These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.
101 related articles for article (PubMed ID: 29901392)
1. Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist. De Marco R; Bedini A; Spampinato S; Comellini L; Zhao J; Artali R; Gentilucci L J Med Chem; 2018 Jul; 61(13):5751-5757. PubMed ID: 29901392 [TBL] [Abstract][Full Text] [Related]
2. Redoubling the ring size of an endomorphin-2 analog transforms a centrally acting mu-opioid receptor agonist into a pure peripheral analgesic. Piekielna J; De Marco R; Gentilucci L; Cerlesi MC; Calo' G; Tömböly C; Artali R; Janecka A Biopolymers; 2016 May; 106(3):309-17. PubMed ID: 27038094 [TBL] [Abstract][Full Text] [Related]
3. Antinociceptive and antidepressant-like action of endomorphin-2 analogs with proline surrogates in position 2. Perlikowska R; Piekielna J; Mazur M; Koralewski R; Olczak J; do Rego JC; Fichna J; Modranka J; Janecki T; Janecka A Bioorg Med Chem; 2014 Sep; 22(17):4803-9. PubMed ID: 25047937 [TBL] [Abstract][Full Text] [Related]
4. A new class of highly potent and selective endomorphin-1 analogues containing α-methylene-β-aminopropanoic acids (map). Wang Y; Xing Y; Liu X; Ji H; Kai M; Chen Z; Yu J; Zhao D; Ren H; Wang R J Med Chem; 2012 Jul; 55(13):6224-36. PubMed ID: 22724433 [TBL] [Abstract][Full Text] [Related]
5. Design, synthesis, and pharmacological characterization of novel endomorphin-1 analogues as extremely potent μ-opioid agonists. Liu X; Wang Y; Xing Y; Yu J; Ji H; Kai M; Wang Z; Wang D; Zhang Y; Zhao D; Wang R J Med Chem; 2013 Apr; 56(7):3102-14. PubMed ID: 23477419 [TBL] [Abstract][Full Text] [Related]
6. Synthesis of tripeptides containing D-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception. De Marco R; Bedini A; Spampinato S; Gentilucci L J Med Chem; 2014 Aug; 57(15):6861-6. PubMed ID: 25051243 [TBL] [Abstract][Full Text] [Related]
7. Synthesis of mixed MOR/KOR efficacy cyclic opioid peptide analogs with antinociceptive activity after systemic administration. Perlikowska R; Piekielna J; Gentilucci L; De Marco R; Cerlesi MC; Calo G; Artali R; Tömböly C; Kluczyk A; Janecka A Eur J Med Chem; 2016 Feb; 109():276-86. PubMed ID: 26785295 [TBL] [Abstract][Full Text] [Related]
8. The inverse type II β-turn on D-Trp-Phe, a pharmacophoric motif for MOR agonists. Gentilucci L; Tolomelli A; De Marco R; Spampinato S; Bedini A; Artali R ChemMedChem; 2011 Sep; 6(9):1640-53. PubMed ID: 21721130 [TBL] [Abstract][Full Text] [Related]
9. Development of potent bifunctional endomorphin-2 analogues with mixed mu-/delta-opioid agonist and delta-opioid antagonist properties. Fujita Y; Tsuda Y; Li T; Motoyama T; Takahashi M; Shimizu Y; Yokoi T; Sasaki Y; Ambo A; Kita A; Jinsmaa Y; Bryant SD; Lazarus LH; Okada Y J Med Chem; 2004 Jul; 47(14):3591-9. PubMed ID: 15214786 [TBL] [Abstract][Full Text] [Related]
10. Endomorphin 1[psi] and endomorphin 2[psi], endomorphins analogues containing a reduced (CH2NH) amide bond between Tyr1 and Pro2, display partial agonist potency but significant antinociception. Zhao QY; Chen Q; Yang DJ; Feng Y; Long Y; Wang P; Wang R Life Sci; 2005 Jul; 77(10):1155-65. PubMed ID: 15878600 [TBL] [Abstract][Full Text] [Related]
11. The Pharmacological Heterogeneity of Nepenthone Analogs in Conferring Highly Selective and Potent κ-Opioid Agonistic Activities. Li W; Long JD; Qian YY; Long Y; Xu XJ; Wang YJ; Shen Q; Wang ZN; Yang XC; Xiao L; Sun HP; Xu YL; Chen YY; Xie Q; Wang YH; Shao LM; Liu JG; Qiu ZB; Fu W ACS Chem Neurosci; 2017 Apr; 8(4):766-776. PubMed ID: 28033462 [TBL] [Abstract][Full Text] [Related]
12. Synthesis and biological evaluations of novel endomorphin analogues containing α-hydroxy-β-phenylalanine (AHPBA) displaying mixed μ/δ opioid receptor agonist and δ opioid receptor antagonist activities. Hu M; Giulianotti MA; McLaughlin JP; Shao J; Debevec G; Maida LE; Geer P; Cazares M; Misler J; Li L; Dooley C; Ganno ML; Eans SO; Mizrachi E; Santos RG; Yongye AB; Houghten RA; Yu Y Eur J Med Chem; 2015 Mar; 92():270-81. PubMed ID: 25559207 [TBL] [Abstract][Full Text] [Related]
13. Design, synthesis, and evaluation of new endomorphin analogs with enhanced central antinociception after peripheral administration. Liu X; Zhao L; Wang Y; Mou L; Yang J; Zhang Y; Wang D; Wang R Bioorg Med Chem Lett; 2015 Nov; 25(22):5393-7. PubMed ID: 26403932 [TBL] [Abstract][Full Text] [Related]
14. Synthesis and characterization of potent and selective mu-opioid receptor antagonists, [Dmt(1), D-2-Nal(4)]endomorphin-1 (Antanal-1) and [Dmt(1), D-2-Nal(4)]endomorphin-2 (Antanal-2). Fichna J; do-Rego JC; Chung NN; Lemieux C; Schiller PW; Poels J; Broeck JV; Costentin J; Janecka A J Med Chem; 2007 Feb; 50(3):512-20. PubMed ID: 17266203 [TBL] [Abstract][Full Text] [Related]
15. Highly Potent and Selective New Diphenethylamines Interacting with the κ-Opioid Receptor: Synthesis, Pharmacology, and Structure-Activity Relationships. Erli F; Guerrieri E; Ben Haddou T; Lantero A; Mairegger M; Schmidhammer H; Spetea M J Med Chem; 2017 Sep; 60(17):7579-7590. PubMed ID: 28825813 [TBL] [Abstract][Full Text] [Related]
16. Pharmacological characterization of EN-9, a novel chimeric peptide of endomorphin-2 and neuropeptide FF that produces potent antinociceptive activity and limited tolerance. Wang ZL; Li N; Wang P; Tang HH; Han ZL; Song JJ; Li XH; Yu HP; Zhang T; Zhang R; Xu B; Zhang MN; Fang Q; Wang R Neuropharmacology; 2016 Sep; 108():364-72. PubMed ID: 26970017 [TBL] [Abstract][Full Text] [Related]
17. Selective MOR activity of DAPEA and Endomorphin-2 analogues containing a (R)-γ-Freidinger lactam in position two. Della Valle A; Stefanucci A; Scioli G; Szűcs E; Benyhe S; Pieretti S; Minosi P; Sturaro C; Calò G; Zengin G; Mollica A Bioorg Chem; 2021 Oct; 115():105219. PubMed ID: 34343741 [TBL] [Abstract][Full Text] [Related]
18. Synthesis of 6,14-epoxymorphinan derivatives and their pharmacologies. Nemoto T; Yamamoto N; Watanabe A; Fujii H; Hasebe K; Nakajima M; Mochizuki H; Nagase H Bioorg Med Chem; 2011 Feb; 19(3):1205-21. PubMed ID: 21256034 [TBL] [Abstract][Full Text] [Related]
19. Biological activity of endomorphin and [Dmt1]endomorphin analogs with six-membered proline surrogates in position 2. Perlikowska R; Gach K; Fichna J; Toth G; Walkowiak B; do-Rego JC; Janecka A Bioorg Med Chem; 2009 Jun; 17(11):3789-94. PubMed ID: 19435668 [TBL] [Abstract][Full Text] [Related]
20. Synthesis and Assessment of Fused β-Carboline Derivatives as Kappa Opioid Receptor Agonists. Yadav VD; Kumar L; Kumari P; Kumar S; Singh M; Siddiqi MI; Yadav PN; Batra S ChemMedChem; 2021 Jun; 16(12):1917-1926. PubMed ID: 33599108 [TBL] [Abstract][Full Text] [Related] [Next] [New Search]