168 related articles for article (PubMed ID: 29869845)
21. Small-molecule modulators for epigenetics targets.
Knapp S; Weinmann H
ChemMedChem; 2013 Nov; 8(11):1885-91. PubMed ID: 24127276
[TBL] [Abstract][Full Text] [Related]
22. Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.
Milite C; Feoli A; Viviano M; Rescigno D; Mai A; Castellano S; Sbardella G
ChemMedChem; 2016 Aug; 11(16):1680-5. PubMed ID: 27411844
[TBL] [Abstract][Full Text] [Related]
23. [Research Progress of Role and Mechanism of SETD7 in Tumor Occurrence
and Progression].
Cao L; Wang M; Xu K
Zhongguo Fei Ai Za Zhi; 2023 Jan; 26(1):38-45. PubMed ID: 36792079
[TBL] [Abstract][Full Text] [Related]
24. Substrate docking-mediated specific and efficient lysine methylation by the SET domain-containing histone methyltransferase SETD7.
Liu H; Li Z; Yang Q; Liu W; Wan J; Li J; Zhang M
J Biol Chem; 2019 Sep; 294(36):13355-13365. PubMed ID: 31324717
[TBL] [Abstract][Full Text] [Related]
25. Discovery of a selective, substrate-competitive inhibitor of the lysine methyltransferase SETD8.
Ma A; Yu W; Li F; Bleich RM; Herold JM; Butler KV; Norris JL; Korboukh V; Tripathy A; Janzen WP; Arrowsmith CH; Frye SV; Vedadi M; Brown PJ; Jin J
J Med Chem; 2014 Aug; 57(15):6822-33. PubMed ID: 25032507
[TBL] [Abstract][Full Text] [Related]
26. Development of novel bisubstrate-type inhibitors of histone methyltransferase SET7/9.
Mori S; Iwase K; Iwanami N; Tanaka Y; Kagechika H; Hirano T
Bioorg Med Chem; 2010 Dec; 18(23):8158-66. PubMed ID: 21036620
[TBL] [Abstract][Full Text] [Related]
27. Amide-derived lysine analogues as substrates and inhibitors of histone lysine methyltransferases and acetyltransferases.
Hintzen JCJ; Merx J; Maas MN; Langens SGHA; White PB; Boltje TJ; Mecinović J
Org Biomol Chem; 2021 Dec; 20(1):173-181. PubMed ID: 34877957
[TBL] [Abstract][Full Text] [Related]
28. Inhibitors of enzymes catalyzing modifications to histone lysine residues: structure, function and activity.
Lillico R; Stesco N; Khorshid Amhad T; Cortes C; Namaka MP; Lakowski TM
Future Med Chem; 2016 May; 8(8):879-97. PubMed ID: 27173004
[TBL] [Abstract][Full Text] [Related]
29. Identification and Characterizations of Novel, Selective Histone Methyltransferase SET7 Inhibitors by Scaffold Hopping- and 2D-Molecular Fingerprint-Based Similarity Search.
Ding H; Lu WC; Hu JC; Liu YC; Zhang CH; Lian FL; Zhang NX; Meng FW; Luo C; Chen KX
Molecules; 2018 Mar; 23(3):. PubMed ID: 29498708
[TBL] [Abstract][Full Text] [Related]
30. Methylation of the Hippo effector YAP by the methyltransferase SETD7 drives myocardial ischaemic injury: a translational study.
Ambrosini S; Montecucco F; Kolijn D; Pedicino D; Akhmedov A; Mohammed SA; Herwig M; Gorica E; Szabó PL; Weber L; Russo G; Vinci R; Matter CM; Liuzzo G; Brown PJ; Rossi FMV; Camici GG; Sciarretta S; Beltrami AP; Crea F; Podesser B; Lüscher TF; Kiss A; Ruschitzka F; Hamdani N; Costantino S; Paneni F
Cardiovasc Res; 2023 Jan; 118(17):3374-3385. PubMed ID: 35709329
[TBL] [Abstract][Full Text] [Related]
31. Transcriptomic Analysis of Histone Methyltransferase Setd7 Knockdown and Phenethyl Isothiocyanate in Human Prostate Cancer Cells.
Wang C; Sargsyan D; Zhang C; Wu R; Yang Y; Kong AN
Anticancer Res; 2018 Nov; 38(11):6069-6083. PubMed ID: 30396921
[TBL] [Abstract][Full Text] [Related]
32. Synthesis and characterization of the first inhibitor of N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD).
Castellani B; Diamanti E; Pizzirani D; Tardia P; Maccesi M; Realini N; Magotti P; Garau G; Bakkum T; Rivara S; Mor M; Piomelli D
Chem Commun (Camb); 2017 Nov; 53(95):12814-12817. PubMed ID: 29143042
[TBL] [Abstract][Full Text] [Related]
33. [Histone lysine methyltransferase Setd7 enhances Ngn 1 gene expression].
Dai JP; Zhang Y; Shen YF
Zhongguo Yi Xue Ke Xue Yuan Xue Bao; 2009 Dec; 31(6):692-5. PubMed ID: 20078936
[TBL] [Abstract][Full Text] [Related]
34. Development of homogeneous nonradioactive methyltransferase and demethylase assays targeting histone H3 lysine 4.
Gauthier N; Caron M; Pedro L; Arcand M; Blouin J; Labonté A; Normand C; Paquet V; Rodenbrock A; Roy M; Rouleau N; Beaudet L; Padrós J; Rodriguez-Suarez R
J Biomol Screen; 2012 Jan; 17(1):49-58. PubMed ID: 21940714
[TBL] [Abstract][Full Text] [Related]
35. The role of SET domain containing lysine methyltransferase 7 in tumorigenesis and development.
Yang S; Wang X; Bai J; Duan B
Cell Cycle; 2023 Feb; 22(3):269-275. PubMed ID: 36101480
[TBL] [Abstract][Full Text] [Related]
36. Biological evaluation of tanshindiols as EZH2 histone methyltransferase inhibitors.
Woo J; Kim HY; Byun BJ; Chae CH; Lee JY; Ryu SY; Park WK; Cho H; Choi G
Bioorg Med Chem Lett; 2014 Jun; 24(11):2486-92. PubMed ID: 24767850
[TBL] [Abstract][Full Text] [Related]
37. Inhibitors of phenylethanolamine N-methyltransferase devoid of alpha2-adrenoceptor affinity.
Grunewald GL; Lu J; Criscione KR; Okoro CO
Bioorg Med Chem Lett; 2005 Dec; 15(23):5319-23. PubMed ID: 16169723
[TBL] [Abstract][Full Text] [Related]
38. LLY-507, a Cell-active, Potent, and Selective Inhibitor of Protein-lysine Methyltransferase SMYD2.
Nguyen H; Allali-Hassani A; Antonysamy S; Chang S; Chen LH; Curtis C; Emtage S; Fan L; Gheyi T; Li F; Liu S; Martin JR; Mendel D; Olsen JB; Pelletier L; Shatseva T; Wu S; Zhang FF; Arrowsmith CH; Brown PJ; Campbell RM; Garcia BA; Barsyte-Lovejoy D; Mader M; Vedadi M
J Biol Chem; 2015 May; 290(22):13641-53. PubMed ID: 25825497
[TBL] [Abstract][Full Text] [Related]
39. Design of a fluorescent ligand targeting the S-adenosylmethionine binding site of the histone methyltransferase MLL1.
Luan Y; Blazer LL; Hu H; Hajian T; Zhang J; Wu H; Houliston S; Arrowsmith CH; Vedadi M; Zheng YG
Org Biomol Chem; 2016 Jan; 14(2):631-638. PubMed ID: 26541578
[TBL] [Abstract][Full Text] [Related]
40. On the histone lysine methyltransferase activity of fungal metabolite chaetocin.
Cherblanc FL; Chapman KL; Reid J; Borg AJ; Sundriyal S; Alcazar-Fuoli L; Bignell E; Demetriades M; Schofield CJ; DiMaggio PA; Brown R; Fuchter MJ
J Med Chem; 2013 Nov; 56(21):8616-25. PubMed ID: 24099080
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]
