143 related articles for article (PubMed ID: 29558439)
1. Potent GH20 N-Acetyl-β-d-hexosaminidase Inhibitors: N-Substituted 3-acetamido-4-amino-5-hydroxymethyl-cyclopentanediols.
Weber P; Nasseri SA; Pabst BM; Torvisco A; Müller P; Paschke E; Tschernutter M; Windischhofer W; Withers SG; Wrodnigg TM; Stütz AE
Molecules; 2018 Mar; 23(3):. PubMed ID: 29558439
[TBL] [Abstract][Full Text] [Related]
2. N-Substituted 5-amino-1-hydroxymethyl-cyclopentanetriols: A new family of activity promotors for a G
Schalli M; Tysoe C; Fischer R; Pabst BM; Thonhofer M; Paschke E; Rappitsch T; Stütz AE; Tschernutter M; Windischhofer W; Withers SG
Carbohydr Res; 2017 Apr; 443-444():15-22. PubMed ID: 28319682
[TBL] [Abstract][Full Text] [Related]
3. Exploring unsymmetrical dyads as efficient inhibitors against the insect β-N-acetyl-D-hexosaminidase OfHex2.
Chen Q; Guo P; Xu L; Liu T; Qian X; Yang Q
Biochimie; 2014 Feb; 97():152-62. PubMed ID: 24140956
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, evaluation, and mechanism of N,N,N-trimethyl-D-glucosamine-(1→4)-chitooligosaccharides as selective inhibitors of glycosyl hydrolase family 20 β-N-acetyl-D-hexosaminidases.
Yang Y; Liu T; Yang Y; Wu Q; Yang Q; Yu B
Chembiochem; 2011 Feb; 12(3):457-67. PubMed ID: 21290547
[TBL] [Abstract][Full Text] [Related]
5. Diaminocyclopentane - l-Lysine Adducts: Potent and selective inhibitors of human O-GlcNAcase.
Weber P; Bojarová P; Brouzdová J; Křen V; Kulik N; Stütz AE; Thonhofer M; Wrodnigg TM
Bioorg Chem; 2024 Jul; 148():107452. PubMed ID: 38763001
[TBL] [Abstract][Full Text] [Related]
6. Synthesis of NAG-thiazoline-derived inhibitors for β-N-acetyl-d-hexosaminidases.
Kong H; Chen W; Lu H; Yang Q; Dong Y; Wang D; Zhang J
Carbohydr Res; 2015 Sep; 413():135-44. PubMed ID: 26142545
[TBL] [Abstract][Full Text] [Related]
7. Structural variation of the 3-acetamido-4,5,6-trihydroxyazepane iminosugar through epimerization and
Bouquet J; Auberger N; Ashmus R; King D; Bordes A; Fontelle N; Nakagawa S; Madden Z; Proceviat C; Kato A; Désiré J; Vocadlo DJ; Blériot Y
Org Biomol Chem; 2022 Jan; 20(3):619-629. PubMed ID: 34940771
[TBL] [Abstract][Full Text] [Related]
8. Active-pocket size differentiating insectile from bacterial chitinolytic β-N-acetyl-D-hexosaminidases.
Liu T; Zhang H; Liu F; Chen L; Shen X; Yang Q
Biochem J; 2011 Sep; 438(3):467-74. PubMed ID: 21692744
[TBL] [Abstract][Full Text] [Related]
9. Modifying the phenyl group of PUGNAc: reactivity tuning to deliver selective inhibitors for N-acetyl-D-glucosaminidases.
Hattie M; Cekic N; Debowski AW; Vocadlo DJ; Stubbs KA
Org Biomol Chem; 2016 Mar; 14(12):3193-7. PubMed ID: 26924385
[TBL] [Abstract][Full Text] [Related]
10. Amino(hydroxymethyl)cyclopentanetriols, an emerging class of potent glycosidase inhibitors--Part I: Synthesis and evaluation of beta-D-pyranoside analogues in the manno, gluco, galacto, and GlcNAc series.
Kleban M; Hilgers P; Greul JN; Kugler RD; Li J; Picasso S; Vogel P; Jäger V
Chembiochem; 2001 May; 2(5):365-8. PubMed ID: 11828465
[No Abstract] [Full Text] [Related]
11. Synthesis and high-throughput screening of N-acetyl-beta-hexosaminidase inhibitor libraries targeting osteoarthritis.
Liu J; Numa MM; Liu H; Huang SJ; Sears P; Shikhman AR; Wong CH
J Org Chem; 2004 Sep; 69(19):6273-83. PubMed ID: 15357586
[TBL] [Abstract][Full Text] [Related]
12. Tautomeric modification of GlcNAc-thiazoline.
Knapp S; Abdo M; Ajayi K; Huhn RA; Emge TJ; Kim EJ; Hanover JA
Org Lett; 2007 Jun; 9(12):2321-4. PubMed ID: 17508759
[TBL] [Abstract][Full Text] [Related]
13. A divergent synthesis of 2-acyl derivatives of PUGNAc yields selective inhibitors of O-GlcNAcase.
Stubbs KA; Zhang N; Vocadlo DJ
Org Biomol Chem; 2006 Mar; 4(5):839-45. PubMed ID: 16493467
[TBL] [Abstract][Full Text] [Related]
14. Stereoselective synthesis of 2-acetamido-1,2-dideoxynojirimycin (DNJNAc) and ureido-DNJNAc derivatives as new hexosaminidase inhibitors.
de la Fuente A; Mena-Barragán T; Farrar-Tobar RA; Verdaguer X; García Fernández JM; Ortiz Mellet C; Riera A
Org Biomol Chem; 2015 Jun; 13(23):6500-10. PubMed ID: 25975710
[TBL] [Abstract][Full Text] [Related]
15. A new type of pharmacological chaperone for G
Schalli M; Weber P; Tysoe C; Pabst BM; Thonhofer M; Paschke E; Stütz AE; Tschernutter M; Windischhofer W; Withers SG
Bioorg Med Chem Lett; 2017 Aug; 27(15):3431-3435. PubMed ID: 28600215
[TBL] [Abstract][Full Text] [Related]
16. Synthesis of NAM-thiazoline derivatives as novel O-GlcNAcase inhibitors.
Kong H; Chen W; Liu T; Lu H; Yang Q; Dong Y; Liang X; Jin S; Zhang J
Carbohydr Res; 2016 Jun; 429():54-61. PubMed ID: 27233493
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and biological evaluation of ureido and thioureido derivatives of 2-amino-2-deoxy-D-glucose and related aminoalcohols as N-acetyl-beta-D-hexosaminidase inhibitors.
Tournaire-Arellano C; Hage SY; Valès P; Caujolle R; Sanon A; Bories C; Loiseau PM
Carbohydr Res; 1998 Dec; 314(1-2):47-63. PubMed ID: 10230037
[TBL] [Abstract][Full Text] [Related]
18. N-acetyl-beta-D-hexosaminidase from Trichomonas vaginalis: substrate specificity and activity of inhibitors.
Sanon A; Tournaire-Arellano C; El Hage SY; Bories C; Caujolle R; Loiseau PM
Biomed Pharmacother; 2005 Jun; 59(5):245-8. PubMed ID: 15890491
[TBL] [Abstract][Full Text] [Related]
19. Design and synthesis of thiazolylhydrazone derivatives as inhibitors of chitinolytic N-acetyl-β-d-hexosaminidase.
Yang H; Liu T; Qi H; Huang Z; Hao Z; Ying J; Yang Q; Qian X
Bioorg Med Chem; 2018 Nov; 26(20):5420-5426. PubMed ID: 30274940
[TBL] [Abstract][Full Text] [Related]
20. Amino(hydroxymethyl)cyclopentanetriols, an emerging class of potent glycosidase inhibitors--Part II: Synthesis, evaluation, and optimization of beta-D-galactopyranoside analogues.
Greul JN; Kleban M; Schneider B; Picasso S; Jäger V
Chembiochem; 2001 May; 2(5):368-70. PubMed ID: 11828466
[No Abstract] [Full Text] [Related]
[Next] [New Search]