182 related articles for article (PubMed ID: 30343193)
1. Identification of potential antivirulence agents by substitution-oriented screening for inhibitors of Streptococcus pyogenes sortase A.
Wójcik M; Eleftheriadis N; Zwinderman MRH; Dömling ASS; Dekker FJ; Boersma YL
Eur J Med Chem; 2019 Jan; 161():93-100. PubMed ID: 30343193
[TBL] [Abstract][Full Text] [Related]
2. Optimized protocols for assessing libraries of poorly soluble sortase A inhibitors for antibacterial activity against medically-relevant bacteria, toxicity and enzyme inhibition.
Alharthi S; Ziora ZM; Moyle PM
Bioorg Med Chem; 2021 Dec; 52():116527. PubMed ID: 34839159
[TBL] [Abstract][Full Text] [Related]
3. Asymmetric Disulfanylbenzamides as Irreversible and Selective Inhibitors of Staphylococcus aureus Sortase A.
Barthels F; Marincola G; Marciniak T; Konhäuser M; Hammerschmidt S; Bierlmeier J; Distler U; Wich PR; Tenzer S; Schwarzer D; Ziebuhr W; Schirmeister T
ChemMedChem; 2020 May; 15(10):839-850. PubMed ID: 32118357
[TBL] [Abstract][Full Text] [Related]
4. Sortase A: an ideal target for anti-virulence drug development.
Cascioferro S; Totsika M; Schillaci D
Microb Pathog; 2014 Dec; 77():105-12. PubMed ID: 25457798
[TBL] [Abstract][Full Text] [Related]
5. Sortase A Inhibitors: Recent Advances and Future Perspectives.
Cascioferro S; Raffa D; Maggio B; Raimondi MV; Schillaci D; Daidone G
J Med Chem; 2015 Dec; 58(23):9108-23. PubMed ID: 26280844
[TBL] [Abstract][Full Text] [Related]
6. Inhibition of sortase-mediated Staphylococcus aureus adhesion to fibronectin via fibronectin-binding protein by sortase inhibitors.
Oh KB; Oh MN; Kim JG; Shin DS; Shin J
Appl Microbiol Biotechnol; 2006 Mar; 70(1):102-6. PubMed ID: 16010573
[TBL] [Abstract][Full Text] [Related]
7. Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform.
Kudryavtsev KV; Bentley ML; McCafferty DG
Bioorg Med Chem; 2009 Apr; 17(7):2886-93. PubMed ID: 19269184
[TBL] [Abstract][Full Text] [Related]
8. NMR structure-based optimization of Staphylococcus aureus sortase A pyridazinone inhibitors.
Chan AH; Yi SW; Weiner EM; Amer BR; Sue CK; Wereszczynski J; Dillen CA; Senese S; Torres JZ; McCammon JA; Miller LS; Jung ME; Clubb RT
Chem Biol Drug Des; 2017 Sep; 90(3):327-344. PubMed ID: 28160417
[TBL] [Abstract][Full Text] [Related]
9. Sortase transpeptidases: insights into mechanism, substrate specificity, and inhibition.
Clancy KW; Melvin JA; McCafferty DG
Biopolymers; 2010; 94(4):385-96. PubMed ID: 20593474
[TBL] [Abstract][Full Text] [Related]
10. Crystal structure of Streptococcus pyogenes sortase A: implications for sortase mechanism.
Race PR; Bentley ML; Melvin JA; Crow A; Hughes RK; Smith WD; Sessions RB; Kehoe MA; McCafferty DG; Banfield MJ
J Biol Chem; 2009 Mar; 284(11):6924-33. PubMed ID: 19129180
[TBL] [Abstract][Full Text] [Related]
11. Molecular basis of Streptococcus mutans sortase A inhibition by the flavonoid natural product trans-chalcone.
Wallock-Richards DJ; Marles-Wright J; Clarke DJ; Maitra A; Dodds M; Hanley B; Campopiano DJ
Chem Commun (Camb); 2015 Jul; 51(52):10483-5. PubMed ID: 26029850
[TBL] [Abstract][Full Text] [Related]
12. Combined pharmacophore and 3D-QSAR study on a series of Staphylococcus aureus Sortase A inhibitors.
Uddin R; Lodhi MU; Ul-Haq Z
Chem Biol Drug Des; 2012 Aug; 80(2):300-14. PubMed ID: 22553957
[TBL] [Abstract][Full Text] [Related]
13. Synthesis of (2R,3S) 3-amino-4-mercapto-2-butanol, a threonine analogue for covalent inhibition of sortases.
Jung ME; Clemens JJ; Suree N; Liew CK; Pilpa R; Campbell DO; Clubb RT
Bioorg Med Chem Lett; 2005 Nov; 15(22):5076-9. PubMed ID: 16169722
[TBL] [Abstract][Full Text] [Related]
14. Antiinfective therapy with a small molecule inhibitor of Staphylococcus aureus sortase.
Zhang J; Liu H; Zhu K; Gong S; Dramsi S; Wang YT; Li J; Chen F; Zhang R; Zhou L; Lan L; Jiang H; Schneewind O; Luo C; Yang CG
Proc Natl Acad Sci U S A; 2014 Sep; 111(37):13517-22. PubMed ID: 25197057
[TBL] [Abstract][Full Text] [Related]
15. Sortase A localizes to distinct foci on the Streptococcus pyogenes membrane.
Raz A; Fischetti VA
Proc Natl Acad Sci U S A; 2008 Nov; 105(47):18549-54. PubMed ID: 19017791
[TBL] [Abstract][Full Text] [Related]
16. Designing of potential inhibitors against Staphylococcus aureus sortase A: Combined analogue and structure based approach with in vitro validation.
Raj KK; Ganesh Kumar V; Leela Madhuri C; Mathi P; Durga Lakshmi R; Ravi M; Sri Ramudu B; Venkata Rao SV; Ramachandran D
J Mol Graph Model; 2015 Jul; 60():89-97. PubMed ID: 26119984
[TBL] [Abstract][Full Text] [Related]
17. Astilbin Inhibits the Activity of Sortase A from
Wang J; Shi Y; Jing S; Dong H; Wang D; Wang T
Molecules; 2019 Jan; 24(3):. PubMed ID: 30696091
[No Abstract] [Full Text] [Related]
18. Quercitrin, an inhibitor of Sortase A, interferes with the adhesion of Staphylococcal aureus.
Liu B; Chen F; Bi C; Wang L; Zhong X; Cai H; Deng X; Niu X; Wang D
Molecules; 2015 Apr; 20(4):6533-43. PubMed ID: 25871372
[TBL] [Abstract][Full Text] [Related]
19. Discovery and structure-activity relationship studies of irreversible benzisothiazolinone-based inhibitors against Staphylococcus aureus sortase A transpeptidase.
Zhulenkovs D; Rudevica Z; Jaudzems K; Turks M; Leonchiks A
Bioorg Med Chem; 2014 Nov; 22(21):5988-6003. PubMed ID: 25282649
[TBL] [Abstract][Full Text] [Related]
20. Synthetic analogs of indole-containing natural products as inhibitors of sortase A and isocitrate lyase.
Lee YJ; Han YR; Park W; Nam SH; Oh KB; Lee HS
Bioorg Med Chem Lett; 2010 Dec; 20(23):6882-5. PubMed ID: 21035332
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]