143 related articles for article (PubMed ID: 30683554)
1. α-Carbonic anhydrases are strongly activated by spinaceamine derivatives.
Akocak S; Lolak N; Bua S; Nocentini A; Karakoc G; Supuran CT
Bioorg Med Chem; 2019 Mar; 27(5):800-804. PubMed ID: 30683554
[TBL] [Abstract][Full Text] [Related]
2. Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives.
Akocak S; Lolak N; Bua S; Nocentini A; Supuran CT
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):1193-1198. PubMed ID: 31237157
[TBL] [Abstract][Full Text] [Related]
3. Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators.
Akocak S; Lolak N; Vullo D; Durgun M; Supuran CT
J Enzyme Inhib Med Chem; 2017 Dec; 32(1):1305-1312. PubMed ID: 29072105
[TBL] [Abstract][Full Text] [Related]
4. Quantum mechanical study on the activation mechanism of human carbonic anhydrase VII cluster model with bis-histamine schiff bases and bis-spinaceamine derivatives.
Ghiasi M; Shahabi P; Supuran CT
Bioorg Med Chem; 2021 Aug; 44():116276. PubMed ID: 34225168
[TBL] [Abstract][Full Text] [Related]
5. Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators.
Angeli A; Chiaramonte N; Manetti D; Romanelli MN; Supuran CT
J Enzyme Inhib Med Chem; 2018 Dec; 33(1):303-308. PubMed ID: 29280407
[TBL] [Abstract][Full Text] [Related]
6. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(arylsulfonylureido-amino acyl)ethyl-1H-imidazole.
Supuran CT; Scozzafava A
J Enzyme Inhib; 2000; 15(5):471-86. PubMed ID: 11030087
[TBL] [Abstract][Full Text] [Related]
7. Carbonic anhydrase activators: synthesis of high affinity isozymes I, II and IV activators, derivatives of 4-(4-tosylureido-amino acyl)ethyl-1H-imidazole (histamine derivatives).
Scozzafava A; Iorga B; Supuran CT
J Enzyme Inhib; 2000; 15(2):139-61. PubMed ID: 10938540
[TBL] [Abstract][Full Text] [Related]
8. Carbonic anhydrases activation with 3-amino-1H-1,2,4-triazole-1-carboxamides: Discovery of subnanomolar isoform II activators.
Le Duc Y; Licsandru E; Vullo D; Barboiu M; Supuran CT
Bioorg Med Chem; 2017 Mar; 25(5):1681-1686. PubMed ID: 28161251
[TBL] [Abstract][Full Text] [Related]
9. Carbonic anhydrase activators. Activation of isozymes I, II, IV, VA, VII, and XIV with l- and d-histidine and crystallographic analysis of their adducts with isoform II: engineering proton-transfer processes within the active site of an enzyme.
Temperini C; Scozzafava A; Vullo D; Supuran CT
Chemistry; 2006 Sep; 12(27):7057-66. PubMed ID: 16807956
[TBL] [Abstract][Full Text] [Related]
10. Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine
Chiaramonte N; Maach S; Biliotti C; Angeli A; Bartolucci G; Braconi L; Dei S; Teodori E; Supuran CT; Romanelli MN
J Enzyme Inhib Med Chem; 2020 Dec; 35(1):1003-1010. PubMed ID: 32336172
[TBL] [Abstract][Full Text] [Related]
11. (Hetero)aryl substituted thiazol-2,4-yl scaffold as human carbonic anhydrase I, II, VII and XIV activators.
Rami M; Winum JY; Supuran CT; Melnyk P; Yous S
J Enzyme Inhib Med Chem; 2019 Dec; 34(1):224-229. PubMed ID: 30734616
[TBL] [Abstract][Full Text] [Related]
12. Carbonic anhydrase inhibitors: synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety.
Sethi KK; Vullo D; Verma SM; Tanç M; Carta F; Supuran CT
Bioorg Med Chem; 2013 Oct; 21(19):5973-82. PubMed ID: 23965175
[TBL] [Abstract][Full Text] [Related]
13. Inhibition of carbonic anhydrase isoforms I, II, IX and XII with novel Schiff bases: identification of selective inhibitors for the tumor-associated isoforms over the cytosolic ones.
Sarikaya B; Ceruso M; Carta F; Supuran CT
Bioorg Med Chem; 2014 Nov; 22(21):5883-90. PubMed ID: 25267005
[TBL] [Abstract][Full Text] [Related]
14. New Histamine-Related Five-Membered N-Heterocycle Derivatives as Carbonic Anhydrase I Activators.
Chiaramonte N; Gabellini A; Angeli A; Bartolucci G; Braconi L; Dei S; Teodori E; Supuran CT; Romanelli MN
Molecules; 2022 Jan; 27(2):. PubMed ID: 35056859
[TBL] [Abstract][Full Text] [Related]
15. Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII.
Sławiński J; Szafrański K; Vullo D; Supuran CT
Eur J Med Chem; 2013 Nov; 69():701-10. PubMed ID: 24095761
[TBL] [Abstract][Full Text] [Related]
16. Activation of carbonic anhydrases from human brain by amino alcohol oxime ethers: towards human carbonic anhydrase VII selective activators.
Nocentini A; Cuffaro D; Ciccone L; Orlandini E; Nencetti S; Nuti E; Rossello A; Supuran CT
J Enzyme Inhib Med Chem; 2021 Dec; 36(1):48-57. PubMed ID: 33103482
[TBL] [Abstract][Full Text] [Related]
17. Carbonic anhydrase activators. Activation of isoforms I, II, IV, VA, VII, and XIV with L- and D-phenylalanine and crystallographic analysis of their adducts with isozyme II: stereospecific recognition within the active site of an enzyme and its consequences for the drug design.
Temperini C; Scozzafava A; Vullo D; Supuran CT
J Med Chem; 2006 May; 49(10):3019-27. PubMed ID: 16686544
[TBL] [Abstract][Full Text] [Related]
18. Carbonic anhydrase activators: design of high affinity isozymes I, II, and IV activators, incorporating tri-/tetrasubstituted-pyridinium-azole moieties.
Ilies M; Banciu MD; Ilies MA; Scozzafava A; Caproiu MT; Supuran CT
J Med Chem; 2002 Jan; 45(2):504-10. PubMed ID: 11784154
[TBL] [Abstract][Full Text] [Related]
19. Pyrazolylbenzo[d]imidazoles as new potent and selective inhibitors of carbonic anhydrase isoforms hCA IX and XII.
Kumar S; Ceruso M; Tuccinardi T; Supuran CT; Sharma PK
Bioorg Med Chem; 2016 Jul; 24(13):2907-2913. PubMed ID: 27166574
[TBL] [Abstract][Full Text] [Related]
20. Synthesis and biological evaluation of novel aromatic and heterocyclic bis-sulfonamide Schiff bases as carbonic anhydrase I, II, VII and IX inhibitors.
Akocak S; Lolak N; Nocentini A; Karakoc G; Tufan A; Supuran CT
Bioorg Med Chem; 2017 Jun; 25(12):3093-3097. PubMed ID: 28400084
[TBL] [Abstract][Full Text] [Related]
[Next] [New Search]