101 related articles for article (PubMed ID: 30004552)
1. Two-step activity-based protein profiling of diacylglycerol lipase.
van Rooden EJ; Kreekel R; Hansen T; Janssen APA; van Esbroeck ACM; den Dulk H; van den Berg RJBHN; Codée JDC; van der Stelt M
Org Biomol Chem; 2018 Jul; 16(29):5250-5253. PubMed ID: 30004552
[TBL] [Abstract][Full Text] [Related]
2. Design and Synthesis of Quenched Activity-based Probes for Diacylglycerol Lipase and α,β-Hydrolase Domain Containing Protein 6.
van Rooden EJ; Kohsiek M; Kreekel R; van Esbroeck ACM; van den Nieuwendijk AMCH; Janssen APA; van den Berg RJBHN; Overkleeft HS; van der Stelt M
Chem Asian J; 2018 Nov; 13(22):3491-3500. PubMed ID: 29901868
[TBL] [Abstract][Full Text] [Related]
3. Development and optimization of piperidyl-1,2,3-triazole ureas as selective chemical probes of endocannabinoid biosynthesis.
Hsu KL; Tsuboi K; Whitby LR; Speers AE; Pugh H; Inloes J; Cravatt BF
J Med Chem; 2013 Nov; 56(21):8257-69. PubMed ID: 24152245
[TBL] [Abstract][Full Text] [Related]
4. Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition.
Ogasawara D; Deng H; Viader A; Baggelaar MP; Breman A; den Dulk H; van den Nieuwendijk AM; Soethoudt M; van der Wel T; Zhou J; Overkleeft HS; Sanchez-Alavez M; Mori S; Nguyen W; Conti B; Liu X; Chen Y; Liu QS; Cravatt BF; van der Stelt M
Proc Natl Acad Sci U S A; 2016 Jan; 113(1):26-33. PubMed ID: 26668358
[TBL] [Abstract][Full Text] [Related]
5. Triazole Ureas Act as Diacylglycerol Lipase Inhibitors and Prevent Fasting-Induced Refeeding.
Deng H; Kooijman S; van den Nieuwendijk AM; Ogasawara D; van der Wel T; van Dalen F; Baggelaar MP; Janssen FJ; van den Berg RJ; den Dulk H; Cravatt BF; Overkleeft HS; Rensen PC; van der Stelt M
J Med Chem; 2017 Jan; 60(1):428-440. PubMed ID: 27992221
[TBL] [Abstract][Full Text] [Related]
6. Chemical tools to modulate 2-arachidonoylglycerol biosynthesis.
Deng H; van der Stelt M
Biotechnol Appl Biochem; 2018 Jan; 65(1):9-15. PubMed ID: 28589628
[TBL] [Abstract][Full Text] [Related]
7. Inhibition of diacylglycerol lipase β modulates lipid and endocannabinoid levels in the
Berger N; van der Wel T; Hirschmugl B; Baernthaler T; Gindlhuber J; Fawzy N; Eichmann T; Birner-Gruenberger R; Zimmermann R; van der Stelt M; Wadsack C
Front Endocrinol (Lausanne); 2023; 14():1092024. PubMed ID: 36864832
[TBL] [Abstract][Full Text] [Related]
8. Brain regional cannabinoid CB(1) receptor signalling and alternative enzymatic pathways for 2-arachidonoylglycerol generation in brain sections of diacylglycerol lipase deficient mice.
Aaltonen N; Riera Ribas C; Lehtonen M; Savinainen JR; Laitinen JT
Eur J Pharm Sci; 2014 Jan; 51():87-95. PubMed ID: 24012970
[TBL] [Abstract][Full Text] [Related]
9. Inhibiting endocannabinoid biosynthesis: a novel approach to the treatment of constipation.
Bashashati M; Nasser Y; Keenan CM; Ho W; Piscitelli F; Nalli M; Mackie K; Storr MA; Di Marzo V; Sharkey KA
Br J Pharmacol; 2015 Jun; 172(12):3099-111. PubMed ID: 25684407
[TBL] [Abstract][Full Text] [Related]
10. Enzymatic characterization of recombinant rat DDHD2: a soluble diacylglycerol lipase.
Araki M; Ohshima N; Aso C; Konishi A; Obinata H; Tatei K; Izumi T
J Biochem; 2016 Nov; 160(5):269-279. PubMed ID: 27198176
[TBL] [Abstract][Full Text] [Related]
11. Liposomal Delivery of Diacylglycerol Lipase-Beta Inhibitors to Macrophages Dramatically Enhances Selectivity and Efficacy in Vivo.
Shin M; Snyder HW; Donvito G; Schurman LD; Fox TE; Lichtman AH; Kester M; Hsu KL
Mol Pharm; 2018 Mar; 15(3):721-728. PubMed ID: 28901776
[TBL] [Abstract][Full Text] [Related]
12. A novel live cell assay to measure diacylglycerol lipase α activity.
Singh PK; Markwick R; Howell FV; Williams G; Doherty P
Biosci Rep; 2016 Jun; 36(3):. PubMed ID: 27013337
[TBL] [Abstract][Full Text] [Related]
13. DAGLβ inhibition perturbs a lipid network involved in macrophage inflammatory responses.
Hsu KL; Tsuboi K; Adibekian A; Pugh H; Masuda K; Cravatt BF
Nat Chem Biol; 2012 Dec; 8(12):999-1007. PubMed ID: 23103940
[TBL] [Abstract][Full Text] [Related]
14. Highly Selective, Reversible Inhibitor Identified by Comparative Chemoproteomics Modulates Diacylglycerol Lipase Activity in Neurons.
Baggelaar MP; Chameau PJ; Kantae V; Hummel J; Hsu KL; Janssen F; van der Wel T; Soethoudt M; Deng H; den Dulk H; Allarà M; Florea BI; Di Marzo V; Wadman WJ; Kruse CG; Overkleeft HS; Hankemeier T; Werkman TR; Cravatt BF; van der Stelt M
J Am Chem Soc; 2015 Jul; 137(27):8851-7. PubMed ID: 26083464
[TBL] [Abstract][Full Text] [Related]
15. Assay and Inhibition of the Purified Catalytic Domain of Diacylglycerol Lipase Beta.
Singh PK; Markwick R; Lu L; Howell FV; Williams G; Doherty P
Biochemistry; 2016 May; 55(19):2713-21. PubMed ID: 27115711
[TBL] [Abstract][Full Text] [Related]
16. Competitive ABPP of Serine Hydrolases: A Case Study on DAGL-Alpha.
Baggelaar MP; Van der Stelt M
Methods Mol Biol; 2017; 1491():161-169. PubMed ID: 27778288
[TBL] [Abstract][Full Text] [Related]
17. Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain.
Baggelaar MP; Janssen FJ; van Esbroeck AC; den Dulk H; Allarà M; Hoogendoorn S; McGuire R; Florea BI; Meeuwenoord N; van den Elst H; van der Marel GA; Brouwer J; Di Marzo V; Overkleeft HS; van der Stelt M
Angew Chem Int Ed Engl; 2013 Nov; 52(46):12081-5. PubMed ID: 24173880
[No Abstract] [Full Text] [Related]
18. DAGL-Beta Functions as a PUFA-Specific Triacylglycerol Lipase in Macrophages.
Shin M; Ware TB; Hsu KL
Cell Chem Biol; 2020 Mar; 27(3):314-321.e5. PubMed ID: 31991095
[TBL] [Abstract][Full Text] [Related]
19. Discovery of glycine sulfonamides as dual inhibitors of sn-1-diacylglycerol lipase α and α/β-hydrolase domain 6.
Janssen FJ; Deng H; Baggelaar MP; Allarà M; van der Wel T; den Dulk H; Ligresti A; van Esbroeck AC; McGuire R; Di Marzo V; Overkleeft HS; van der Stelt M
J Med Chem; 2014 Aug; 57(15):6610-22. PubMed ID: 24988361
[TBL] [Abstract][Full Text] [Related]
20.
; ; . PubMed ID:
[No Abstract] [Full Text] [Related]
[Next] [New Search]