BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

145 related articles for article (PubMed ID: 30380445)

  • 1. Synthesis of 1,2,4-triazole-5-on derivatives and determination of carbonic anhydrase II isoenzyme inhibition effects.
    Akin S; Ayaloglu H; Gultekin E; Colak A; Bekircan O; Akatin MY
    Bioorg Chem; 2019 Mar; 83():170-179. PubMed ID: 30380445
    [TBL] [Abstract][Full Text] [Related]  

  • 2. Design and synthesis of novel benzenesulfonamide containing 1,2,3-triazoles as potent human carbonic anhydrase isoforms I, II, IV and IX inhibitors.
    Kumar R; Vats L; Bua S; Supuran CT; Sharma PK
    Eur J Med Chem; 2018 Jul; 155():545-551. PubMed ID: 29909339
    [TBL] [Abstract][Full Text] [Related]  

  • 3. Novel Re(I) tricarbonyl coordination compounds based on 2-pyridyl-1,2,3-triazole derivatives bearing a 4-amino-substituted benzenesulfonamide arm: synthesis, crystal structure, computational studies and inhibitory activity against carbonic anhydrase I, II, and IX isoforms†.
    Aimene Y; Eychenne R; Mallet-Ladeira S; Saffon N; Winum JY; Nocentini A; Supuran CT; Benoist E; Seridi A
    J Enzyme Inhib Med Chem; 2019 Dec; 34(1):773-782. PubMed ID: 30843736
    [TBL] [Abstract][Full Text] [Related]  

  • 4. Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors.
    Vats L; Sharma V; Angeli A; Kumar R; Supuran CT; Sharma PK
    Eur J Med Chem; 2018 Apr; 150():678-686. PubMed ID: 29571155
    [TBL] [Abstract][Full Text] [Related]  

  • 5. The synthesis of (Z)-4-oxo-4-(arylamino)but-2-enoic acids derivatives and determination of their inhibition properties against human carbonic anhydrase I and II isoenzymes.
    Oktay K; Köse LP; Şendil K; Gültekin MS; Gülçin İ; Supuran CT
    J Enzyme Inhib Med Chem; 2016 Dec; 31(6):939-45. PubMed ID: 26308288
    [TBL] [Abstract][Full Text] [Related]  

  • 6. Potential inhibitors of human carbonic anhydrase isozymes I and II: Design, synthesis and docking studies of new 1,3,4-thiadiazole derivatives.
    Altıntop MD; Sever B; Özdemir A; Kucukoglu K; Onem H; Nadaroglu H; Kaplancıklı ZA
    Bioorg Med Chem; 2017 Jul; 25(13):3547-3554. PubMed ID: 28511907
    [TBL] [Abstract][Full Text] [Related]  

  • 7. Sulfamates of methyl triterpenoates are effective and competitive inhibitors of carbonic anhydrase II.
    Schwarz S; Sommerwerk S; Lucas SD; Heller L; Csuk R
    Eur J Med Chem; 2014 Oct; 86():95-102. PubMed ID: 25147151
    [TBL] [Abstract][Full Text] [Related]  

  • 8. Oxidation of cyanobenzocycloheptatrienes: Synthesis, photooxygenation reaction and carbonic anhydrase isoenzymes inhibition properties of some new benzotropone derivatives.
    Güney M; Coşkun A; Topal F; Daştan A; Gülçin I; Supuran CT
    Bioorg Med Chem; 2014 Jul; 22(13):3537-43. PubMed ID: 24856184
    [TBL] [Abstract][Full Text] [Related]  

  • 9. Synthesis and evaluation of N-heteroarylsubstituted triazolosulfonamides as carbonic anhydrase inhibitors.
    Balci A; Arslan M; Nixha AR; Bilen C; Ergun A; Gençer N
    J Enzyme Inhib Med Chem; 2015 Jun; 30(3):377-82. PubMed ID: 25068730
    [TBL] [Abstract][Full Text] [Related]  

  • 10. Synthesis and carbonic anhydrase inhibitory activities of new thienyl-substituted pyrazoline benzenesulfonamides.
    Mete E; Comez B; Inci Gul H; Gulcin I; Supuran CT
    J Enzyme Inhib Med Chem; 2016; 31(sup2):1-5. PubMed ID: 27435177
    [TBL] [Abstract][Full Text] [Related]  

  • 11. The effects of some bromophenols on human carbonic anhydrase isoenzymes.
    Taslimi P; Gülçin İ; Öztaşkın N; Çetinkaya Y; Göksu S; Alwasel SH; Supuran CT
    J Enzyme Inhib Med Chem; 2016 Aug; 31(4):603-7. PubMed ID: 26133541
    [TBL] [Abstract][Full Text] [Related]  

  • 12. Synthesis of 5-methyl-2,4-dihydro-3H-1,2,4-triazole-3-one's aryl Schiff base derivatives and investigation of carbonic anhydrase and cholinesterase (AChE, BuChE) inhibitory properties.
    Özil M; Balaydın HT; Şentürk M
    Bioorg Chem; 2019 May; 86():705-713. PubMed ID: 30836234
    [TBL] [Abstract][Full Text] [Related]  

  • 13. Carbonic anhydrase inhibitors. Inhibition of the cytosolic and tumor-associated carbonic anhydrase isozymes I, II and IX with some 1,3,4-oxadiazole- and 1,2,4-triazole-thiols.
    Almajan GL; Barbuceanu SF; Innocenti A; Scozzafava A; Supuran CT
    J Enzyme Inhib Med Chem; 2008 Feb; 23(1):101-7. PubMed ID: 18341261
    [TBL] [Abstract][Full Text] [Related]  

  • 14. Inhibition of human carbonic anhydrase isozymes I, II and VI with a series of bisphenol, methoxy and bromophenol compounds.
    Balaydin HT; Durdaği S; Ekinci D; Sentürk M; Göksu S; Menzek A
    J Enzyme Inhib Med Chem; 2012 Aug; 27(4):467-75. PubMed ID: 21815772
    [TBL] [Abstract][Full Text] [Related]  

  • 15. Three-component synthesis and carbonic anhydrase inhibitory properties of novel octahydroacridines incorporating sulfaguanidine scaffold.
    Ulus R; Kaya M; Demir D; Tunca E; Bülbül M
    J Enzyme Inhib Med Chem; 2016; 31(sup2):63-69. PubMed ID: 27237188
    [TBL] [Abstract][Full Text] [Related]  

  • 16. Synthesis and biological evaluation of benzenesulphonamide-bearing 1,4,5-trisubstituted-1,2,3-triazoles possessing human carbonic anhydrase I, II, IV, and IX inhibitory activity.
    Kumar R; Sharma V; Bua S; Supuran CT; Sharma PK
    J Enzyme Inhib Med Chem; 2017 Dec; 32(1):1187-1194. PubMed ID: 28891338
    [TBL] [Abstract][Full Text] [Related]  

  • 17. The human carbonic anhydrase isoenzymes I and II (hCA I and II) inhibition effects of trimethoxyindane derivatives.
    Taslimi P; Gulcin I; Ozgeris B; Goksu S; Tumer F; Alwasel SH; Supuran CT
    J Enzyme Inhib Med Chem; 2016; 31(1):152-7. PubMed ID: 25697270
    [TBL] [Abstract][Full Text] [Related]  

  • 18. Design, Synthesis and Molecular Docking Study of Novel 3-Phenyl-β-Alanine-Based Oxadiazole Analogues as Potent Carbonic Anhydrase II Inhibitors.
    Rafiq K; Ur Rehman N; Halim SA; Khan M; Khan A; Al-Harrasi A
    Molecules; 2022 Jan; 27(3):. PubMed ID: 35164091
    [TBL] [Abstract][Full Text] [Related]  

  • 19. Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors.
    Lolak N; Akocak S; Bua S; Koca M; Supuran CT
    Bioorg Chem; 2018 Apr; 77():542-547. PubMed ID: 29462772
    [TBL] [Abstract][Full Text] [Related]  

  • 20. Inhibition of carbonic anhydrases with glycosyltriazole benzene sulfonamides.
    Wilkinson BL; Innocenti A; Vullo D; Supuran CT; Poulsen SA
    J Med Chem; 2008 Mar; 51(6):1945-53. PubMed ID: 18307288
    [TBL] [Abstract][Full Text] [Related]  

    [Next]    [New Search]
    of 8.