182 related articles for article (PubMed ID: 29791525)
1. 2,3,8-Trisubstituted Quinolines with Antimalarial Activity.
Martinez PDG; Krake SH; Poggi ML; Campbell SF; Willis PA; Dias LC
An Acad Bras Cienc; 2018; 90(1 Suppl 2):1215-1231. PubMed ID: 29791525
[TBL] [Abstract][Full Text] [Related]
2. Quinoline hybrids and their antiplasmodial and antimalarial activities.
Hu YQ; Gao C; Zhang S; Xu L; Xu Z; Feng LS; Wu X; Zhao F
Eur J Med Chem; 2017 Oct; 139():22-47. PubMed ID: 28800458
[TBL] [Abstract][Full Text] [Related]
3. New Potential Antimalarial Agents: Design, Synthesis and Biological Evaluation of Some Novel Quinoline Derivatives as Antimalarial Agents.
Radini IA; Elsheikh TM; El-Telbani EM; Khidre RE
Molecules; 2016 Jul; 21(7):. PubMed ID: 27428939
[TBL] [Abstract][Full Text] [Related]
4. Design, Synthesis, Antimalarial Activity and Docking Study of 7-Chloro-4- (2-(substituted benzylidene)hydrazineyl)quinolines.
Kalita J; Chetia D; Rudrapal M
Med Chem; 2020; 16(7):928-937. PubMed ID: 31385774
[TBL] [Abstract][Full Text] [Related]
5. Synthesis and in vitro antiplasmodial activity of ferrocenyl aminoquinoline derivatives.
Mwande Maguene G; Lekana-Douki JB; Mouray E; Bousquet T; Grellier P; Pellegrini S; Toure Ndouo FS; Lebibi J; Pélinski L
Eur J Med Chem; 2015 Jan; 90():519-25. PubMed ID: 25486423
[TBL] [Abstract][Full Text] [Related]
6. New compounds hybrids 1h-1,2,3-triazole-quinoline against Plasmodium falciparum.
Boechat N; Ferreira Mde L; Pinheiro LC; Jesus AM; Leite MM; Júnior CC; Aguiar AC; de Andrade IM; Krettli AU
Chem Biol Drug Des; 2014 Sep; 84(3):325-32. PubMed ID: 24803084
[TBL] [Abstract][Full Text] [Related]
7. Synthesis and in vitro antimalarial testing of neocryptolepines: SAR study for improved activity by introduction and modifications of side chains at C2 and C11 on indolo[2,3-b]quinolines.
Mei ZW; Wang L; Lu WJ; Pang CQ; Maeda T; Peng W; Kaiser M; El Sayed I; Inokuchi T
J Med Chem; 2013 Feb; 56(4):1431-42. PubMed ID: 23360309
[TBL] [Abstract][Full Text] [Related]
8. Evaluation of Antiplasmodial Potential of C2 and C8 Modified Quinolines: in vitro and in silico Study.
Kumar R; Sharma R; Kumar I; Upadhyay P; Dhiman AK; Kumar R; Kumar R; Purohit R; Sahal D; Sharma U
Med Chem; 2019; 15(7):790-800. PubMed ID: 30324888
[TBL] [Abstract][Full Text] [Related]
9. Synthesis and antimalarial testing of neocryptolepine analogues: addition of ester function in SAR study of 2,11-disubstituted indolo[2,3-b]quinolines.
Lu WJ; Wicht KJ; Wang L; Imai K; Mei ZW; Kaiser M; El Sayed Iel T; Egan TJ; Inokuchi T
Eur J Med Chem; 2013 Jun; 64():498-511. PubMed ID: 23685569
[TBL] [Abstract][Full Text] [Related]
10. Design, synthesis and biological evaluation of mono- and bisquinoline methanamine derivatives as potential antiplasmodial agents.
Bokosi FRB; Beteck RM; Mbaba M; Mtshare TE; Laming D; Hoppe HC; Khanye SD
Bioorg Med Chem Lett; 2021 Apr; 38():127855. PubMed ID: 33609655
[TBL] [Abstract][Full Text] [Related]
11. Design and synthesis of novel ferrocene-quinoline conjugates and evaluation of their electrochemical and antiplasmodium properties.
Minić A; Van de Walle T; Van Hecke K; Combrinck J; Smith PJ; Chibale K; D'hooghe M
Eur J Med Chem; 2020 Feb; 187():111963. PubMed ID: 31865015
[TBL] [Abstract][Full Text] [Related]
12. Discovery of a Quinoline-4-carboxamide Derivative with a Novel Mechanism of Action, Multistage Antimalarial Activity, and Potent in Vivo Efficacy.
Baragaña B; Norcross NR; Wilson C; Porzelle A; Hallyburton I; Grimaldi R; Osuna-Cabello M; Norval S; Riley J; Stojanovski L; Simeons FR; Wyatt PG; Delves MJ; Meister S; Duffy S; Avery VM; Winzeler EA; Sinden RE; Wittlin S; Frearson JA; Gray DW; Fairlamb AH; Waterson D; Campbell SF; Willis P; Read KD; Gilbert IH
J Med Chem; 2016 Nov; 59(21):9672-9685. PubMed ID: 27631715
[TBL] [Abstract][Full Text] [Related]
13. New quinoline derivatives demonstrate a promising antimalarial activity against Plasmodium falciparum in vitro and Plasmodium berghei in vivo.
Soares RR; da Silva JM; Carlos BC; da Fonseca CC; de Souza LS; Lopes FV; de Paula Dias RM; Moreira PO; Abramo C; Viana GH; de Pila Varotti F; da Silva AD; Scopel KK
Bioorg Med Chem Lett; 2015 Jun; 25(11):2308-13. PubMed ID: 25920564
[TBL] [Abstract][Full Text] [Related]
14. Quinoline Containing Side-chain Antimalarial Analogs: Recent Advances and Therapeutic Application.
Joshi MC; Egan TJ
Curr Top Med Chem; 2020; 20(8):617-697. PubMed ID: 31985377
[TBL] [Abstract][Full Text] [Related]
15. Novel Quinolinyl-pyrrolo[3,4-d]pyrimidine-2,5-dione Derivatives Against Chloroquine-resistant Plasmodium falciparum.
Rogerio KR; Graebin CS; Pinto Domingues LH; Oliveira LS; de Souza Fernandes da Silva V; Daniel-Ribeiro CT; Carvalho LJM; Boechat N
Curr Top Med Chem; 2020; 20(2):99-110. PubMed ID: 31648638
[TBL] [Abstract][Full Text] [Related]
16. Synthesis and antimalarial evaluation of novel isocryptolepine derivatives.
Whittell LR; Batty KT; Wong RP; Bolitho EM; Fox SA; Davis TM; Murray PE
Bioorg Med Chem; 2011 Dec; 19(24):7519-25. PubMed ID: 22055713
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and biological evaluation of novel quinoline-piperidine scaffolds as antiplasmodium agents.
Van de Walle T; Boone M; Van Puyvelde J; Combrinck J; Smith PJ; Chibale K; Mangelinckx S; D'hooghe M
Eur J Med Chem; 2020 Jul; 198():112330. PubMed ID: 32408064
[TBL] [Abstract][Full Text] [Related]
18. Discovery of Marinoquinolines as Potent and Fast-Acting Plasmodium falciparum Inhibitors with in Vivo Activity.
Aguiar ACC; Panciera M; Simão Dos Santos EF; Singh MK; Garcia ML; de Souza GE; Nakabashi M; Costa JL; Garcia CRS; Oliva G; Correia CRD; Guido RVC
J Med Chem; 2018 Jul; 61(13):5547-5568. PubMed ID: 29879353
[TBL] [Abstract][Full Text] [Related]
19. New derivatives of quinoline-4-carboxylic acid with antiplasmodial activity.
Hochegger P; Faist J; Seebacher W; Saf R; Mäser P; Kaiser M; Weis R
Bioorg Med Chem; 2017 Apr; 25(7):2251-2259. PubMed ID: 28279559
[TBL] [Abstract][Full Text] [Related]
20. Quinoline carboxamide core moiety-based compounds inhibit P. falciparumfalcipain-2: Design, synthesis and antimalarial efficacy studies.
Singh A; Kalamuddin M; Maqbool M; Mohmmed A; Malhotra P; Hoda N
Bioorg Chem; 2021 Mar; 108():104514. PubMed ID: 33280833
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]