201 related articles for article (PubMed ID: 30569867)
21. Caffeoyl naphthalenesulfonamide derivatives as HIV integrase inhibitors.
Xu YW; Zhao GS; Shin CG; Zang HC; Lee CK; Lee YS
Bioorg Med Chem; 2003 Aug; 11(17):3589-93. PubMed ID: 12901903
[TBL] [Abstract][Full Text] [Related]
22. Structure-activity relationships and binding mode of styrylquinolines as potent inhibitors of HIV-1 integrase and replication of HIV-1 in cell culture.
Zouhiri F; Mouscadet JF; Mekouar K; Desmaële D; Savouré D; Leh H; Subra F; Le Bret M; Auclair C; d'Angelo J
J Med Chem; 2000 Apr; 43(8):1533-40. PubMed ID: 10780910
[TBL] [Abstract][Full Text] [Related]
23. Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomers.
Rivero-Buceta E; Carrero P; Casanova E; Doyagüez EG; Madrona A; Quesada E; Peréz-Pérez MJ; Mateos R; Bravo L; Mathys L; Noppen S; Kiselev E; Marchand C; Pommier Y; Liekens S; Balzarini J; Camarasa MJ; San-Félix A
Eur J Med Chem; 2015 Dec; 106():132-43. PubMed ID: 26540494
[TBL] [Abstract][Full Text] [Related]
24. Exploration of novel thiobarbituric acid-, rhodanine- and thiohydantoin-based HIV-1 integrase inhibitors.
Rajamaki S; Innitzer A; Falciani C; Tintori C; Christ F; Witvrouw M; Debyser Z; Massa S; Botta M
Bioorg Med Chem Lett; 2009 Jul; 19(13):3615-8. PubMed ID: 19447621
[TBL] [Abstract][Full Text] [Related]
25. Diketoacid chelating ligands as dual inhibitors of HIV-1 integration process.
Rogolino D; Carcelli M; Compari C; De Luca L; Ferro S; Fisicaro E; Rispoli G; Neamati N; Debyser Z; Christ F; Chimirri A
Eur J Med Chem; 2014 May; 78():425-30. PubMed ID: 24704615
[TBL] [Abstract][Full Text] [Related]
26. Synthesis, anti-HIV activity, integrase enzyme inhibition and molecular modeling of catechol, hydroquinone and quinol labdane analogs.
Pawar R; Das T; Mishra S; Nutan ; Pancholi B; Gupta SK; Bhat SV
Bioorg Med Chem Lett; 2014 Jan; 24(1):302-7. PubMed ID: 24291042
[TBL] [Abstract][Full Text] [Related]
27. Design and discovery of 5-hydroxy-6-oxo-1,6-dihydropyrimidine-4-carboxamide inhibitors of HIV-1 integrase.
Zhang D; Debnath B; Yu S; Sanchez TW; Christ F; Liu Y; Debyser Z; Neamati N; Zhao G
Bioorg Med Chem; 2014 Oct; 22(19):5446-53. PubMed ID: 25150089
[TBL] [Abstract][Full Text] [Related]
28. Structure activity of 3-aryl-1,3-diketo-containing compounds as HIV-1 integrase inhibitors.
Pais GC; Zhang X; Marchand C; Neamati N; Cowansage K; Svarovskaia ES; Pathak VK; Tang Y; Nicklaus M; Pommier Y; Burke TR
J Med Chem; 2002 Jul; 45(15):3184-94. PubMed ID: 12109903
[TBL] [Abstract][Full Text] [Related]
29. Design of a series of bicyclic HIV-1 integrase inhibitors. Part 1: selection of the scaffold.
Jones ED; Vandegraaff N; Le G; Choi N; Issa W; Macfarlane K; Thienthong N; Winfield LJ; Coates JA; Lu L; Li X; Feng X; Yu C; Rhodes DI; Deadman JJ
Bioorg Med Chem Lett; 2010 Oct; 20(19):5913-7. PubMed ID: 20727748
[TBL] [Abstract][Full Text] [Related]
30. Design and synthesis of N-methylpyrimidone derivatives as HIV-1 integrase inhibitors.
Wang Y; Rong J; Zhang B; Hu L; Wang X; Zeng C
Bioorg Med Chem; 2015 Feb; 23(4):735-41. PubMed ID: 25618597
[TBL] [Abstract][Full Text] [Related]
31. Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity.
Esposito F; Ambrosio FA; Maleddu R; Costa G; Rocca R; Maccioni E; Catalano R; Romeo I; Eleftheriou P; Karia DC; Tsirides P; Godvani N; Pandya H; Corona A; Alcaro S; Artese A; Geronikaki A; Tramontano E
Eur J Med Chem; 2019 Nov; 182():111617. PubMed ID: 31442684
[TBL] [Abstract][Full Text] [Related]
32. Design, synthesis, and anti-integrase activity of catechol-DKA hybrids.
Maurin C; Bailly F; Mbemba G; Mouscadet JF; Cotelle P
Bioorg Med Chem; 2006 May; 14(9):2978-84. PubMed ID: 16412645
[TBL] [Abstract][Full Text] [Related]
33. Synthesis and biological evaluation of geminal disulfones as HIV-1 integrase inhibitors.
Meadows DC; Mathews TB; North TW; Hadd MJ; Kuo CL; Neamati N; Gervay-Hague J
J Med Chem; 2005 Jul; 48(14):4526-34. PubMed ID: 15999991
[TBL] [Abstract][Full Text] [Related]
34. Novel 4-Oxo-4,10-dihydrobenzo[4,5]imidazo[1,2-a]pyrimidine-3-carboxylic Acid Derivatives as HIV-1 Integrase Inhibitors: Synthesis, Docking Studies, Molecular Dynamics Simulation and Biological Activities.
Zadeh EE; Vahabpour R; Beirami AD; Hajimahdi Z; Zarghi A
Med Chem; 2021; 17(9):1060-1071. PubMed ID: 32901587
[TBL] [Abstract][Full Text] [Related]
35. Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action.
Di Santo R; Costi R; Roux A; Artico M; Lavecchia A; Marinelli L; Novellino E; Palmisano L; Andreotti M; Amici R; Galluzzo CM; Nencioni L; Palamara AT; Pommier Y; Marchand C
J Med Chem; 2006 Mar; 49(6):1939-45. PubMed ID: 16539381
[TBL] [Abstract][Full Text] [Related]
36. Preclinical evaluation of 1H-benzylindole derivatives as novel human immunodeficiency virus integrase strand transfer inhibitors.
Hombrouck A; Van Remoortel B; Michiels M; Noppe W; Christ F; Eneroth A; Sahlberg BL; Benkestock K; Vrang L; Johansson NG; Barreca ML; De Luca L; Ferro S; Chimirri A; Debyser Z; Witvrouw M
Antimicrob Agents Chemother; 2008 Aug; 52(8):2861-9. PubMed ID: 18541726
[TBL] [Abstract][Full Text] [Related]
37. Synthesis and HIV-1 integrase inhibitory activities of caffeoylglucosides.
Kim SN; Lee JY; Kim HJ; Shin CG; Park H; Lee YS
Bioorg Med Chem Lett; 2000 Aug; 10(16):1879-82. PubMed ID: 10969990
[TBL] [Abstract][Full Text] [Related]
38. Design and synthesis of 8-hydroxy-[1,6]naphthyridines as novel inhibitors of HIV-1 integrase in vitro and in infected cells.
Zhuang L; Wai JS; Embrey MW; Fisher TE; Egbertson MS; Payne LS; Guare JP; Vacca JP; Hazuda DJ; Felock PJ; Wolfe AL; Stillmock KA; Witmer MV; Moyer G; Schleif WA; Gabryelski LJ; Leonard YM; Lynch JJ; Michelson SR; Young SD
J Med Chem; 2003 Feb; 46(4):453-6. PubMed ID: 12570367
[TBL] [Abstract][Full Text] [Related]
39. Design and synthesis of novel β-diketo derivatives as HIV-1 integrase inhibitors.
Hu L; Zhang S; He X; Luo Z; Wang X; Liu W; Qin X
Bioorg Med Chem; 2012 Jan; 20(1):177-82. PubMed ID: 22154762
[TBL] [Abstract][Full Text] [Related]
40. Rational design of 2-pyrrolinones as inhibitors of HIV-1 integrase.
Ma K; Wang P; Fu W; Wan X; Zhou L; Chu Y; Ye D
Bioorg Med Chem Lett; 2011 Nov; 21(22):6724-7. PubMed ID: 21996518
[TBL] [Abstract][Full Text] [Related]
[Previous] [Next] [New Search]