334 related articles for article (PubMed ID: 30009876)
1. Reengineering the ligand sensitivity of the broadly tuned human bitter taste receptor TAS2R14.
Nowak S; Di Pizio A; Levit A; Niv MY; Meyerhof W; Behrens M
Biochim Biophys Acta Gen Subj; 2018 Oct; 1862(10):2162-2173. PubMed ID: 30009876
[TBL] [Abstract][Full Text] [Related]
2. Probing the Binding Pocket of the Broadly Tuned Human Bitter Taste Receptor TAS2R14 by Chemical Modification of Cognate Agonists.
Karaman R; Nowak S; Di Pizio A; Kitaneh H; Abu-Jaish A; Meyerhof W; Niv MY; Behrens M
Chem Biol Drug Des; 2016 Jul; 88(1):66-75. PubMed ID: 26825540
[TBL] [Abstract][Full Text] [Related]
3. Rational design of agonists for bitter taste receptor TAS2R14: from modeling to bench and back.
Di Pizio A; Waterloo LAW; Brox R; Löber S; Weikert D; Behrens M; Gmeiner P; Niv MY
Cell Mol Life Sci; 2020 Feb; 77(3):531-542. PubMed ID: 31236627
[TBL] [Abstract][Full Text] [Related]
4. The bitter pill: clinical drugs that activate the human bitter taste receptor TAS2R14.
Levit A; Nowak S; Peters M; Wiener A; Meyerhof W; Behrens M; Niv MY
FASEB J; 2014 Mar; 28(3):1181-97. PubMed ID: 24285091
[TBL] [Abstract][Full Text] [Related]
5. Plasticity of the ligand binding pocket in the bitter taste receptor T2R7.
Liu K; Jaggupilli A; Premnath D; Chelikani P
Biochim Biophys Acta Biomembr; 2018 May; 1860(5):991-999. PubMed ID: 29355483
[TBL] [Abstract][Full Text] [Related]
6. Structural requirements of bitter taste receptor activation.
Brockhoff A; Behrens M; Niv MY; Meyerhof W
Proc Natl Acad Sci U S A; 2010 Jun; 107(24):11110-5. PubMed ID: 20534469
[TBL] [Abstract][Full Text] [Related]
7. The human bitter taste receptor TAS2R10 is tailored to accommodate numerous diverse ligands.
Born S; Levit A; Niv MY; Meyerhof W; Behrens M
J Neurosci; 2013 Jan; 33(1):201-13. PubMed ID: 23283334
[TBL] [Abstract][Full Text] [Related]
8. Bitter taste receptor activation by cholesterol and an intracellular tastant.
Kim Y; Gumpper RH; Liu Y; Kocak DD; Xiong Y; Cao C; Deng Z; Krumm BE; Jain MK; Zhang S; Jin J; Roth BL
Nature; 2024 Apr; 628(8008):664-671. PubMed ID: 38600377
[TBL] [Abstract][Full Text] [Related]
9. The Odorant ( R)-Citronellal Attenuates Caffeine Bitterness by Inhibiting the Bitter Receptors TAS2R43 and TAS2R46.
Suess B; Brockhoff A; Meyerhof W; Hofmann T
J Agric Food Chem; 2018 Mar; 66(10):2301-2311. PubMed ID: 27569025
[TBL] [Abstract][Full Text] [Related]
10. Bitter substances from plants used in traditional Chinese medicine exert biased activation of human bitter taste receptors.
Behrens M; Gu M; Fan S; Huang C; Meyerhof W
Chem Biol Drug Des; 2018 Feb; 91(2):422-433. PubMed ID: 28834122
[TBL] [Abstract][Full Text] [Related]
11. Inhibiting a promiscuous GPCR: iterative discovery of bitter taste receptor ligands.
Fierro F; Peri L; Hübner H; Tabor-Schkade A; Waterloo L; Löber S; Pfeiffer T; Weikert D; Dingjan T; Margulis E; Gmeiner P; Niv MY
Cell Mol Life Sci; 2023 Apr; 80(4):114. PubMed ID: 37012410
[TBL] [Abstract][Full Text] [Related]
12. The Bitter Taste Receptor TAS2R14 as a Drug Target.
Waterloo LAW; Löber S; Gmeiner P
Chimia (Aarau); 2022 May; 76(5):418-424. PubMed ID: 38069713
[TBL] [Abstract][Full Text] [Related]
13. Ligand binding modes from low resolution GPCR models and mutagenesis: chicken bitter taste receptor as a test-case.
Di Pizio A; Kruetzfeldt LM; Cheled-Shoval S; Meyerhof W; Behrens M; Niv MY
Sci Rep; 2017 Aug; 7(1):8223. PubMed ID: 28811548
[TBL] [Abstract][Full Text] [Related]
14. Amino acid derivatives as bitter taste receptor (T2R) blockers.
Pydi SP; Sobotkiewicz T; Billakanti R; Bhullar RP; Loewen MC; Chelikani P
J Biol Chem; 2014 Sep; 289(36):25054-66. PubMed ID: 25059668
[TBL] [Abstract][Full Text] [Related]
15. Numerous Compounds Orchestrate Coffee's Bitterness.
Lang T; Lang R; Di Pizio A; Mittermeier VK; Schlagbauer V; Hofmann T; Behrens M
J Agric Food Chem; 2020 Jun; 68(24):6692-6700. PubMed ID: 32437139
[TBL] [Abstract][Full Text] [Related]
16. Highly conserved intracellular H208 residue influences agonist selectivity in bitter taste receptor T2R14.
Shaik FA; Jaggupilli A; Chelikani P
Biochim Biophys Acta Biomembr; 2019 Dec; 1861(12):183057. PubMed ID: 31493373
[TBL] [Abstract][Full Text] [Related]
17. Abscisic Acid Acts as a Blocker of the Bitter Taste G Protein-Coupled Receptor T2R4.
Pydi SP; Jaggupilli A; Nelson KM; Abrams SR; Bhullar RP; Loewen MC; Chelikani P
Biochemistry; 2015 Apr; 54(16):2622-31. PubMed ID: 25844797
[TBL] [Abstract][Full Text] [Related]
18. β2-Adrenergic Receptors Chaperone Trapped Bitter Taste Receptor 14 to the Cell Surface as a Heterodimer and Exert Unidirectional Desensitization of Taste Receptor Function.
Kim D; Pauer SH; Yong HM; An SS; Liggett SB
J Biol Chem; 2016 Aug; 291(34):17616-28. PubMed ID: 27342779
[TBL] [Abstract][Full Text] [Related]
19. The short third intracellular loop and cytoplasmic tail of bitter taste receptors provide functionally relevant GRK phosphorylation sites in TAS2R14.
Kim D; Castaño M; Lujan LK; Woo JA; Liggett SB
J Biol Chem; 2021; 296():100216. PubMed ID: 33465377
[TBL] [Abstract][Full Text] [Related]
20. Bitter taste TAS2R14 activation by intracellular tastants and cholesterol.
Hu X; Ao W; Gao M; Wu L; Pei Y; Liu S; Wu Y; Zhao F; Sun Q; Liu J; Jiang L; Wang X; Li Y; Tan Q; Cheng J; Yang F; Yang C; Sun J; Hua T; Liu ZJ
Nature; 2024 May; ():. PubMed ID: 38776963
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]
