BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

185 related articles for article (PubMed ID: 29748053)

  • 1. Design, synthesis and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl)transferases PARP10 and PARP14.
    Holechek J; Lease R; Thorsell AG; Karlberg T; McCadden C; Grant R; Keen A; Callahan E; Schüler H; Ferraris D
    Bioorg Med Chem Lett; 2018 Jun; 28(11):2050-2054. PubMed ID: 29748053
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design and synthesis of potent inhibitors of the mono(ADP-ribosyl)transferase, PARP14.
    Upton K; Meyers M; Thorsell AG; Karlberg T; Holechek J; Lease R; Schey G; Wolf E; Lucente A; Schüler H; Ferraris D
    Bioorg Med Chem Lett; 2017 Jul; 27(13):2907-2911. PubMed ID: 28495083
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Analogs of TIQ-A as inhibitors of human mono-ADP-ribosylating PARPs.
    Maksimainen MM; Murthy S; Sowa ST; Galera-Prat A; Rolina E; Heiskanen JP; Lehtiö L
    Bioorg Med Chem; 2021 Dec; 52():116511. PubMed ID: 34801828
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Selective inhibition of PARP10 using a chemical genetics strategy.
    Morgan RK; Carter-O'Connell I; Cohen MS
    Bioorg Med Chem Lett; 2015 Nov; 25(21):4770-4773. PubMed ID: 26231158
    [TBL] [Abstract][Full Text] [Related]  

  • 5. Design, synthesis and evaluation of potential inhibitors for poly(ADP-ribose) polymerase members 1 and 14.
    Kam CM; Tauber AL; Levonis SM; Schweiker SS
    Future Med Chem; 2020 Dec; 12(24):2179-2190. PubMed ID: 33225736
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Structure, Function and Inhibition of Poly(ADP-ribose)polymerase, Member 14 (PARP14).
    Schweiker SS; Tauber AL; Sherry ME; Levonis SM
    Mini Rev Med Chem; 2018; 18(19):1659-1669. PubMed ID: 30112992
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Small Molecule Microarray Based Discovery of PARP14 Inhibitors.
    Peng B; Thorsell AG; Karlberg T; Schüler H; Yao SQ
    Angew Chem Int Ed Engl; 2017 Jan; 56(1):248-253. PubMed ID: 27918638
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2.
    Moustakim M; Riedel K; Schuller M; Gehring AP; Monteiro OP; Martin SP; Fedorov O; Heer J; Dixon DJ; Elkins JM; Knapp S; Bracher F; Brennan PE
    Bioorg Med Chem; 2018 Jul; 26(11):2965-2972. PubMed ID: 29567296
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Activity-based assay for human mono-ADP-ribosyltransferases ARTD7/PARP15 and ARTD10/PARP10 aimed at screening and profiling inhibitors.
    Venkannagari H; Fallarero A; Feijs KL; Lüscher B; Lehtiö L
    Eur J Pharm Sci; 2013 May; 49(2):148-56. PubMed ID: 23485441
    [TBL] [Abstract][Full Text] [Related]  

  • 10.
    Kam CM; Tauber AL; Oosthuizen DL; Levonis SM; Schweiker SS
    Future Med Chem; 2020 Dec; 12(23):2105-2122. PubMed ID: 33225737
    [No Abstract]   [Full Text] [Related]  

  • 11. PARP14 is a PARP with both ADP-ribosyl transferase and hydrolase activities.
    Đukić N; Strømland Ø; Elsborg JD; Munnur D; Zhu K; Schuller M; Chatrin C; Kar P; Duma L; Suyari O; Rack JGM; Baretić D; Crudgington DRK; Groslambert J; Fowler G; Wijngaarden S; Prokhorova E; Rehwinkel J; Schüler H; Filippov DV; Sanyal S; Ahel D; Nielsen ML; Smith R; Ahel I
    Sci Adv; 2023 Sep; 9(37):eadi2687. PubMed ID: 37703374
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Identification of Poly(ADP-Ribose) Polymerase Macrodomain Inhibitors Using an AlphaScreen Protocol.
    Ekblad T; Verheugd P; Lindgren AE; Nyman T; Elofsson M; Schüler H
    SLAS Discov; 2018 Apr; 23(4):353-362. PubMed ID: 29316839
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Towards small molecule inhibitors of mono-ADP-ribosyltransferases.
    Ekblad T; Lindgren AE; Andersson CD; Caraballo R; Thorsell AG; Karlberg T; Spjut S; Linusson A; Schüler H; Elofsson M
    Eur J Med Chem; 2015 May; 95():546-51. PubMed ID: 25847771
    [TBL] [Abstract][Full Text] [Related]  

  • 14. [1,2,4]Triazolo[3,4-
    Murthy S; Nizi MG; Maksimainen MM; Massari S; Alaviuhkola J; Lippok BE; Vagaggini C; Sowa ST; Galera-Prat A; Ashok Y; Venkannagari H; Prunskaite-Hyyryläinen R; Dreassi E; Lüscher B; Korn P; Tabarrini O; Lehtiö L
    J Med Chem; 2023 Jan; 66(2):1301-1320. PubMed ID: 36598465
    [TBL] [Abstract][Full Text] [Related]  

  • 15. 4-(Phenoxy) and 4-(benzyloxy)benzamides as potent and selective inhibitors of mono-ADP-ribosyltransferase PARP10/ARTD10.
    Murthy S; Desantis J; Verheugd P; Maksimainen MM; Venkannagari H; Massari S; Ashok Y; Obaji E; Nkizinkinko Y; Lüscher B; Tabarrini O; Lehtiö L
    Eur J Med Chem; 2018 Aug; 156():93-102. PubMed ID: 30006177
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Mono-ADP-ribosylation by PARP10 and PARP14 in genome stability.
    Dhoonmoon A; Nicolae CM
    NAR Cancer; 2023 Mar; 5(1):zcad009. PubMed ID: 36814782
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Potent 2,3-dihydrophthalazine-1,4-dione derivatives as dual inhibitors for mono-ADP-ribosyltransferases PARP10 and PARP15.
    Nizi MG; Maksimainen MM; Murthy S; Massari S; Alaviuhkola J; Lippok BE; Sowa ST; Galera-Prat A; Prunskaite-Hyyryläinen R; Lüscher B; Korn P; Lehtiö L; Tabarrini O
    Eur J Med Chem; 2022 Jul; 237():114362. PubMed ID: 35500474
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Recent developments in PARP14 research.
    Tauber AL; Levonis SM; Schweiker SS
    Future Med Chem; 2020 Sep; 12(18):1657-1667. PubMed ID: 32893678
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Identification of novel PARP-1 inhibitors: Drug design, synthesis and biological evaluation.
    Xie Z; Zhou Y; Zhao W; Jiao H; Chen Y; Yang Y; Li Z
    Bioorg Med Chem Lett; 2015 Oct; 25(20):4557-61. PubMed ID: 26342868
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Evaluation of 3- and 4-Phenoxybenzamides as Selective Inhibitors of the Mono-ADP-Ribosyltransferase PARP10.
    Korn P; Classen A; Murthy S; Guareschi R; Maksimainen MM; Lippok BE; Galera-Prat A; Sowa ST; Voigt C; Rossetti G; Lehtiö L; Bolm C; Lüscher B
    ChemistryOpen; 2021 Oct; 10(10):939-948. PubMed ID: 34145784
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 10.