These tools will no longer be maintained as of December 31, 2024. Archived website can be found here. PubMed4Hh GitHub repository can be found here. Contact NLM Customer Service if you have questions.


BIOMARKERS

Molecular Biopsy of Human Tumors

- a resource for Precision Medicine *

201 related articles for article (PubMed ID: 30569867)

  • 41. The discovery and preclinical evaluation of BMS-707035, a potent HIV-1 integrase strand transfer inhibitor.
    Naidu BN; Walker MA; Sorenson ME; Ueda Y; Matiskella JD; Connolly TP; Dicker IB; Lin Z; Bollini S; Terry BJ; Higley H; Zheng M; Parker DD; Wu D; Adams S; Krystal MR; Meanwell NA
    Bioorg Med Chem Lett; 2018 Jul; 28(12):2124-2130. PubMed ID: 29779976
    [TBL] [Abstract][Full Text] [Related]  

  • 42. Authentic HIV-1 integrase inhibitors.
    Liao C; Marchand C; Burke TR; Pommier Y; Nicklaus MC
    Future Med Chem; 2010 Jul; 2(7):1107-22. PubMed ID: 21426159
    [TBL] [Abstract][Full Text] [Related]  

  • 43. Targeting HIV-1 integrase with strand transfer inhibitors.
    Li Y; Xuan S; Feng Y; Yan A
    Drug Discov Today; 2015 Apr; 20(4):435-49. PubMed ID: 25486307
    [TBL] [Abstract][Full Text] [Related]  

  • 44. Structure-based amelioration of PXR transactivation in a novel series of macrocyclic allosteric inhibitors of HIV-1 integrase.
    Sivaprakasam P; Wang Z; Meanwell NA; Khan JA; Langley DR; Johnson SR; Li G; Pendri A; Connolly TP; Gao M; Camac DM; Klakouski C; Zvyaga T; Cianci C; McAuliffe B; Ding B; Discotto L; Krystal MR; Jenkins S; Peese KM; Narasimhulu Naidu B
    Bioorg Med Chem Lett; 2020 Nov; 30(22):127531. PubMed ID: 32890685
    [TBL] [Abstract][Full Text] [Related]  

  • 45. Design, synthesis and biological evaluation of imidazole and oxazole fragments as HIV-1 integrase-LEDGF/p75 disruptors and inhibitors of microbial pathogens.
    Rashamuse TJ; Harrison AT; Mosebi S; van Vuuren S; Coyanis EM; Bode ML
    Bioorg Med Chem; 2020 Jan; 28(1):115210. PubMed ID: 31753802
    [TBL] [Abstract][Full Text] [Related]  

  • 46. 3D-QSAR studies of quinoline ring derivatives as HIV-1 integrase inhibitors.
    Sun XH; Guan JQ; Tan JJ; Liu C; Wang CX
    SAR QSAR Environ Res; 2012 Oct; 23(7-8):683-703. PubMed ID: 22991976
    [TBL] [Abstract][Full Text] [Related]  

  • 47. Styrylquinoline derivatives: a new class of potent HIV-1 integrase inhibitors that block HIV-1 replication in CEM cells.
    Mekouar K; Mouscadet JF; Desmaële D; Subra F; Leh H; Savouré D; Auclair C; d'Angelo J
    J Med Chem; 1998 Jul; 41(15):2846-57. PubMed ID: 9667973
    [TBL] [Abstract][Full Text] [Related]  

  • 48. Depsides and depsidones as inhibitors of HIV-1 integrase: discovery of novel inhibitors through 3D database searching.
    Neamati N; Hong H; Mazumder A; Wang S; Sunder S; Nicklaus MC; Milne GW; Proksa B; Pommier Y
    J Med Chem; 1997 Mar; 40(6):942-51. PubMed ID: 9083483
    [TBL] [Abstract][Full Text] [Related]  

  • 49. Synthesis and evaluation of 3-hydroxy-3-phenylpropanoate ester–AZT conjugates as potential dual-action HIV-1 Integrase and Reverse Transcriptase inhibitors.
    Manyeruke MH; Olomola TO; Majumder S; Abrahams S; Isaacs M; Mautsa N; Mosebi S; Mnkandhla D; Hewer R; Hoppe HC; Klein R; Kaye PT
    Bioorg Med Chem; 2015 Dec; 23(24):7521-8. PubMed ID: 26775541
    [TBL] [Abstract][Full Text] [Related]  

  • 50. Development of tricyclic hydroxy-1H-pyrrolopyridine-trione containing HIV-1 integrase inhibitors.
    Zhao XZ; Maddali K; Metifiot M; Smith SJ; Vu BC; Marchand C; Hughes SH; Pommier Y; Burke TR
    Bioorg Med Chem Lett; 2011 May; 21(10):2986-90. PubMed ID: 21493066
    [TBL] [Abstract][Full Text] [Related]  

  • 51. Design, synthesis, and biological evaluation of novel tricyclic HIV-1 integrase inhibitors by modification of its pyridine ring.
    Metobo SE; Jin H; Tsiang M; Kim CU
    Bioorg Med Chem Lett; 2006 Aug; 16(15):3985-8. PubMed ID: 16723226
    [TBL] [Abstract][Full Text] [Related]  

  • 52. Petra/Osiris/Molinspiration and Molecular Docking Analyses of 3-Hydroxy-Indolin-2-one Derivatives as Potential Antiviral Agents.
    Hadda TB; Rastija V; AlMalki F; Titi A; Touzani R; Mabkhot YN; Khalid S; Zarrouk A; Siddiqui BS
    Curr Comput Aided Drug Des; 2021; 17(1):123-133. PubMed ID: 31878861
    [TBL] [Abstract][Full Text] [Related]  

  • 53. New anti-HIV derivatives: synthesis and antiviral evaluation.
    De Michelis C; Rocheblave L; Priem G; Chermann JC; Kraus JL
    Bioorg Med Chem; 2000 Jun; 8(6):1253-62. PubMed ID: 10896105
    [TBL] [Abstract][Full Text] [Related]  

  • 54. Discovery of HIV-1 integrase inhibitors: pharmacophore mapping, virtual screening, molecular docking, synthesis, and biological evaluation.
    Bhatt H; Patel P; Pannecouque C
    Chem Biol Drug Des; 2014 Feb; 83(2):154-66. PubMed ID: 23957390
    [TBL] [Abstract][Full Text] [Related]  

  • 55. New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase--discovery of a new polyhydroxylated antiviral agent.
    Maurin C; Lion C; Bailly F; Touati N; Vezin H; Mbemba G; Mouscadet JF; Debyser Z; Witvrouw M; Cotelle P
    Bioorg Med Chem; 2010 Jul; 18(14):5194-201. PubMed ID: 20541944
    [TBL] [Abstract][Full Text] [Related]  

  • 56. Beta-diketo acid pharmacophore hypothesis. 1. Discovery of a novel class of HIV-1 integrase inhibitors.
    Dayam R; Sanchez T; Clement O; Shoemaker R; Sei S; Neamati N
    J Med Chem; 2005 Jan; 48(1):111-20. PubMed ID: 15634005
    [TBL] [Abstract][Full Text] [Related]  

  • 57. Pharmacophore-based design of HIV-1 integrase strand-transfer inhibitors.
    Barreca ML; Ferro S; Rao A; De Luca L; Zappalà M; Monforte AM; Debyser Z; Witvrouw M; Chimirri A
    J Med Chem; 2005 Nov; 48(22):7084-8. PubMed ID: 16250669
    [TBL] [Abstract][Full Text] [Related]  

  • 58. Novel inhibitors of HIV integrase: the discovery of potential anti-HIV therapeutic agents.
    Nair V
    Curr Pharm Des; 2003; 9(31):2553-65. PubMed ID: 14529542
    [TBL] [Abstract][Full Text] [Related]  

  • 59. Study on the interactions between diketo-acid inhibitors and prototype foamy virus integrase-DNA complex via molecular docking and comparative molecular dynamics simulation methods.
    Hu JP; He HQ; Tang DY; Sun GF; Zhang YQ; Fan J; Chang S
    J Biomol Struct Dyn; 2013; 31(7):734-47. PubMed ID: 22913375
    [TBL] [Abstract][Full Text] [Related]  

  • 60. The design of 8-hydroxyquinoline tetracyclic lactams as HIV-1 integrase strand transfer inhibitors.
    Velthuisen EJ; Johns BA; Temelkoff DP; Brown KW; Danehower SC
    Eur J Med Chem; 2016 Jul; 117():99-112. PubMed ID: 27092410
    [TBL] [Abstract][Full Text] [Related]  

    [Previous]   [Next]    [New Search]
    of 11.