These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

113 related articles for article (PubMed ID: 3005567)

  • 1. Glycine antagonists. Synthesis, structure, and biological effects of some bicyclic 5-isoxazolol zwitterions.
    Brehm L; Krogsgaard-Larsen P; Schaumburg K; Johansen JS; Falch E; Curtis DR
    J Med Chem; 1986 Feb; 29(2):224-9. PubMed ID: 3005567
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Glycine antagonists structurally related to muscimol, THIP, or isoguvacine.
    Krogsgaard-Larsen P; Hjeds H; Curtis DR; Leah JD; Peet MJ
    J Neurochem; 1982 Nov; 39(5):1319-24. PubMed ID: 6288870
    [TBL] [Abstract][Full Text] [Related]  

  • 3. 4,5,6,7-Tetrahydroisothiazolo[5,4-c]pyridin-3-ol and related analogues of THIP. Synthesis and biological activity.
    Krogsgaard-Larsen P; Mikkelsen H; Jacobsen P; Falch E; Curtis DR; Peet MJ; Leah JD
    J Med Chem; 1983 Jun; 26(6):895-900. PubMed ID: 6304315
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Glycine antagonists structurally related to 4,5,6,7-tetrahydroisoxazolo [5,4-c]pyridin-3-ol inhibit binding of [3H]strychnine to rat brain membranes.
    Braestrup C; Nielsen M; Krogsgaard-Larsen P
    J Neurochem; 1986 Sep; 47(3):691-6. PubMed ID: 3016180
    [TBL] [Abstract][Full Text] [Related]  

  • 5. 3- and 5-isoxazolol zwitterions: an ab initio molecular orbital study relating to GABA agonism and antagonism.
    Boulanger T; Vercauteren DP; Durant F; Andre JM
    J Theor Biol; 1987 Aug; 127(4):479-89. PubMed ID: 2832660
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
    Byberg JR; Labouta IM; Falch E; Hjeds H; Krogsgaard-Larsen P; Curtis DR; Gynther BD
    Drug Des Deliv; 1987 May; 1(4):261-74. PubMed ID: 2855566
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Selective inhibitors of glial GABA uptake: synthesis, absolute stereochemistry, and pharmacology of the enantiomers of 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and analogues.
    Falch E; Perregaard J; FrŁlund B; SŁkilde B; Buur A; Hansen LM; Frydenvang K; Brehm L; Bolvig T; Larsson OM; Sanchez C; White HS; Schousboe A; Krogsgaard-Larsen P
    J Med Chem; 1999 Dec; 42(26):5402-14. PubMed ID: 10639282
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Molecular modeling of the weak glycine antagonist iso-THAO.
    Aprison MH; Lipkowitz KB
    J Neurosci Res; 1991 Oct; 30(2):442-6. PubMed ID: 1724675
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Novel class of potent 4-arylalkyl substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.
    Frølund B; Jørgensen AT; Tagmose L; Stensbøl TB; Vestergaard HT; Engblom C; Kristiansen U; Sanchez C; Krogsgaard-Larsen P; Liljefors T
    J Med Chem; 2002 Jun; 45(12):2454-68. PubMed ID: 12036354
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Action of bicyclic isoxazole GABA analogues on GABA transporters and its relation to anticonvulsant activity.
    Bolvig T; Larsson OM; Pickering DS; Nelson N; Falch E; Krogsgaard-Larsen P; Schousboe A
    Eur J Pharmacol; 1999 Jun; 375(1-3):367-74. PubMed ID: 10443590
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Kinetic cooperative effect of glycine receptor agonists and antagonists on the dissociation of strychnine binding.
    Maksay G
    Eur J Pharmacol; 1993 Apr; 245(2):183-5. PubMed ID: 8387928
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Design, synthesis, and pharmacological characterization of N- and O-substituted 5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol analogues: novel 5-HT(2A)/5-HT(2C) receptor agonists with pro-cognitive properties.
    Jensen AA; Plath N; Pedersen MH; Isberg V; Krall J; Wellendorph P; Stensbøl TB; Gloriam DE; Krogsgaard-Larsen P; Frølund B
    J Med Chem; 2013 Feb; 56(3):1211-27. PubMed ID: 23301527
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Anticonvulsant activity of the glial GABA uptake inhibitor, THAO, in chemical seizures.
    Gonsalves SF; Twitchell B; Harbaugh RE; Krogsgaard-Larsen P; Schousboe A
    Eur J Pharmacol; 1989 Sep; 168(2):265-8. PubMed ID: 2532604
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Amplification by glycine of the effect of the GABA transport inhibitor THPO on synaptosomal GABA level.
    Wood JD; Krogsgaard-Larsen P; Schousboe A
    Neurochem Res; 1988 Oct; 13(10):917-21. PubMed ID: 3216948
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Potent 4-aryl- or 4-arylalkyl-substituted 3-isoxazolol GABA(A) antagonists: synthesis, pharmacology, and molecular modeling.
    Frølund B; Jensen LS; Guandalini L; Canillo C; Vestergaard HT; Kristiansen U; Nielsen B; Stensbøl TB; Madsen C; Krogsgaard-Larsen P; Liljefors T
    J Med Chem; 2005 Jan; 48(2):427-39. PubMed ID: 15658856
    [TBL] [Abstract][Full Text] [Related]  

  • 16. On a molecular comparison of strong and weak antagonists at the glycinergic receptor.
    Aprison MH; Galvez-Ruano E; Lipkowitz KB
    J Neurosci Res; 1995 Jun; 41(2):259-69. PubMed ID: 7650761
    [TBL] [Abstract][Full Text] [Related]  

  • 17. Prolongation of gamma-aminobutyric acid-mediated inhibitory postsynaptic potentials by 4,5,6,7-tetrahydroisoxazolo[4,5-c]pyridin-3-ol (THPO).
    Korn SJ; Dingledine R
    Neurosci Lett; 1986 Feb; 64(1):47-52. PubMed ID: 3960387
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Organic hydroxylamine derivatives. X. Structural analogues of gamma-aminobutyric acid (GABA) of the isoxazole enol-betaine type. Synthesis of 5,6,7,8-tetrahydro-4H-isoxazolo (4,5-D) azepin-3-ol zwitterion and 4,5,6,7-tetrahydroisoxazole (4,5-c) pyridin-3-ol zwitterion.
    Krogsgaard-Larsen P; Hjeds H
    Acta Chem Scand B; 1974; 28(5):533-8. PubMed ID: 4153428
    [No Abstract]   [Full Text] [Related]  

  • 19. Correlation between anticonvulsant activity and inhibitory action on glial gamma-aminobutyric acid uptake of the highly selective mouse gamma-aminobutyric acid transporter 1 inhibitor 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and its N-alkylated analogs.
    White HS; Sarup A; Bolvig T; Kristensen AS; Petersen G; Nelson N; Pickering DS; Larsson OM; Frølund B; Krogsgaard-Larsen P; Schousboe A
    J Pharmacol Exp Ther; 2002 Aug; 302(2):636-44. PubMed ID: 12130726
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Design and synthesis of a new series of 4-alkylated 3-isoxazolol GABA A antagonists.
    Frølund B; Tagmose L; Jørgensen AT; Kristiansen U; Stensbøl TB; Liljefors T; Krogsgaard-Larsen P
    Eur J Med Chem; 2003 Apr; 38(4):447-9. PubMed ID: 12750034
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 6.