These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
199 related articles for article (PubMed ID: 29459279)
1. Cyclic peptide inhibitors of lysine-specific demethylase 1 with improved potency identified by alanine scanning mutagenesis. Kumarasinghe IR; Woster PM Eur J Med Chem; 2018 Mar; 148():210-220. PubMed ID: 29459279 [TBL] [Abstract][Full Text] [Related]
2. Annual review of lysine-specific demethylase 1 (LSD1/KDM1A) inhibitors in 2021. Song Y; Zhang H; Yang X; Shi Y; Yu B Eur J Med Chem; 2022 Jan; 228():114042. PubMed ID: 34915312 [TBL] [Abstract][Full Text] [Related]
5. LSD1 promotes S-phase entry and tumorigenesis via chromatin co-occupation with E2F1 and selective H3K9 demethylation. He Y; Zhao Y; Wang L; Bohrer LR; Pan Y; Wang L; Huang H Oncogene; 2018 Jan; 37(4):534-543. PubMed ID: 28991226 [TBL] [Abstract][Full Text] [Related]
6. A comprehensive review of lysine-specific demethylase 1 and its roles in cancer. Hosseini A; Minucci S Epigenomics; 2017 Aug; 9(8):1123-1142. PubMed ID: 28699367 [TBL] [Abstract][Full Text] [Related]
7. Structure-activity study for (bis)ureidopropyl- and (bis)thioureidopropyldiamine LSD1 inhibitors with 3-5-3 and 3-6-3 carbon backbone architectures. Nowotarski SL; Pachaiyappan B; Holshouser SL; Kutz CJ; Li Y; Huang Y; Sharma SK; Casero RA; Woster PM Bioorg Med Chem; 2015 Apr; 23(7):1601-12. PubMed ID: 25725609 [TBL] [Abstract][Full Text] [Related]
8. Inhibitors of LSD1 as a potential therapy for acute myeloid leukemia. Przespolewski A; Wang ES Expert Opin Investig Drugs; 2016 Jul; 25(7):771-80. PubMed ID: 27077938 [TBL] [Abstract][Full Text] [Related]
9. (Bis)urea and (bis)thiourea inhibitors of lysine-specific demethylase 1 as epigenetic modulators. Sharma SK; Wu Y; Steinbergs N; Crowley ML; Hanson AS; Casero RA; Woster PM J Med Chem; 2010 Jul; 53(14):5197-212. PubMed ID: 20568780 [TBL] [Abstract][Full Text] [Related]
10. Reversible Lysine Specific Demethylase 1 (LSD1) Inhibitors: A Promising Wrench to Impair LSD1. Dai XJ; Liu Y; Xue LP; Xiong XP; Zhou Y; Zheng YC; Liu HM J Med Chem; 2021 Mar; 64(5):2466-2488. PubMed ID: 33619958 [TBL] [Abstract][Full Text] [Related]
11. Synthesis and evaluation of novel cyclic Peptide inhibitors of lysine-specific demethylase 1. Kumarasinghe IR; Woster PM ACS Med Chem Lett; 2014 Jan; 5(1):29-33. PubMed ID: 24883177 [TBL] [Abstract][Full Text] [Related]
12. A Systematic Review of Histone Lysine-Specific Demethylase 1 and Its Inhibitors. Zheng YC; Ma J; Wang Z; Li J; Jiang B; Zhou W; Shi X; Wang X; Zhao W; Liu HM Med Res Rev; 2015 Sep; 35(5):1032-71. PubMed ID: 25990136 [TBL] [Abstract][Full Text] [Related]
13. High-throughput TR-FRET assays for identifying inhibitors of LSD1 and JMJD2C histone lysine demethylases. Yu V; Fisch T; Long AM; Tang J; Lee JH; Hierl M; Chen H; Yakowec P; Schwandner R; Emkey R J Biomol Screen; 2012 Jan; 17(1):27-38. PubMed ID: 21859682 [TBL] [Abstract][Full Text] [Related]
14. Discovery of tranylcypromine analogs with an acylhydrazone substituent as LSD1 inactivators: Design, synthesis and their biological evaluation. Sun K; Peng JD; Suo FZ; Zhang T; Fu YD; Zheng YC; Liu HM Bioorg Med Chem Lett; 2017 Nov; 27(22):5036-5039. PubMed ID: 29037950 [TBL] [Abstract][Full Text] [Related]
15. The epigenetic promotion of osteogenic differentiation of human adipose-derived stem cells by the genetic and chemical blockade of histone demethylase LSD1. Ge W; Liu Y; Chen T; Zhang X; Lv L; Jin C; Jiang Y; Shi L; Zhou Y Biomaterials; 2014 Jul; 35(23):6015-25. PubMed ID: 24794925 [TBL] [Abstract][Full Text] [Related]
16. Irreversible LSD1 Inhibitors: Application of Tranylcypromine and Its Derivatives in Cancer Treatment. Zheng YC; Yu B; Jiang GZ; Feng XJ; He PX; Chu XY; Zhao W; Liu HM Curr Top Med Chem; 2016; 16(19):2179-88. PubMed ID: 26881714 [TBL] [Abstract][Full Text] [Related]
17. Development and crystallographic evaluation of histone H3 peptide with N-terminal serine substitution as a potent inhibitor of lysine-specific demethylase 1. Amano Y; Kikuchi M; Sato S; Yokoyama S; Umehara T; Umezawa N; Higuchi T Bioorg Med Chem; 2017 May; 25(9):2617-2624. PubMed ID: 28336409 [TBL] [Abstract][Full Text] [Related]
18. Novel oligoamine analogues inhibit lysine-specific demethylase 1 and induce reexpression of epigenetically silenced genes. Huang Y; Stewart TM; Wu Y; Baylin SB; Marton LJ; Perkins B; Jones RJ; Woster PM; Casero RA Clin Cancer Res; 2009 Dec; 15(23):7217-28. PubMed ID: 19934284 [TBL] [Abstract][Full Text] [Related]
19. Regulation of tissue factor pathway inhibitor-2 (TFPI-2) expression by lysine-specific demethylase 1 and 2 (LSD1 and LSD2). Mino K; Nishimura S; Ninomiya S; Tujii H; Matsumori Y; Tsuchida M; Hosoi M; Koseki K; Wada S; Hasegawa M; Sasaki R; Murakami-Yamaguchi Y; Narita H; Suzuki T; Miyata N; Mizukami T Biosci Biotechnol Biochem; 2014; 78(6):1010-7. PubMed ID: 25036127 [TBL] [Abstract][Full Text] [Related]
20. Tranylcypromine Based Lysine-Specific Demethylase 1 Inhibitor: Summary and Perspective. Dai XJ; Liu Y; Xiong XP; Xue LP; Zheng YC; Liu HM J Med Chem; 2020 Dec; 63(23):14197-14215. PubMed ID: 32931269 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]