These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

32 related articles for article (PubMed ID: 29748052)

  • 1. Evaluation of a Covalent Library of Diverse Warheads (CovLib) Binding to JNK3, USP7, or p53.
    Klett T; Schwer M; Ernst LN; Engelhardt MU; Jaag SJ; Masberg B; Knappe C; Lämmerhofer M; Gehringer M; Boeckler FM
    Drug Des Devel Ther; 2024; 18():2653-2679. PubMed ID: 38974119
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Two key cathepsins, TgCPB and TgCPL, are targeted by the vinyl sulfone inhibitor K11777 in in vitro and in vivo models of toxoplasmosis.
    Chaparro JD; Cheng T; Tran UP; Andrade RM; Brenner SBT; Hwang G; Cohn S; Hirata K; McKerrow JH; Reed SL
    PLoS One; 2018; 13(3):e0193982. PubMed ID: 29565998
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Impact of the Warhead of Dipeptidyl Keto Michael Acceptors on the Inhibition Mechanism of Cysteine Protease Cathepsin L.
    Fernández-de-la-Pradilla A; Royo S; Schirmeister T; Barthels F; Świderek K; González FV; Moliner V
    ACS Catal; 2023 Oct; 13(20):13354-13368. PubMed ID: 37881790
    [TBL] [Abstract][Full Text] [Related]  

  • 4. The vinyl sulfone motif as a structural unit for novel drug design and discovery.
    Xiao YC; Chen FE
    Expert Opin Drug Discov; 2024 Feb; 19(2):239-251. PubMed ID: 37978948
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Julia Olefination as a General Route to Phenyl (alpha-Fluoro)vinyl Sulfones.
    He M; Ghosh AK; Zajc B
    Synlett; 2008 Apr; 2008(7):999-1004. PubMed ID: 19888442
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Targeting the Main Protease of SARS-CoV-2: From the Establishment of High Throughput Screening to the Design of Tailored Inhibitors.
    Breidenbach J; Lemke C; Pillaiyar T; Schäkel L; Al Hamwi G; Diett M; Gedschold R; Geiger N; Lopez V; Mirza S; Namasivayam V; Schiedel AC; Sylvester K; Thimm D; Vielmuth C; Phuong Vu L; Zyulina M; Bodem J; Gütschow M; Müller CE
    Angew Chem Int Ed Engl; 2021 Apr; 60(18):10423-10429. PubMed ID: 33655614
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Synthesis and structure-activity relationship studies of cruzain and rhodesain inhibitors.
    Rocha DA; Silva EB; Fortes IS; Lopes MS; Ferreira RS; Andrade SF
    Eur J Med Chem; 2018 Sep; 157():1426-1459. PubMed ID: 30282318
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Development of nitrile-based peptidic inhibitors of cysteine cathepsins.
    Frizler M; Stirnberg M; Sisay MT; Gütschow M
    Curr Top Med Chem; 2010; 10(3):294-322. PubMed ID: 20166952
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Development of peptidomimetics with a vinyl sulfone warhead as irreversible falcipain-2 inhibitors.
    Ettari R; Nizi E; Di Francesco ME; Dude MA; Pradel G; Vicík R; Schirmeister T; Micale N; Grasso S; Zappalà M
    J Med Chem; 2008 Feb; 51(4):988-96. PubMed ID: 18232656
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs.
    Tber Z; Wartenberg M; Jacques JE; Roy V; Lecaille F; Warszycki D; Bojarski AJ; Lalmanach G; Agrofoglio LA
    Bioorg Med Chem; 2018 Aug; 26(14):4310-4319. PubMed ID: 30049585
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Synthesis and kinetic characterization of hyperbolic inhibitors of human cathepsins K and S based on a succinimide scaffold.
    Goričan T; Ciber L; Petek N; Svete J; Novinec M
    Bioorg Chem; 2021 Oct; 115():105213. PubMed ID: 34364050
    [TBL] [Abstract][Full Text] [Related]  

  • 12. 6-Acylamino-penam derivatives: synthesis and inhibition of cathepsins B, L, K, and S.
    Zhou NE; Kaleta J; Purisima E; Menard R; Micetich RG; Singh R
    Bioorg Med Chem Lett; 2002 Dec; 12(23):3417-9. PubMed ID: 12419374
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Peptidyl allyl sulfones: a new class of inhibitors for clan CA cysteine proteases.
    Götz MG; Caffrey CR; Hansell E; McKerrow JH; Powers JC
    Bioorg Med Chem; 2004 Oct; 12(19):5203-11. PubMed ID: 15351403
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Synthesis and kinetic evaluation of ethyl acrylate and vinyl sulfone derived inhibitors for human cysteine cathepsins.
    Breuer C; Lemke C; Schmitz J; Bartz U; Gütschow M
    Bioorg Med Chem Lett; 2018 Jun; 28(11):2008-2012. PubMed ID: 29748052
    [TBL] [Abstract][Full Text] [Related]  

  • 15.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 16.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 17.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 18.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 19.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

  • 20.
    ; ; . PubMed ID:
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 2.