123 related articles for article (PubMed ID: 30143421)
1. New piperidine-based derivatives as sigma receptor ligands. Synthesis and pharmacological evaluation.
Zampieri D; Romano M; Menegazzi R; Mamolo MG
Bioorg Med Chem Lett; 2018 Oct; 28(19):3206-3209. PubMed ID: 30143421
[TBL] [Abstract][Full Text] [Related]
2. Improving selectivity preserving affinity: new piperidine-4-carboxamide derivatives as effective sigma-1-ligands.
Zampieri D; Laurini E; Vio L; Fermeglia M; Pricl S; Wünsch B; Schepmann D; Mamolo MG
Eur J Med Chem; 2015 Jan; 90():797-808. PubMed ID: 25528334
[TBL] [Abstract][Full Text] [Related]
3. Spiro[1,2,4-benzotriazine-3(4H),4'-(1'-substituted)piperidines] and related compounds as ligands for sigma receptors.
Novelli F; Sparatore F
Farmaco; 2002 Nov; 57(11):871-82. PubMed ID: 12484535
[TBL] [Abstract][Full Text] [Related]
4. Synthesis, binding, and functional properties of tetrahydroisoquinolino-2-alkyl phenones as selective σ
Xie XY; Li YY; Ma WH; Chen AF; Sun YT; Lee JY; Riad A; Xu DH; Mach RH; Huang YS
Eur J Med Chem; 2021 Jan; 209():112906. PubMed ID: 33049607
[TBL] [Abstract][Full Text] [Related]
5. Novel piperidine sigma receptor ligands as potential antipsychotic drugs.
Gilligan PJ; Cain GA; Christos TE; Cook L; Drummond S; Johnson AL; Kergaye AA; McElroy JF; Rohrbach KW; Schmidt WK
J Med Chem; 1992 Nov; 35(23):4344-61. PubMed ID: 1360026
[TBL] [Abstract][Full Text] [Related]
6. Oxa-Pictet-Spengler reaction as key step in the synthesis of novel σ receptor ligands with 2-benzopyran structure.
Knappmann I; Schepmann D; Wünsch B
Bioorg Med Chem; 2016 Sep; 24(18):4045-4055. PubMed ID: 27396684
[TBL] [Abstract][Full Text] [Related]
7. Synthesis of Aminoethyl-Substituted Piperidine Derivatives as σ
Holtschulte C; Börgel F; Westphälinger S; Schepmann D; Civenni G; Laurini E; Marson D; Catapano CV; Pricl S; Wünsch B
ChemMedChem; 2022 Apr; 17(7):e202100735. PubMed ID: 35077612
[TBL] [Abstract][Full Text] [Related]
8. High-affinity sigma-1 (σ
Niso M; Mosier PD; Marottoli R; Ferorelli S; Cassano G; Gasparre G; Leopoldo M; Berardi F; Abate C
Future Med Chem; 2019 Oct; 11(19):2547-2562. PubMed ID: 31633399
[No Abstract] [Full Text] [Related]
9. Synthesis and receptor binding studies of novel 4,4-disubstituted arylalkyl/arylalkylsulfonyl piperazine and piperidine-based derivatives as a new class of σ1 ligands.
Sadeghzadeh M; Sheibani S; Ghandi M; Daha FJ; Amanlou M; Arjmand M; Hasani Bozcheloie A
Eur J Med Chem; 2013 Jun; 64():488-97. PubMed ID: 23680866
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and binding assays of novel 3,3-dimethylpiperidine derivatives with various lipophilicities as σ₁ receptor ligands.
Ferorelli S; Abate C; Pedone MP; Colabufo NA; Contino M; Perrone R; Berardi F
Bioorg Med Chem; 2011 Dec; 19(24):7612-22. PubMed ID: 22075234
[TBL] [Abstract][Full Text] [Related]
11. Investigating isoindoline, tetrahydroisoquinoline, and tetrahydrobenzazepine scaffolds for their sigma receptor binding properties.
Linkens K; Schmidt HR; Sahn JJ; Kruse AC; Martin SF
Eur J Med Chem; 2018 May; 151():557-567. PubMed ID: 29656199
[TBL] [Abstract][Full Text] [Related]
12. Preparation of novel analogs of 2-arylpiperidines and evaluation of their sigma receptor binding affinities.
Walby GD; Martin SF
Eur J Med Chem; 2022 May; 235():114310. PubMed ID: 35395511
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of sigma receptor ligands with unsymmetrical spiro connection of the piperidine moiety.
Jasper A; Schepmann D; Lehmkuhl K; Vela JM; Buschmann H; Holenz J; Wünsch B
Eur J Med Chem; 2009 Nov; 44(11):4306-14. PubMed ID: 19709783
[TBL] [Abstract][Full Text] [Related]
14. Synthesis and evaluation of a 18F-labeled spirocyclic piperidine derivative as promising σ1 receptor imaging agent.
Chen YY; Wang X; Zhang JM; Deuther-Conrad W; Zhang XJ; Huang Y; Li Y; Ye JJ; Cui MC; Steinbach J; Brust P; Liu BL; Jia HM
Bioorg Med Chem; 2014 Oct; 22(19):5270-8. PubMed ID: 25189691
[TBL] [Abstract][Full Text] [Related]
15. Pharmacological characterization of high-affinity σ
Schepmann D; Neue C; Westphälinger S; Müller C; Bracher F; Lange C; Bednarski P; Almansa C; Friedland K; Räbiger V; Düfer M; Wünsch B
J Pharm Pharmacol; 2020 Feb; 72(2):236-248. PubMed ID: 31743446
[TBL] [Abstract][Full Text] [Related]
16. Targeting σ
Wood MD; Sahn JJ; Martin SF
Eur J Med Chem; 2022 Dec; 243():114696. PubMed ID: 36088757
[TBL] [Abstract][Full Text] [Related]
17. Synthesis and structure-activity relationships of 1-aralkyl-4-benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent sigma ligands.
Costantino L; Gandolfi F; Sorbi C; Franchini S; Prezzavento O; Vittorio F; Ronsisvalle G; Leonardi A; Poggesi E; Brasili L
J Med Chem; 2005 Jan; 48(1):266-73. PubMed ID: 15634021
[TBL] [Abstract][Full Text] [Related]
18. Neuroprotective Efficacy of a Sigma 2 Receptor/TMEM97 Modulator (DKR-1677) after Traumatic Brain Injury.
Vázquez-Rosa E; Watson MR; Sahn JJ; Hodges TR; Schroeder RE; Cintrón-Pérez CJ; Shin MK; Yin TC; Emery JL; Martin SF; Liebl DJ; Pieper AA
ACS Chem Neurosci; 2019 Mar; 10(3):1595-1602. PubMed ID: 30421909
[TBL] [Abstract][Full Text] [Related]
19. N-arylalkylpiperidines as high-affinity sigma-1 and sigma-2 receptor ligands: phenylpropylamines as potential leads for selective sigma-2 agents.
Maeda DY; Williams W; Kim WE; Thatcher LN; Bowen WD; Coop A
Bioorg Med Chem Lett; 2002 Feb; 12(3):497-500. PubMed ID: 11814827
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and in vitro biological evaluation of carbonyl group-containing analogues for σ1 receptors.
Wang W; Cui J; Lu X; Padakanti PK; Xu J; Parsons SM; Luedtke RR; Rath NP; Tu Z
J Med Chem; 2011 Aug; 54(15):5362-72. PubMed ID: 21732626
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]