182 related articles for article (PubMed ID: 29258235)
1. GPCR Modulation of Thieno[2,3-b]pyridine Anti-Proliferative Agents.
Zafar A; Sari S; Leung E; Pilkington LI; van Rensburg M; Barker D; Reynisson J
Molecules; 2017 Dec; 22(12):. PubMed ID: 29258235
[TBL] [Abstract][Full Text] [Related]
2. Investigation into Improving the Aqueous Solubility of the Thieno[2,3-b]pyridine Anti-Proliferative Agents.
Zafar A; Pilkington LI; Haverkate NA; van Rensburg M; Leung E; Kumara S; Denny WA; Barker D; Alsuraifi A; Hoskins C; Reynisson J
Molecules; 2018 Jan; 23(1):. PubMed ID: 29324695
[TBL] [Abstract][Full Text] [Related]
3. 3-Amino-thieno[2,3-b]pyridines as microtubule-destabilising agents: Molecular modelling and biological evaluation in the sea urchin embryo and human cancer cells.
Eurtivong C; Semenov V; Semenova M; Konyushkin L; Atamanenko O; Reynisson J; Kiselyov A
Bioorg Med Chem; 2017 Jan; 25(2):658-664. PubMed ID: 27956038
[TBL] [Abstract][Full Text] [Related]
4. Identification of anticancer agents based on the thieno[2,3-b]pyridine and 1H-pyrazole molecular scaffolds.
Eurtivong C; Reynisdóttir I; Kuczma S; Furkert DP; Brimble MA; Reynisson J
Bioorg Med Chem; 2016 Aug; 24(16):3521-6. PubMed ID: 27288184
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and cytotoxicity of thieno[2,3-b]pyridine and furo[2,3-b]pyridine derivatives.
Hung JM; Arabshahi HJ; Leung E; Reynisson J; Barker D
Eur J Med Chem; 2014 Oct; 86():420-37. PubMed ID: 25194934
[TBL] [Abstract][Full Text] [Related]
6. Design, synthesis, molecular modeling and biological evaluation of novel 1H-pyrazolo[3,4-b]pyridine derivatives as potential anticancer agents.
Eissa IH; El-Naggar AM; El-Hashash MA
Bioorg Chem; 2016 Aug; 67():43-56. PubMed ID: 27253830
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and antiproliferative activity of 2-chlorophenyl carboxamide thienopyridines.
van Rensburg M; Leung E; Haverkate NA; Eurtivong C; Pilkington LI; Reynisson J; Barker D
Bioorg Med Chem Lett; 2017 Jan; 27(2):135-138. PubMed ID: 27979592
[TBL] [Abstract][Full Text] [Related]
8. Synthesis and cytotoxicity of thieno[2,3-b]quinoline-2-carboxamide and cycloalkyl[b]thieno[3,2-e]pyridine-2-carboxamide derivatives.
Leung E; Pilkington LI; van Rensburg M; Jeon CY; Song M; Arabshahi HJ; De Zoysa GH; Sarojini V; Denny WA; Reynisson J; Barker D
Bioorg Med Chem; 2016 Mar; 24(5):1142-54. PubMed ID: 26853836
[TBL] [Abstract][Full Text] [Related]
9. Current assessment of docking into GPCR crystal structures and homology models: successes, challenges, and guidelines.
Beuming T; Sherman W
J Chem Inf Model; 2012 Dec; 52(12):3263-77. PubMed ID: 23121495
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and biological evaluation of curcumin inspired imidazo[1,2-a]pyridine analogues as tubulin polymerization inhibitors.
Ramya PVS; Guntuku L; Angapelly S; Digwal CS; Lakshmi UJ; Sigalapalli DK; Babu BN; Naidu VGM; Kamal A
Eur J Med Chem; 2018 Jan; 143():216-231. PubMed ID: 29174816
[TBL] [Abstract][Full Text] [Related]
11. Discovery of novel 2-phenyl-imidazo[1,2-a]pyridine analogues targeting tubulin polymerization as antiproliferative agents.
An W; Wang W; Yu T; Zhang Y; Miao Z; Meng T; Shen J
Eur J Med Chem; 2016 Apr; 112():367-372. PubMed ID: 26927488
[TBL] [Abstract][Full Text] [Related]
12. Disruption of Crystal Packing in Thieno[2,3-
Haverkate NA; Leung E; Pilkington LI; Barker D
Molecules; 2022 Jan; 27(3):. PubMed ID: 35164101
[TBL] [Abstract][Full Text] [Related]
13. X-ray structure breakthroughs in the GPCR transmembrane region.
Topiol S; Sabio M
Biochem Pharmacol; 2009 Jul; 78(1):11-20. PubMed ID: 19447219
[TBL] [Abstract][Full Text] [Related]
14. Synthesis, and docking studies of phenylpyrimidine-carboxamide derivatives bearing 1H-pyrrolo[2,3-b]pyridine moiety as c-Met inhibitors.
Zhu W; Wang W; Xu S; Wang J; Tang Q; Wu C; Zhao Y; Zheng P
Bioorg Med Chem; 2016 Apr; 24(8):1749-56. PubMed ID: 26964675
[TBL] [Abstract][Full Text] [Related]
15. Anti-proliferative potential of cyclotetrapeptides from Bacillus velezensis RA5401 and their molecular docking on G-Protein-Coupled Receptors.
Rehman NU; Abed RMM; Hussain H; Khan HY; Khan A; Khan AL; Ali M; Al-Nasri A; Al-Harrasi K; Al-Rawahi AN; Wadood A; Al-Rawahi A; Al-Harrasi A
Microb Pathog; 2018 Oct; 123():419-425. PubMed ID: 30075241
[TBL] [Abstract][Full Text] [Related]
16. Design, synthesis, and molecular docking study of 3H-imidazole[4,5-c]pyridine derivatives as CDK2 inhibitors.
Wu YZ; Ying HZ; Xu L; Cheng G; Chen J; Hu YZ; Liu T; Dong XW
Arch Pharm (Weinheim); 2018 Jun; 351(6):e1700381. PubMed ID: 29708285
[TBL] [Abstract][Full Text] [Related]
17. Design, synthesis, biological evaluation and molecular modeling of novel 2-amino-4-(1-phenylethoxy) pyridine derivatives as potential ROS1 inhibitors.
Tian Y; Zhang T; Long L; Li Z; Wan S; Wang G; Yu Y; Hou J; Wu X; Zhang J
Eur J Med Chem; 2018 Jan; 143():182-199. PubMed ID: 29174814
[TBL] [Abstract][Full Text] [Related]
18. Exploration on natural product anibamine side chain modification toward development of novel CCR5 antagonists and potential anti-prostate cancer agents.
Xu GG; Zaidi SA; Zhang F; Singh S; Raborg TJ; Yuan Y; Zhang Y
Bioorg Med Chem Lett; 2015 Sep; 25(17):3721-5. PubMed ID: 26096680
[TBL] [Abstract][Full Text] [Related]
19. Synthesis and biological evaluation of pyrrolo[2,3-b]pyridine analogues as antiproliferative agents and their interaction with calf thymus DNA.
Narva S; Chitti S; Bala BR; Alvala M; Jain N; Kondapalli VG
Eur J Med Chem; 2016 May; 114():220-31. PubMed ID: 26994690
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and Anti-Proliferative Activity of 5-Benzoyl and 5-Benzylhydroxy Derivatives of 3-Amino-2-Arylcarboxamido-Thieno[2-3-
Morphet B; Rees SWP; Haverkate NA; Aziz H; Leung E; Pilkington LI; Barker D
Int J Mol Sci; 2023 Jul; 24(14):. PubMed ID: 37511173
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]