBL] [Abstract][Full Text] [Related]
14. Pharmacophore based discovery of potential antimalarial agent targeting haem detoxification pathway.
Acharya BN; Saraswat D; Kaushik MP
Eur J Med Chem; 2008 Dec; 43(12):2840-52. PubMed ID: 18395298
[TBL] [Abstract][Full Text] [Related]
15. A quantitative high throughput assay for identifying gametocytocidal compounds.
Tanaka TQ; Dehdashti SJ; Nguyen DT; McKew JC; Zheng W; Williamson KC
Mol Biochem Parasitol; 2013 Mar; 188(1):20-5. PubMed ID: 23454872
[TBL] [Abstract][Full Text] [Related]
16. Methylene blue induced morphological deformations in Plasmodium falciparum gametocytes: implications for transmission-blocking.
Wadi I; Pillai CR; Anvikar AR; Sinha A; Nath M; Valecha N
Malar J; 2018 Jan; 17(1):11. PubMed ID: 29310655
[TBL] [Abstract][Full Text] [Related]
17. [Benzo[c][2,7]naphthyridine-5-yl-amines and benzo[h][1,6]naphthyridine-5-yl-amines--potential antimalarials].
Görlitzer K; Bode M; Jones PG; Jomaa H; Wiesner J
Pharmazie; 2007 Jan; 62(1):15-26. PubMed ID: 17294807
[TBL] [Abstract][Full Text] [Related]
18. [Benzo[c][2,7]naphthyridine-5-yl-arylamines-phenol Mannich bases of the amodiaquine-, cycloquine- and pyronaridine-type].
Görlitzer K; Enge C; Jones PG; Jomaa H; Wiesner J
Pharmazie; 2007 Feb; 62(2):89-93. PubMed ID: 17341024
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and evaluation of the performance of a small molecule library based on diverse tropane-related scaffolds.
Lowe RA; Taylor D; Chibale K; Nelson A; Marsden SP
Bioorg Med Chem; 2020 May; 28(9):115442. PubMed ID: 32209295
[TBL] [Abstract][Full Text] [Related]
20. Novel synthetic route for antimalarial benzo[a]phenoxazine derivative SSJ-183 and two active metabolites.
Mizukawa Y; Ge JF; Bakar Md A; Itoh I; Scheurer C; Wittlin S; Brun R; Matsuoka H; Ihara M
Bioorg Med Chem; 2014 Jul; 22(14):3749-52. PubMed ID: 24856305
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
