BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

358 related articles for article (PubMed ID: 30104277)

  • 1. Activity of Aromathecins against African Trypanosomes.
    Nenortas NP; Cinelli MA; Morrell AE; Cushman M; Shapiro TA
    Antimicrob Agents Chemother; 2018 Nov; 62(11):. PubMed ID: 30104277
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Newly identified antibacterial compounds are topoisomerase poisons in African trypanosomes.
    Tang SC; Shapiro TA
    Antimicrob Agents Chemother; 2010 Feb; 54(2):620-6. PubMed ID: 20008775
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Anti-trypanosomal activities of DNA topoisomerase inhibitors.
    Deterding A; Dungey FA; Thompson KA; Steverding D
    Acta Trop; 2005 Mar; 93(3):311-6. PubMed ID: 15715983
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro.
    Ferrigno F; Biancofiore I; Malancona S; Ponzi S; Paonessa G; Graziani R; Bresciani A; Gennari N; Di Marco A; Kaiser M; Summa V; Harper S; Ontoria JM
    Bioorg Med Chem Lett; 2018 Dec; 28(23-24):3689-3692. PubMed ID: 30482621
    [TBL] [Abstract][Full Text] [Related]  

  • 5. 9- and 11-Substituted 4-azapaullones are potent and selective inhibitors of African trypanosoma.
    Maiwald F; Benítez D; Charquero D; Dar MA; Erdmann H; Preu L; Koch O; Hölscher C; Loaëc N; Meijer L; Comini MA; Kunick C
    Eur J Med Chem; 2014 Aug; 83():274-83. PubMed ID: 24973661
    [TBL] [Abstract][Full Text] [Related]  

  • 6. The kinetoplastid chemotherapy revisited: current drugs, recent advances and future perspectives.
    Castillo E; Dea-Ayuela MA; Bolás-Fernández F; Rangel M; González-Rosende ME
    Curr Med Chem; 2010; 17(33):4027-51. PubMed ID: 20939823
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Identification of novel inhibitors of UDP-Glc 4'-epimerase, a validated drug target for african sleeping sickness.
    Urbaniak MD; Tabudravu JN; Msaki A; Matera KM; Brenk R; Jaspars M; Ferguson MA
    Bioorg Med Chem Lett; 2006 Nov; 16(22):5744-7. PubMed ID: 16962325
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Sleeping sickness pathogen (Trypanosoma brucei) and natural products: therapeutic targets and screening systems.
    Hannaert V
    Planta Med; 2011 Apr; 77(6):586-97. PubMed ID: 20945274
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Identification and Characterization of FTY720 for the Treatment of Human African Trypanosomiasis.
    Jones AJ; Kaiser M; Avery VM
    Antimicrob Agents Chemother; 2015 Dec; 60(3):1859-61. PubMed ID: 26666915
    [TBL] [Abstract][Full Text] [Related]  

  • 10. 3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis.
    Ferrins L; Rahmani R; Sykes ML; Jones AJ; Avery VM; Teston E; Almohaywi B; Yin J; Smith J; Hyland C; White KL; Ryan E; Campbell M; Charman SA; Kaiser M; Baell JB
    Eur J Med Chem; 2013 Aug; 66():450-65. PubMed ID: 23831695
    [TBL] [Abstract][Full Text] [Related]  

  • 11. Optimization of physicochemical properties for 4-anilinoquinazoline inhibitors of trypanosome proliferation.
    Woodring JL; Bachovchin KA; Brady KG; Gallerstein MF; Erath J; Tanghe S; Leed SE; Rodriguez A; Mensa-Wilmot K; Sciotti RJ; Pollastri MP
    Eur J Med Chem; 2017 Dec; 141():446-459. PubMed ID: 29049963
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Chemotherapeutic strategies against Trypanosoma brucei: drug targets vs. drug targeting.
    Lüscher A; de Koning HP; Mäser P
    Curr Pharm Des; 2007; 13(6):555-67. PubMed ID: 17346174
    [TBL] [Abstract][Full Text] [Related]  

  • 13. New heterocyclic compounds: Synthesis and antitrypanosomal properties.
    Pomel S; Dubar F; Forge D; Loiseau PM; Biot C
    Bioorg Med Chem; 2015 Aug; 23(16):5168-74. PubMed ID: 25835356
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Potent antitrypanosomal activities of heat shock protein 90 inhibitors in vitro and in vivo.
    Meyer KJ; Shapiro TA
    J Infect Dis; 2013 Aug; 208(3):489-99. PubMed ID: 23630365
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Activity of indenoisoquinolines against African trypanosomes.
    Bakshi RP; Sang D; Morrell A; Cushman M; Shapiro TA
    Antimicrob Agents Chemother; 2009 Jan; 53(1):123-8. PubMed ID: 18824603
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Screening of acyl hydrazide proteinase inhibitors for antiparasitic activity against Trypanosoma brucei.
    Caffrey CR; Schanz M; Nkemngu NJ; Brush M; Hansell E; Cohen FE; Flaherty TM; McKerrow JH; Steverding D
    Int J Antimicrob Agents; 2002 Mar; 19(3):227-31. PubMed ID: 11932146
    [TBL] [Abstract][Full Text] [Related]  

  • 17. [Prophylactic and curative action of Ridzol-S and Ronidazole in experimental trypanosomiasis caused by Trypanosoma brucei et T. evansi].
    Tchalim TK
    Ann Soc Belg Med Trop; 1980 Sep; 60(3):263-70. PubMed ID: 7195691
    [No Abstract]   [Full Text] [Related]  

  • 18. Novel distamycin analogues that block the cell cycle of African trypanosomes with high selectivity and potency.
    Franco J; Scarone L; Comini MA
    Eur J Med Chem; 2020 Mar; 189():112043. PubMed ID: 31978782
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Diamidine activity against trypanosomes: the state of the art.
    Soeiro MN; de Castro SL; de Souza EM; Batista DG; Silva CF; Boykin DW
    Curr Mol Pharmacol; 2008 Jun; 1(2):151-61. PubMed ID: 20021429
    [TBL] [Abstract][Full Text] [Related]  

  • 20. The biochemistry of African trypanosomes and its significance for chemotherapy.
    Braide VB
    J Vet Pharmacol Ther; 1987 Sep; 10(3):191-201. PubMed ID: 3309362
    [No Abstract]   [Full Text] [Related]  

    [Next]    [New Search]
    of 18.