BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

220 related articles for article (PubMed ID: 29660786)

  • 1. Activity and selectivity cliffs for DPP-IV inhibitors: Lessons we can learn from SAR studies and their application to virtual screening.
    Ojeda-Montes MJ; Gimeno A; Tomas-Hernández S; Cereto-Massagué A; Beltrán-Debón R; Valls C; Mulero M; Pujadas G; Garcia-Vallvé S
    Med Res Rev; 2018 Sep; 38(6):1874-1915. PubMed ID: 29660786
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Identification of novel human dipeptidyl peptidase-IV inhibitors of natural origin (part I): virtual screening and activity assays.
    Guasch L; Ojeda MJ; González-Abuín N; Sala E; Cereto-Massagué A; Mulero M; Valls C; Pinent M; Ardévol A; Garcia-Vallvé S; Pujadas G
    PLoS One; 2012; 7(9):e44971. PubMed ID: 22984596
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Dipeptidyl peptidase IV and its inhibitors: therapeutics for type 2 diabetes and what else?
    Juillerat-Jeanneret L
    J Med Chem; 2014 Mar; 57(6):2197-212. PubMed ID: 24099035
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Design, synthesis and anti-diabetic activity of triazolotriazine derivatives as dipeptidyl peptidase-4 (DPP-4) inhibitors.
    Patel BD; Bhadada SV; Ghate MD
    Bioorg Chem; 2017 Jun; 72():345-358. PubMed ID: 28302310
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Recent progress of the development of dipeptidyl peptidase-4 inhibitors for the treatment of type 2 diabetes mellitus.
    Li N; Wang LJ; Jiang B; Li XQ; Guo CL; Guo SJ; Shi DY
    Eur J Med Chem; 2018 May; 151():145-157. PubMed ID: 29609120
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Identification of novel dipeptidyl peptidase IV (DPP-IV) inhibitory peptides in camel milk protein hydrolysates.
    Nongonierma AB; Paolella S; Mudgil P; Maqsood S; FitzGerald RJ
    Food Chem; 2018 Apr; 244():340-348. PubMed ID: 29120791
    [TBL] [Abstract][Full Text] [Related]  

  • 7. The discovery of novel 5,6,5- and 5,5,6-tricyclic pyrrolidines as potent and selective DPP-4 inhibitors.
    Cox JM; Chu HD; Kuethe JT; Gao YD; Scapin G; Eiermann G; He H; Li X; Lyons KA; Metzger J; Petrov A; Wu JK; Xu S; Sinha-Roy R; Weber AE; Biftu T
    Bioorg Med Chem Lett; 2016 Jun; 26(11):2622-6. PubMed ID: 27106708
    [TBL] [Abstract][Full Text] [Related]  

  • 8. DPP-IV Inhibitory Potentials of Flavonol Glycosides Isolated from the Seeds of
    Kim BR; Kim HY; Choi I; Kim JB; Jin CH; Han AR
    Molecules; 2018 Aug; 23(8):. PubMed ID: 30103438
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel hydrazine derivatives as selective DPP-IV inhibitors: findings from virtual screening and validation through molecular dynamics simulations.
    Tanwar O; Deora GS; Tanwar L; Kumar G; Janardhan S; Alam M; Shaquiquzzaman ; Akhter M
    J Mol Model; 2014 Apr; 20(4):2118. PubMed ID: 24687332
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Finding a Potential Dipeptidyl Peptidase-4 (DPP-4) Inhibitor for Type-2 Diabetes Treatment Based on Molecular Docking, Pharmacophore Generation, and Molecular Dynamics Simulation.
    Meduru H; Wang YT; Tsai JJ; Chen YC
    Int J Mol Sci; 2016 Jun; 17(6):. PubMed ID: 27304951
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Discovery of tight-binding competitive inhibitors of dipeptidyl peptidase IV.
    Pascual Alonso I; Valiente PA; Valdés-Tresanco ME; Arrebola Y; Almeida García F; Díaz L; García G; Guirola O; Pastor D; Bergado G; Sánchez B; Charli JL
    Int J Biol Macromol; 2022 Jan; 196():120-130. PubMed ID: 34920066
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Predicting DPP-IV inhibitors with machine learning approaches.
    Cai J; Li C; Liu Z; Du J; Ye J; Gu Q; Xu J
    J Comput Aided Mol Des; 2017 Apr; 31(4):393-402. PubMed ID: 28155089
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Prolyl peptidases related to dipeptidyl peptidase IV: potential of specific inhibitors in drug discovery.
    Van der Veken P; Haemers A; Augustyns K
    Curr Top Med Chem; 2007; 7(6):621-35. PubMed ID: 17352682
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and biological evaluation of novel benzyl-substituted (S)-phenylalanine derivatives as potent dipeptidyl peptidase 4 inhibitors.
    Liu Y; Si M; Tang L; Shangguan S; Wu H; Li J; Wu P; Ma X; Liu T; Hu Y
    Bioorg Med Chem; 2013 Sep; 21(18):5679-87. PubMed ID: 23938053
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Structure based virtual screening of MDPI database: discovery of structurally diverse and novel DPP-IV inhibitors.
    Tanwar O; Tanwar L; Shaquiquzzaman M; Alam MM; Akhter M
    Bioorg Med Chem Lett; 2014 Aug; 24(15):3447-51. PubMed ID: 24948564
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Identification of Potential Dipeptidyl Peptidase (DPP)-IV Inhibitors among
    Yang Y; Shi CY; Xie J; Dai JH; He SL; Tian Y
    Molecules; 2020 Jan; 25(1):. PubMed ID: 31906524
    [No Abstract]   [Full Text] [Related]  

  • 17. Discovery of anthraquinones as DPP-IV inhibitors: Structure-activity relationships and inhibitory mechanism.
    Ma HH; Zhang J; Li CQ; Zou LW
    Fitoterapia; 2023 Jul; 168():105549. PubMed ID: 37244503
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Recent advances in non-peptidomimetic dipeptidyl peptidase 4 inhibitors: medicinal chemistry and preclinical aspects.
    Liu Y; Hu Y; Liu T
    Curr Med Chem; 2012; 19(23):3982-99. PubMed ID: 22709010
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Exploration of DPP-IV inhibitors with a novel scaffold by multistep in silico screening.
    Uchida T; Wakasugi M; Kitamura T; Yamamoto T; Asakura M; Fujiwara R; Itoh T; Fujii H; Hirono S
    J Mol Graph Model; 2018 Jan; 79():254-263. PubMed ID: 29274572
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Discovery of triazole-based uracil derivatives bearing amide moieties as novel dipeptidyl peptidase-IV inhibitors.
    Deng X; Han L; Zhou J; Zhang H; Li Q
    Bioorg Chem; 2017 Dec; 75():357-367. PubMed ID: 29096096
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 11.